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List of works by Daniele Bolognini

A Novel Allosteric Activator of Free Fatty Acid 2 Receptor Displays Unique Gi-functional Bias

scientific article published on 05 July 2016

A single extracellular amino acid in Free Fatty Acid Receptor 2 defines antagonist species selectivity and G protein selection bias

scientific article

AM630 behaves as a protean ligand at the human cannabinoid CB2 receptor.

scientific article

CB(1) receptor allosteric modulators display both agonist and signaling pathway specificity.

scientific article published on 15 November 2012

CB2 cannabinoid receptor agonist enantiomers HU-433 and HU-308: An inverse relationship between binding affinity and biological potency

scientific article published on 29 June 2015

Cannabidiol, a non-psychoactive cannabinoid compound, inhibits proliferation and invasion in U87-MG and T98G glioma cells through a multitarget effect

scientific article (publication date: 2013)

Chemogenetics defines receptor-mediated functions of short chain free fatty acids

scientific article published on 15 April 2019

Discovery of a Potent Thiazolidine Free Fatty Acid Receptor 2 Agonist with Favorable Pharmacokinetic Properties

scientific article published on 12 October 2018

Expression and function of the endocannabinoid system in glial cells

scientific article published on January 2008

In vitro and in vivo pharmacological characterization of two novel selective cannabinoid CB(2) receptor inverse agonists

scientific article published on 2 December 2009

Investigations on the 4-quinolone-3-carboxylic acid motif part 5: modulation of the physicochemical profile of a set of potent and selective cannabinoid-2 receptor ligands through a bioisosteric approach.

scientific article

Investigations on the 4-quinolone-3-carboxylic acid motif. 3. Synthesis, structure-affinity relationships, and pharmacological characterization of 6-substituted 4-quinolone-3-carboxamides as highly selective cannabinoid-2 receptor ligands

scientific article

Investigations on the 4-quinolone-3-carboxylic acid motif. 6. Synthesis and pharmacological evaluation of 7-substituted quinolone-3-carboxamide derivatives as high affinity ligands for cannabinoid receptors

scientific article

Ligands at the Free Fatty Acid Receptors 2/3 (GPR43/GPR41).

scientific article published on 19 October 2016

Metabolic and inflammatory functions of short-chain fatty acid receptors

scientific article published on 03 July 2020

On-target and off-target effects of novel orthosteric and allosteric activators of GPR84

scientific article published in Scientific Reports

Structural and pharmacological analysis of O-2050, a putative neutral cannabinoid CB(1) receptor antagonist.

scientific article

The Pharmacology and Function of Receptors for Short-Chain Fatty Acids.

scientific article published on 30 December 2015

The plant cannabinoid Delta9-tetrahydrocannabivarin can decrease signs of inflammation and inflammatory pain in mice

scientific article

Treatment of Active Crohn’s Disease With an Ordinary Food-based Diet That Replicates Exclusive Enteral Nutrition

scientific article published on 11 December 2018

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