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List of works by Harald Hübner

Analogues of FAUC 73 revealing new insights into the structural requirements of nonaromatic dopamine D3 receptor agonists

scientific article published in January 2004

CoMFA and CoMSIA investigations of dopamine D3 receptor ligands leading to the prediction, synthesis, and evaluation of rigidized FAUC 365 analogues

scholarly article by Ismail Salama et al published September 2006 in Bioorganic & Medicinal Chemistry

CoMFA and CoMSIA investigations revealing novel insights into the binding modes of dopamine D3 receptor agonists

scientific article published in April 2005

FAUC 213, a highly selective dopamine D4 receptor full antagonist, exhibits atypical antipsychotic properties in behavioural and neurochemical models of schizophrenia

scientific article published on 6 March 2004

Fancy bioisosteres: metallocene-derived G-protein-coupled receptor ligands with subnanomolar binding affinity and novel selectivity profiles

scientific article published in June 2005

Fancy bioisosteres: novel paracyclophane derivatives as super-affinity dopamine D3 receptor antagonists

scientific article published in June 2006

Fancy bioisosteres: synthesis and dopaminergic properties of the endiyne FAUC 88 as a novel non-aromatic D3 agonist

scientific article published in January 2005

Fancy bioisosteres: synthesis, SAR, and pharmacological investigations of novel nonaromatic dopamine D3 receptor ligands

scientific article published in July 2005

Pharmacophore-guided drug discovery investigations leading to bioactive 5-aminotetrahydropyrazolopyridines. Implications for the binding mode of heterocyclic dopamine D3 receptor agonists

scientific article published in September 2005

Structure-based development of a subtype-selective orexin 1 receptor antagonist

scientific article published on 15 July 2020

Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands

scientific article

Visualization of β-adrenergic receptor dynamics and differential localization in cardiomyocytes

scientific article published in 2021