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List of works by Paolo Ruzza

(99m)Tc-radiolabelled peptides for tumour imaging: present and future.

scientific article published on January 2010

4-Fluoroproline derivative peptides: effect on PPII conformation and SH3 affinity

scientific article

A synthetic hexapeptide designed to resemble a proteinaceous P-loop nest is shown to bind inorganic phosphate.

scientific article

Antamanide, a derivative of Amanita phalloides, is a novel inhibitor of the mitochondrial permeability transition pore

scientific article

Assessment of the best N(3-) donors in preparation of [M(N)(PNP)]-based (M=(99m)Tc-; (188)Re) target-specific radiopharmaceuticals: Comparison among succinic dihydrazide (SDH), N-methyl-S-methyl dithiocarbazate (HDTCZ) and PEGylated N-methyl-S-methy

scientific article published on 24 April 2014

Carnosine and carnosine-related antioxidants: a review

scientific article

Ceftriaxone blocks the polymerization of α-synuclein and exerts neuroprotective effects in vitro

scientific article published on 24 October 2013

Cell-Penetrating Peptides: A Comparative Study on Lipid Affinity and Cargo Delivery Properties

scientific article

Conformational constraints of tyrosine in protein tyrosine kinase substrates: Information about preferred bioactive side-chain orientation.

scientific article published in January 2003

Editorial [Hot Topic: Enzymes as Useful Tools and Potential Targets in Cancer Chemotherapy (Guest Editor: P. Ruzza and L. Quintieri)]

scientific article published on 01 September 2009

Effect of 4-fluoro-L-proline on the SH3 binding affinity

scientific article

Flavonoids diosmetin and luteolin inhibit midazolam metabolism by human liver microsomes and recombinant CYP 3A4 and CYP3A5 enzymes.

scientific article

Glutathione Transferase (GST)-Activated Prodrugs.

scientific article published on 02 April 2013

Glutathione transferases as targets for cancer therapy.

scientific article published on September 2009

H-Content Is Not Predictive of Perfluorocarbon Ocular Endotamponade Cytotoxicity in Vitro

scientific article published on 02 August 2019

Hydroxylated biphenyls as tyrosinase inhibitor: A spectrophotometric and electrochemical study.

scientific article published on 13 December 2016

Interactions of GFAP with ceftriaxone and phenytoin: SRCD and molecular docking and dynamic simulation.

scientific article

Introduction of N-alkyl residues in proline-rich peptides: effect on SH3 binding affinity and peptide conformation

scientific article

Ion-binding and pharmacological properties of Tyr6 and Tyr9 antamanide analogs

scientific article published on 01 April 1999

Isolation of a tyrosinase inhibitor from unripe grapes juice: A spectrophotometric study

scientific article published on 10 September 2019

Malondialdehyde scavenging and aldose-derived Schiff bases’ transglycation properties of synthetic histidyl-hydrazide carnosine analogs

scientific article published on 20 June 2007

Melanoma targeting with [99mTc(N)(PNP3)]-labeled α-melanocyte stimulating hormone peptide analogs: Effects of cyclization on the radiopharmaceutical properties.

scientific article published on 31 August 2016

Neuroprotective actions of a histidine analogue in models of ischemic stroke

scientific article

Probing the E/K Peptide Coiled-Coil Assembly by Double Electron-Electron Resonance and Circular Dichroism

scientific article published on 15 December 2020

Radiolabeled peptide-receptor ligands in tumor imaging.

scientific article published on 15 June 2011

Recognition of lysine-rich peptide ligands by murine cortactin SH3 domain: CD, ITC, and NMR studies

scientific article

Separation of acidic peptides by reversed-phase ion-pair chromatography

scientific article published on 01 July 1991

Small molecules interacting with α-synuclein: antiaggregating and cytoprotective properties.

scientific article published on 5 May 2013

Spatial Conformation and Topography of the Tyrosine Aromatic Ring in Substrate Recognition by Protein Tyrosine Kinases†

Specific monitoring of Syk protein kinase activity by peptide substrates including constrained analogs of tyrosine.

scientific article

Specificity of T-cell protein tyrosine phosphatase toward phosphorylated synthetic peptides

scientific article published on 01 January 1993

Spectroscopy data of ceftriaxone-lysozyme interaction and computational studies.

scientific article published on 30 April 2018

Spectroscopy reveals that ethyl esters interact with proteins in wine.

scientific article published on 2 September 2016

Synthesis and Studies of the Inhibitory Effect of Hydroxylated Phenylpropanoids and Biphenols Derivatives on Tyrosinase and Laccase Enzymes

scientific article published on 11 June 2020

Synthesis and preliminary in vitro biological evaluation of 4-[(4-hydroxyphenyl)sulfanyl]but-3-en-2-one, a 4-mercaptophenol derivative designed as a novel bifunctional antimelanoma agent.

scientific article published in August 2009

Synthetic peptide substrates for casein kinase 2. Assessment of minimum structural requirements for phosphorylation

scientific article published on 01 October 1988

Synthetic peptides reproducing the EGF-receptor segment homologous to the pp60v-src phosphoacceptor site. Phosphorylation by tyrosine protein kinases

scientific article published on 01 July 1989

Tat cell-penetrating peptide has the characteristics of a poly(proline) II helix in aqueous solution and in SDS micelles.

scientific article

The SH3 domain of HS1 protein recognizes lysine-rich polyproline motifs

scientific article

The Secondary Structure of a Major Wine Protein is Modified upon Interaction with Polyphenols

scientific article published on 03 April 2020

The impact of either 4-R-hydroxyproline or 4-R-fluoroproline on the conformation and SH3m-cort binding of HPK1 proline-rich peptide

scientific article published on 14 September 2012