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List of works by Sylvia Els-Heindl

A Selective Carborane-Functionalized Gastrin-Releasing Peptide Receptor Agonist as Boron Delivery Agent for Boron Neutron Capture Therapy

scientific article published on 23 December 2019

A stable meta -carborane enables the generation of boron-rich peptide agonists targeting the ghrelin receptor

scientific article published on 31 August 2018

Adrenomedullin - Current Perspective on a Peptide Hormone with Significant Therapeutic Potential

scientific article published on 19 June 2020

Adrenomedullin - new perspectives of a potent peptide hormone

scientific article published on 2 February 2017

Adrenomedullin 2.0: Adjusting Key Levers for Metabolic Stability

scientific article published on 10 May 2016

Adrenomedullin disulfide bond mimetics uncover structural requirements for AM1 receptor activation

scientific article published on 24 January 2019

Automated solid-phase peptide synthesis to obtain therapeutic peptides

scientific article

Bioorthogonal Labeling of Ghrelin Receptor to Facilitate Studies of Ligand-Dependent Conformational Dynamics

scientific article published on 3 November 2015

C-terminus of a hexapeptidic ghrelin receptor inverse agonist can switch peptide behavior from inverse agonism to agonism

scientific article published on 01 January 2016

Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging.

scientific article published on 05 April 2017

Development of Potent and Metabolically Stable APJ Ligands with High Therapeutic Potential.

scientific article

Expression, Functional Characterization, and Solid-State NMR Investigation of the G Protein-Coupled GHS Receptor in Bilayer Membranes

scientific article published on 7 April 2017

High metabolic in vivo stability and bioavailability of a palmitoylated ghrelin receptor ligand assessed by mass spectrometry

scientific article published on 10 December 2014

Identification and stabilization of a highly selective gastrin-releasing peptide receptor agonist

scientific article published on 19 November 2019

Integrating solid-state NMR and computational modeling to investigate the structure and dynamics of membrane-associated ghrelin

scientific article

Peptide chemistry toolbox - Transforming natural peptides into peptide therapeutics

scientific article published on 29 January 2018

Peptide mini-scaffold facilitates JNK3 activation in cells

scientific article published on 12 February 2016

Peptide-Drug Conjugates and Their Targets in Advanced Cancer Therapies

scientific article published on 07 July 2020

Rational design of dual peptides targeting ghrelin and Y2 receptors to regulate food intake and body weight

scientific article published on 7 May 2015

Selective Neuropeptide Y Conjugates with Maximized Carborane Loading as Promising Boron Delivery Agents for Boron Neutron Capture Therapy

scientific article published on 22 October 2019

Side Chain Orientation of Tryptophan Analogues Determines Agonism and Inverse Agonism in Short Ghrelin Peptides

scientific article published on 16 September 2019

Structural Model of Ghrelin Bound to its G Protein-Coupled Receptor

scientific article published on 24 January 2019

The Impact of Adrenomedullin Thr22 on Selectivity within the Calcitonin Receptor-like Receptor/Receptor Activity-Modifying Protein System

scientific article published on 31 July 2018

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