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List of works by Józef Oleksyszyn

3,4-dimethoxybenzyl isothiocyanate enhances doxorubicin efficacy in LoVoDX doxorubicin-resistant colon cancer and attenuates its toxicity in vivo

scientific article published on 04 June 2019

Adjuvant-dependent immunogenicity of Staphylococcus aureus Efb and Map proteins in chickens.

scientific article published on 16 May 2015

Application of specific cell permeable cathepsin G inhibitors resulted in reduced antigen processing in primary dendritic cells.

scientific article published on 16 July 2009

Comparision of the cytotoxic effects of birch bark extract, betulin and betulinic acid towards human gastric carcinoma and pancreatic carcinoma drug-sensitive and drug-resistant cell lines.

scientific article published on 24 April 2009

Cover Picture: Phosphonic Analogs of Alanine as Acylpeptide Hydrolase Inhibitors (Chem. Biodiversity 2/2021)

scientific article published in 2021

Design, Synthesis, and Evaluation of ω-(Isothiocyanato)alkylphosphinates and Phosphine Oxides as Antiproliferative Agents

scientific article published on 24 November 2017

Development and Evaluation of an Immunoglobulin Y-Based ELISA for Measuring Prostate Specific Antigen in Human Serum

scientific article published on 01 July 2019

Development and binding characteristics of phosphonate inhibitors of SplA protease from Staphylococcus aureus

scientific article

Development of Adenosine Deaminase-Specific IgY Antibodies: Diagnostic and Inhibitory Application

scientific article published on 17 October 2017

First synthesis of alpha-aminoalkyl-(N-substituted)thiocarbamoyl-phosphinates: inhibitors of aminopeptidase N (APN/CD13) with the new zinc-binding group

scientific article published on 17 May 2008

Generation and application of polyclonal IgY antibodies specific for full-length and nicked prostate-specific antigen

scientific article published on 01 January 2014

Highly sensitive detection of cancer antigen 15-3 using novel avian IgY antibodies.

scientific article published on 19 November 2013

Human neutrophil elastase phosphonic inhibitors with improved potency of action

scientific article published on 12 July 2012

Identification of a serine protease inhibitor which causes inclusion vacuole reduction and is lethal to Chlamydia trachomatis.

scientific article published on 12 July 2013

Identification of very potent inhibitor of human aminopeptidase N (CD13)

scientific article published on 04 March 2010

Inhibition of trypsin and urokinase by Cbz-amino(4-guanidinophenyl)methanephosphonate aromatic ester derivatives: the influence of the ester group on their biological activity

scientific article published on 20 March 2006

Invariant chain processing is independent of cathepsin variation between primary human B cells/dendritic cells and B-lymphoblastoid cells ⬇️

scientific article published on March 17, 2011

Method for generation of peptide-specific IgY antibodies directed to Staphylococcus aureus extracellular fibrinogen binding protein epitope.

scientific article published on 11 June 2015

New aromatic monoesters of alpha-aminoaralkylphosphonic acids as inhibitors of aminopeptidase N/CD13.

scientific article published on March 2010

New potent cathepsin G phosphonate inhibitors

scientific article published on 31 August 2008

Novel diphenyl esters of peptidyl alpha-aminoalkylphosphonates as inhibitors of chymotrypsin and subtilisin

scientific article published in December 2009

Novel hydroxamic acid-related phosphinates: inhibition of neutral aminopeptidase N (APN)

scientific article published on 19 January 2007

Novel peptidyl α-aminoalkylphosphonates as inhibitors of hepatitis C virus NS3/4A protease.

scientific article published on 30 June 2017

Novel phosphonate analogs of sulforaphane: Synthesis, in vitro and in vivo anticancer activity.

scientific article

Phosphonate inhibitors of West Nile virus NS2B/NS3 protease

scientific article published on 01 December 2019

Phosphonic Analogs of Alanine as Acylpeptide Hydrolase Inhibitors

scientific article published in 2021

Phosphonic analogues of glutamic acid as irreversible inhibitors of Staphylococcus aureus endoproteinase GluC: An efficient synthesis and inhibition of the human IgG degradation ⬇️

scientific article published on January 5, 2013

Phosphonic pseudopeptides as human neutrophil elastase inhibitors--a combinatorial approach

scientific article

Phosphorus-containing isothiocyanate-derived mercapturic acids as a useful alternative for parental isothiocyanates in experimental oncology

scientific article published on 20 June 2018

Simple phosphonic inhibitors of human neutrophil elastase.

scientific article published on 22 January 2011

Structure-based design, synthesis, and evaluation of the biological activity of novel phosphoroorganic small molecule IAP antagonists

scientific article published on 08 April 2020

Substrate profiling of Finegoldia magna SufA protease, inhibitor screening and application to prevent human fibrinogen degradation and bacteria growth in vitro.

scientific article

Synthesis and antiproliferative activity of novel α- and β-dialkoxyphosphoryl isothiocyanates.

scientific article published on 6 June 2011

Synthesis and biological activity of diisothiocyanate-derived mercapturic acids.

scientific article published on 27 November 2015

The complete control of glucose level utilizing the composition of ketogenic diet with the gluconeogenesis inhibitor, the anti-diabetic drug metformin, as a potential anti-cancer therapy ⬇️

scientific article published on 06 May 2011

The molecular basis of urokinase inhibition: from the nonempirical analysis of intermolecular interactions to the prediction of binding affinity

scientific article published on 20 March 2007

Viability of glioblastoma stem cells is effectively reduced by diisothiocyanate-derived mercapturic acids

scientific article published on 21 August 2018

Was the serine protease cathepsin G discovered by S. G. Hedin in 1903 in bovine spleen?

scientific article published on 07 March 2011

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