Search filters

List of works by Lauren T May

Allosteric modulation of endogenous metabolites as an avenue for drug discovery.

scientific article published on 10 May 2012

Allosteric modulators of G-protein-coupled receptors

scientific article published on October 1, 2003

Correspondence: Reply to 'Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury'.

scientific article published on 7 February 2018

Extracellular Loop 2 of the Adenosine A1 Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy.

scientific article published on 28 September 2016

GraphormerDTI: A graph transformer-based approach for drug-target interaction prediction

scientific article published in 2024

New Paradigms in Adenosine Receptor Pharmacology: Allostery, Oligomerization and Biased Agonism

scientific article published on 21 April 2018

Novel Irreversible Agonists Acting at the A1 Adenosine Receptor

scientific article

Positive allosteric mechanisms of adenosine A<sub>1</sub> receptor-mediated analgesia

scientific article published on 08 September 2021

Quantification of adenosine A(1) receptor biased agonism: Implications for drug discovery

scientific article published on 12 November 2015

Role of the Second Extracellular Loop of the Adenosine A1 Receptor on Allosteric Modulator Binding, Signaling, and Cooperativity.

scientific article published on 28 September 2016

Separation of on-target efficacy from adverse effects through rational design of a bitopic adenosine receptor agonist

scientific article published on 11 March 2014

Small-molecule-biased formyl peptide receptor agonist compound 17b protects against myocardial ischaemia-reperfusion injury in mice.

scientific article published on 07 February 2017

Structure of the Adenosine A1 Receptor Reveals the Basis for Subtype Selectivity

scientific article published in February 2017

Structure of the adenosine-bound human adenosine A1 receptor–Gi complex

scientific article published in Nature

Structure-function studies of allosteric agonism at M2 muscarinic acetylcholine receptors

scientific article published on 24 May 2007

The apelin receptor inhibits the angiotensin II type 1 receptor via allosteric trans‐inhibition

scientific article published on March 1, 2013