List of works - Bogdan Musielak

A Unique Mdm2-Binding Mode of the 3-Pyrrolin-2-one- and 2-Furanone-Based Antagonists of the p53-Mdm2 Interaction

scientific article

A concerted evolution of supramolecular interactions in a {cation; metal complex; π-acid; solvent} anion-π system

scientific article published in 2020

Application of bioorthogonal hetero-Diels–Alder cycloaddition of 5-arylidene derivatives of 1,3-dimethylbarbituric acid and vinyl thioether for imaging inside living cells

scientific article published in 2021

Application of dimedone enamines as dienophiles: stereoselective synthesis of amino enols of fused uracils containing a sugar moiety by hetero-Diels–Alder reactions of barbituric acid 5-ylidene alditols with dimedone enamines

scientific article published in November 2015

Application of pyrrolo[2,3-b]quinoxaline with an N,N-bis(pyridin-2-ylmethyl)ethylenediamine chain for Zn(II) detection in Candida albicans and fibroblast cells

scientific article published in September 2019

Artificial Macrocycles as Potent p53-MDM2 Inhibitors.

scientific article published on 20 September 2017

Bioactive Macrocyclic Inhibitors of the PD-1/PD-L1 Immune Checkpoint.

scientific article

CA-170 - A Potent Small-Molecule PD-L1 Inhibitor or Not?

scientific article published on 01 August 2019

CA-170 – a potent small-molecule PD-L1 inhibitor or not?

scientific article published on 6 June 2019

Chelate Ring Size Effect as a Factor of Selective Fluorescent Recognition of Zn(2+) Ions by Pyrrolo[2,3-b]quinoxaline with a Substituted 2-Pyridyl Group Receptor

scientific article published on 20 August 2015

Clinical applications of artificial intelligence in cardiology on the verge of the decade

scientific article published on 10 July 2020

Cobalt(II), copper(II), and zinc(II) isostructural, pseudotetrahedral, racemic complexes of pyrrolo[2,3-b]quinoxaline with bis(2-thienylmethyl)propylenediamine chain: Synthesis, crystal structure, spectroscopy

scientific article published in February 2019

Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions

scientific article published on 01 July 2020

Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions

scientific article published on 13 June 2020

Composite Nitride Nanoceramics in the System Titanium Nitride (TiN)-Aluminum Nitride (AlN) through High Pressure and High Temperature Sintering of Synthesis-Mixed Nanocrystalline Powders

scientific article published on 27 January 2021

Conformation of Eight-Membered Benzoannulated Lactams by Combined NMR and DFT Studies ⬇️

scientific article published on October 24, 2012

Conformations and Conformational Processes of Hexahydrobenzazocines by NMR and DFT Studies

scientific article published on 28 August 2015

Crystal structure of the FAS1 domain of the hyaluronic acid receptor stabilin-2

scientific article published on 27 June 2018

Design, Synthesis, Evaluation, and Structural Studies of C2-Symmetric Small Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction

scientific article published on 25 July 2019

Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists

scientific article published on 28 April 2021

Di-Bromo-based small-molecule inhibitors of the PD-1/PD-L1 immune checkpoint

scientific article published on 16 September 2020

Human and mouse PD-L1: similar molecular structure, but different druggability profiles

scientific article published on 22 January 2021

Identification of small-molecule inhibitors of USP2a

scientific article published on 5 March 2018

Macrocyclic Peptide Inhibitor of PD‐1/PD‐L1 Immune Checkpoint

scientific article published on 18 November 2020

Mechanism of MyD88S mediated signal termination

scientific article published on 20 January 2022

Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

scientific article published on 12 December 2019

PD-L1 Inhibitors: Different Classes, Activities, and Mechanisms of Action

scientific article published on 30 October 2021

Rational design and synthesis of 1,5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction.

scientific article published on 16 November 2016

Small-Molecule Inhibitors of the Programmed Cell Death-1/Programmed Death-Ligand 1 (PD-1/PD-L1) Interaction via Transiently Induced Protein States and Dimerization of PD-L1.

scientific article published on 14 June 2017

Small-molecule inhibitors of PD-1/PD-L1 immune checkpoint alleviate the PD-L1-induced exhaustion of T-cells.

scientific article published on 7 August 2017

Structural Characterization of a Macrocyclic Peptide Modulator of the PD-1/PD-L1 Immune Checkpoint Axis

scientific article published on 11 August 2021

Structural basis for small molecule targeting of the programmed death ligand 1 (PD-L1)

scientific article (publication date: 24 May 2016)

Structure of the Complex of Human Programmed Death 1, PD-1, and Its Ligand PD-L1.

scientific article published on 22 October 2015

Synthesis of the New Heterocyclic System 5,6,10b-Triazaacephenanthrylene, a Nitrogen Analogue of Aristolactams

scientific article published in 2016

Synthesis, structure, and photophysical properties of luminescent zinc and cadmium complexes containing 2-pyridyl-substituted pyrrolo[2,3- b ]quinoxaline

scientific article published in September 2017

Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction

scientific article published on 12 August 2021

Terphenyl-based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein−Protein Interaction

scientific article published on 11 February 2021

Terphenyl-based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein−Protein Interaction

scientific article

The neutralization of heparan sulfate by heparin-binding copolymer as a potential therapeutic target

scientific article published on 22 January 2019

The synthesis and characterization of tetramic acid derivatives as Mdm2-p53 inhibitors

scientific article published in August 2019

Two-Step Synthesis of Complex Artificial Macrocyclic Compounds

scientific article

π-π-Induced aggregation and single-crystal fluorescence anisotropy of 5,6,10b-tri-aza-acephenanthrylene.

scientific article

List of works by Bogdan Musielak

A Unique Mdm2-Binding Mode of the 3-Pyrrolin-2-one- and 2-Furanone-Based Antagonists of the p53-Mdm2 Interaction

A concerted evolution of supramolecular interactions in a {cation; metal complex; π-acid; solvent} anion-π system

Application of bioorthogonal hetero-Diels–Alder cycloaddition of 5-arylidene derivatives of 1,3-dimethylbarbituric acid and vinyl thioether for imaging inside living cells

Application of dimedone enamines as dienophiles: stereoselective synthesis of amino enols of fused uracils containing a sugar moiety by hetero-Diels–Alder reactions of barbituric acid 5-ylidene alditols with dimedone enamines

Application of pyrrolo[2,3-b]quinoxaline with an N,N-bis(pyridin-2-ylmethyl)ethylenediamine chain for Zn(II) detection in Candida albicans and fibroblast cells

Artificial Macrocycles as Potent p53-MDM2 Inhibitors.

Bioactive Macrocyclic Inhibitors of the PD-1/PD-L1 Immune Checkpoint.

CA-170 - A Potent Small-Molecule PD-L1 Inhibitor or Not?

CA-170 – a potent small-molecule PD-L1 inhibitor or not?

Chelate Ring Size Effect as a Factor of Selective Fluorescent Recognition of Zn(2+) Ions by Pyrrolo[2,3-b]quinoxaline with a Substituted 2-Pyridyl Group Receptor

Clinical applications of artificial intelligence in cardiology on the verge of the decade

Cobalt(II), copper(II), and zinc(II) isostructural, pseudotetrahedral, racemic complexes of pyrrolo[2,3-b]quinoxaline with bis(2-thienylmethyl)propylenediamine chain: Synthesis, crystal structure, spectroscopy

Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions

Competition NMR for Detection of Hit/Lead Inhibitors of Protein-Protein Interactions

Composite Nitride Nanoceramics in the System Titanium Nitride (TiN)-Aluminum Nitride (AlN) through High Pressure and High Temperature Sintering of Synthesis-Mixed Nanocrystalline Powders

Conformation of Eight-Membered Benzoannulated Lactams by Combined NMR and DFT Studies ⬇️

Conformations and Conformational Processes of Hexahydrobenzazocines by NMR and DFT Studies

Crystal structure of the FAS1 domain of the hyaluronic acid receptor stabilin-2

Design, Synthesis, Evaluation, and Structural Studies of C2-Symmetric Small Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction

Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists

Di-Bromo-based small-molecule inhibitors of the PD-1/PD-L1 immune checkpoint

Human and mouse PD-L1: similar molecular structure, but different druggability profiles

Identification of small-molecule inhibitors of USP2a

Macrocyclic Peptide Inhibitor of PD‐1/PD‐L1 Immune Checkpoint

Mechanism of MyD88S mediated signal termination

Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

PD-L1 Inhibitors: Different Classes, Activities, and Mechanisms of Action

Rational design and synthesis of 1,5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction.

Small-Molecule Inhibitors of the Programmed Cell Death-1/Programmed Death-Ligand 1 (PD-1/PD-L1) Interaction via Transiently Induced Protein States and Dimerization of PD-L1.

Small-molecule inhibitors of PD-1/PD-L1 immune checkpoint alleviate the PD-L1-induced exhaustion of T-cells.

Structural Characterization of a Macrocyclic Peptide Modulator of the PD-1/PD-L1 Immune Checkpoint Axis

Structural basis for small molecule targeting of the programmed death ligand 1 (PD-L1)

Structure of the Complex of Human Programmed Death 1, PD-1, and Its Ligand PD-L1.

Synthesis of the New Heterocyclic System 5,6,10b-Triazaacephenanthrylene, a Nitrogen Analogue of Aristolactams

Synthesis, structure, and photophysical properties of luminescent zinc and cadmium complexes containing 2-pyridyl-substituted pyrrolo[2,3- b ]quinoxaline

Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein-Protein Interaction

Terphenyl-based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein−Protein Interaction

Terphenyl-based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein−Protein Interaction

The neutralization of heparan sulfate by heparin-binding copolymer as a potential therapeutic target

The synthesis and characterization of tetramic acid derivatives as Mdm2-p53 inhibitors

Two-Step Synthesis of Complex Artificial Macrocyclic Compounds

π-π-Induced aggregation and single-crystal fluorescence anisotropy of 5,6,10b-tri-aza-acephenanthrylene.