Search filters

Authors whose works are in public domain in at least one jurisdiction

List of works by Gavril W. Pasternak

1-Aminocyclopropane carboxylic acid (ACPC) prevents mu and delta opioid tolerance

scientific article

3H-naloxone benzoylhydrazone binding in MOR-1-transfected Chinese hamster ovary cells: evidence for G-protein-dependent antagonist binding ⬇️

scientific article published on July 1, 1998

A heroin addiction severity-associated intronic single nucleotide polymorphism modulates alternative pre-mRNA splicing of the μ opioid receptor gene OPRM1 via hnRNPH interactions

scientific article

Affinity labeling of mu and kappa receptors with naloxone benzoylhydrazone ⬇️

scientific article published on March 1, 1991

An all D-amino acid opioid peptide with central analgesic activity from a combinatorial library

scientific article published on December 1994

An endogenous morphine-like factor in mammalian brain ⬇️

scientific article published on June 15, 1975

Analgesic activity of tricyclic antidepressants

scientific article published on 01 April 1983

Analgesic potency of TRIMU-5: a mixed mu 2 opioid receptor agonist/mu 1 opioid receptor antagonist

scientific article published on June 5, 1992

Analgesic synergy between topical lidocaine and topical opioids

scientific article published in November 2000

Antagonism of morphine analgesia by intracerebroventricular naloxonazine

scientific article published in June 1986

Antagonist effects of beta-funaltrexamine and naloxonazine on alfentanil-induced antinociception and muscle rigidity in the rat.

scientific article published in February 1993

Antisense mapping DOR-1 in mice: further support for delta receptor subtypes

scientific article

Antisense mapping KOR-1: evidence for multiple kappa analgesic mechanisms

scientific article published in May 1999

Antisense mapping of the MOR-1 opioid receptor clone: modulation of hyperphagia induced by DAMGO ⬇️

scientific article published on September 1, 1997

Antisense oligodeoxynucleotides against the MOR-1 clone alter weight and ingestive responses in rats

scientific article published in May 1996

Autoradiography of [3H]β-endorphin binding in brain ⬇️

scientific article published on December 12, 1983

Beta-endorphin-induced feeding: pharmacological characterization using selective opioid antagonists and antisense probes in rats.

scientific article published in May 2001

Binding of 3H-β-endorphin in rat brain ⬇️

scientific article published on September 20, 1982

Binding of [3H]naloxonazine to rat brain membranes ⬇️

scientific article published on November 1, 1984

Biochemical and pharmacological characterization of mu, delta and kappa 3 opioid receptors expressed in BE(2)-C neuroblastoma cells

scientific article published on September 1994

Biochemical and pharmacological evidence for opioid receptor multiplicity in the central nervous system

scientific article published on January 1983

Biochemical characterization of high-affinity 3H-opioid binding. Further evidence for Mu1 sites ⬇️

scientific article published on January 1, 1984

Blockade of U50,488H analgesia by antisense oligodeoxynucleotides to a kappa-opioid receptor

scientific article published on March 1994

Blockade of morphine analgesia by an antisense oligodeoxynucleotide against the mu receptor

scientific article published in January 1994

Blockade of morphine-induced hindlimb myoclonic seizures in mice by ketamine

scientific article published on March 1997

Blockade of mu and kappa 1 opioid analgesic tolerance by NPC17742, a novel NMDA antagonist

scientific article

Brain and caudate nucleus adenylate cyclase: Effects of dopamine, GTP, E prostaglandins and morphine ⬇️

scientific article published on March 1, 1975

Central mechanisms of opioid analgesia

scientific article published on January 1981

Characterization of an endogenous morphine-like factor(enkephalin) in mammalian brain ⬇️

scientific article published on May 1, 1976

Characterization of the opioid receptor binding and animal pharmacology of meptazinol

scientific article published in January 1985

Characterizing kappa3 opioid receptors with a selective monoclonal antibody

scientific article published on March 1996

Cloning and functional characterization through antisense mapping of a kappa 3-related opioid receptor ⬇️

scientific article published on June 1, 1995

Comparison of effects of chronic administration of naloxone and naloxonazine upon food intake and maintainance of body weight in rats ⬇️

scientific article published on April 1, 1988

Comparison of naloxonazine and β-funaltrexamine antagonism of μ1 and μ2 opioid actions ⬇️

scientific article published on January 1, 1991

Correction to: Mu Opioids Induce Biased Signaling at the Full-Length Seven Transmembrane C-Terminal Splice Variants of the mu Opioid Receptor Gene, Oprm1

scientific article published on 31 October 2020

Correlating the pharmacology and molecular biology of opioid receptors. Cloning and antisense mapping a kappa 3-related opiate receptor

scientific article

Demonstration of kappa 3-opioid receptors in the SH-SY5Y human neuroblastoma cell line

scientific article

Developmental differences between high and low affinity opiate binding sites: Their relationship to analgesia and respiratory depression ⬇️

scientific article published on September 29, 1980

Differential blockade of opioid analgesia by antisense oligodeoxynucleotides directed against various G protein alpha subunits

scientific article

Differential effects of protein-modifying reagents on receptor binding of opiate agonists and antagonists ⬇️

scientific article published on May 1, 1975

Differentiation of opiate agonist and antagonist receptor binding by protein modifying reagents ⬇️

scientific article published on February 6, 1975

Discrimination by temperature of opiate agonist and antagonist receptor binding ⬇️

scientific article published on June 15, 1975

Effects of beta-funaltrexamine on radiolabeled opioid binding

scientific article

Endogenous opioid systems in brain ⬇️

scientific article published on February 1, 1980

Functional antagonism of morphine analgesia by (+)-pentazocine: evidence for an anti-opioid sigma 1 system

scientific article

Gender effects and central opioid analgesia ⬇️

scientific article published on April 1, 1991

High and low affinity opioid binding sites: Relationship to mu and delta sites ⬇️

scientific article published on September 20, 1982

Hydrocephalic dementia and spinal cord tumor. Report of a case and review of the literature

scientific article published on July 1986

Identification of novel high affinity opiate receptor binding in rat brain ⬇️

scientific article published on February 13, 1975

Immunohistochemical localization of the carboxy terminus of the novel mu opioid receptor splice variant MOR-1C within the human spinal cord

scientific article published in June 2000

Incomplete cross tolerance and multiple mu opioid peptide receptors

scientific article

Increased analgesic potency of morphine and increased brain opioid binding sites in the rat following chronic naltrexone treatment

scientific article

Independent expression of two pharmacologically distinct supraspinal mu analgesic systems in genetically different mouse strains

scientific article published in April 1993

Individual variability in the response to different opioids: report of five cases

scientific article published on April 1, 1992

Interaction of [D-Ser2,Leu5]enkephalin-Thr6 (DSLET), a relatively selective delta ligand, with mu1 opioid binding sites

scientific article published in January 1987

Interaction of two phencyclidine opiate-like derivatives with 3H-opioid binding sites

scientific article

Interactions of chloroquine with benzodiazepine, γ-aminobutyric acid and opiate receptors ⬇️

scientific article published on May 15, 1991

Involvement of opioid receptor subtypes in rat feeding behavior

scientific article

Irreversible opiate agonists and antagonists. II. Evidence against a bivalent mechanism of action for opiate azines and diacylhydrazones

scientific article published on 01 December 1985

Irreversible opiate agonists and antagonists. III. Phenylhydrazone derivatives of naloxone and oxymorphone.

scientific article published in December 1985

Irreversible opiate agonists and antagonists. IV. Analgesic actions of 14-hydroxydihydromorphinone hydrazones

scientific article (publication date: April 1988)

Irreversible opiate agonists and antagonists: V. Hydrazone and acylhydrazone derivatives of naltrexone

scientific article

Kappa 3 opiate receptor binding in the mouse and rat

scientific article published on May 12, 1992

Kappa 3 receptors and levorphanol-induced analgesia

scientific article published on September 1, 1992

Kappa opiate receptor multiplicity: evidence for two U50,488-sensitive kappa 1 subtypes and a novel kappa 3 subtype.

scientific article

Kappa-opiate binding to rat brain and guinea pig cerebellum: sensitivity towards ions and nucleotides

scientific article published in February 1986

Lack of morphine and enkephalin tolerance in 129/SvEv mice: evidence for a NMDA receptor defect ⬇️

scientific article published on 01 February 1998

Loss of striatal mu1 opiate binding by substantia nigra lesions in the rat.

scientific article

Mapping of opioid receptors using antisense oligodeoxynucleotides: correlating their molecular biology and pharmacology

scientific article published on October 1995

Mediation of anorexia by human recombinant tumor necrosis factor through a peripheral action in the rat

scientific article published on 01 November 1989

Meptazinol: a novel Mu-1 selective opioid analgesic ⬇️

scientific article published on February 1, 1984

Mercaptoacetate induces feeding through central opioid-mediated mechanisms in rats

scientific article published in May 2000

Methadone analgesia in morphine-insensitive CXBK mice ⬇️

scientific article published on June 19, 1998

Metkephamid (Tyr-D-Ala-Gly-Phe-N(Me)Met-NH2), a potent opioid peptide: Receptor binding and analgesic properties ⬇️

scientific article published on September 1, 1982

Modulation of Mu1 opioid binding by magnesium: evidence for multiple receptor conformations

scientific article

Modulation of morphine tolerance by the competitive N-methyl-D-aspartate receptor antagonist LY274614: assessment of opioid receptor changes

scientific article

Modulation of mu 1, mu 2, and delta opioid binding by divalent cations

scientific article

Modulation of opioid analgesia by agmatine

scientific article

Molecular cloning and pharmacological characterization of the rat sigma1 receptor

scientific article published in August 2001

Mu 1 opioid receptor involvement in maternal behavior

scientific article

Mu Opioids Induce Biased Signaling at the Full-Length Seven Transmembrane C-Terminal Splice Variants of the mu Opioid Receptor Gene, Oprm1

scientific article published on 08 October 2020

Mu and delta opioid synergy between the periaqueductal gray and the rostro-ventral medulla

scientific article

Multiple morphine and enkephalin receptors: biochemical and pharmacological aspects

scientific article

Multiple mu opiate receptors

scientific article

Multiple mu receptors: evidence for mu2 sites in the guinea pig ileum ⬇️

scientific article published on August 19, 1983

Nalbuphine, a mixed kappa 1 and kappa 3 analgesic in mice ⬇️

scientific article published on 01 September 1992

Naloxazone, a long-acting opiate antagonist: effects on analgesia in intact animals and on opiate receptor binding in vitro ⬇️

scientific article published on 01 September 1980

Naloxonazine actions in vivo

scientific article

Naloxonazine, a potent, long-lasting inhibitor of opiate binding sites ⬇️

scientific article published on September 20, 1982

Naloxone benzoylhydrazone (NalBzoH) analgesia

scientific article published on 01 November 1990

Naloxone benzoylhydrazone, a kappa 3 opioid agonist, stimulates food intake in rats

scientific article published on May 29, 1992

Naloxozone pretreatment modifies cardiorespiratory, temperature, and behavioral effects of morphine ⬇️

scientific article published on June 16, 1983

Nitric oxide and opioid tolerance.

scientific article

Ontogeny of opioid pharmacology and receptors: High and low affinity site differences ⬇️

scientific article published on July 17, 1981

Opiate Analgesia: Evidence for Mediation by a Subpopulation of Opiate Receptors ⬇️

scientific article published on May 2, 1980

Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity ⬇️

scientific article published on September 23, 1982

Opiate binding in calf thalamic membranes: a selective mu 1 binding assay

scientific article

Opiate receptor binding: effects of enzymatic treatments

scientific article

Opiate receptor multiplicity: evidence for multiple mu receptors

scientific article published on January 1987

Opiates, opioid peptides, and their receptors

scientific article published on December 1987

Opioid binding in giant toad and goldfish brain.

scientific article

Oxymorphazone: A long-acting opiate analgesic ⬇️

scientific article published on March 1, 1984

Oxymorphone-naltrexonazine, a mixed opiate agonist-antagonist

scientific article

Peripheral blockade of topical morphine tolerance by ketamine

scientific article published in June 1999

Peripheral kappa 1-opioid receptor-mediated analgesia in mice

scientific article

Pharmacodynamic supersensitivity and opioid receptor upregulation in the mouse

scientific article published in October 1986

Pharmacological actions of a novel mixed opiate agonist/antagonist: naloxone benzoylhydrazone

scientific article published in November 1989

Pharmacological characterization of morphine-6-sulfate and codeine-6-sulfate

scientific article published in September 1999

Pharmacological characterization of nalorphine, a kappa 3 analgesic ⬇️

scientific article published on 01 April 1991

Phenylmorphans and analogs: opioid receptor subtype selectivity and effect of conformation on activity ⬇️

scientific article published on May 1, 1992

Potentiation of opioid analgesia by the antidepressant nefazodone

scientific article published on February 18, 1992

Presynaptic localization of the carboxy-terminus epitopes of the μ opioid receptor splice variants MOR-1C and MOR-1D in the superficial laminae of the rat spinal cord ⬇️

scientific article published on January 1, 2001

Proglumide selectively potentiates supraspinal mu 1 opioid analgesia in mice

scientific article

Receptor binding of [3H]naloxone benzoylhydrazone: a reversible kappa and slowly dissociable mu opiate.

scientific article published in January 1989

Reductions in body weight following chronic central opioid receptor subtype antagonists during development of dietary obesity in rats

scientific article

Regional differences in mu 1-binding of [3H][D-Ala2,D-Leu5]-enkephalin: comparisons of thalamus and cortex in the rat.

scientific article published in August 1985

Retention of supraspinal delta-like analgesia and loss of morphine tolerance in delta opioid receptor knockout mice

scientific article published in September 1999

Role of mu 1-opiate receptors in supraspinal opiate analgesia: a microinjection study

scientific article published in April 1988

Selective antagonism of opioid analgesia by a sigma system

scientific article

Selective enhancement of [3H]opiate agonist binding by divalent cations ⬇️

scientific article published on November 1, 1975

Selective loss of delta opioid analgesia and binding by antisense oligodeoxynucleotides to a delta opioid receptor

scientific article published on April 1994

Separation of opioid analgesia from respiratory depression: evidence for different receptor mechanisms

scientific article

Sigma antagonists potentiate opioid analgesia in rats ⬇️

scientific article published on May 5, 1995

Spinal and supraspinal opioid analgesia in the mouse: the role of subpopulations of opioid binding sites ⬇️

scientific article published on July 18, 1983

Structure and characterization of the gene encoding a mouse kappa3-related opioid receptor

scientific article published on June 1996

Supraspinal mu 2-opioid receptors mediate spinal/supraspinal morphine synergy

scientific article published on September 22, 1992

Synergistic analgesic interactions between the periaqueductal gray and the locus coeruleus

scientific article

Synthesis and Characterization of Azido Aryl Analogs of IBNtxA for Radio-Photoaffinity Labeling Opioid Receptors in Cell Lines and in Mouse Brain

scientific article published on 18 May 2020

The NMDA receptor antagonists, LY274614 and MK-801, and the nitric oxide synthase inhibitor, NG-nitro-L-arginine, attenuate analgesic tolerance to the mu-opioid morphine but not to kappa opioids

scientific article published in January 1994

The binding and analgesic properties of a sigma opiate, SKF 10,047 ⬇️

scientific article published on 01 October 1981

The binding to rat brain homogenates of Mr2034, a universal opiate ⬇️

scientific article published on September 5, 1983

The central questions in pain perception may be peripheral ⬇️

scientific article published on September 1, 1998

The effects of cell isolation techniques on neuronal membrane receptors ⬇️

scientific article published on August 8, 1975

Transport of opioids from the brain to the periphery by P-glycoprotein: peripheral actions of central drugs

scientific article

U50,488: a kappa-selective agent with poor affinity for mu1 opiate binding sites

scientific article published in March 1988

Upregulation of opioid receptor subtypes correlates with potency changes of morphine and DADLE.

scientific article

Visualization of mu1 opiate receptors in rat brain by using a computerized autoradiographic subtraction technique

scientific article published on October 1985

X-ray crystal structure of the opioid ligand naltrexonazine

scientific article published in August 1987

[D-Pen2,D-Pen5]enkephalin (DPDPE): a delta-selective enkephalin with low affinity for mu 1 opiate binding sites

scientific article

σ Receptor ligand binding: an open-and-shut case

scientific article published on 01 November 2018

Paulina is supported by:

About Paulina

Help