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List of works by Mark Turlington

Activation of Vinyl Iodides for the Highly Enantioselective Addition to Aldehydes ⬇️

scientific article published on February 7, 2011

Acyl dihydropyrazolo[1,5-a]pyrimidinones as metabotropic glutamate receptor 5 positive allosteric modulators

scientific article published on 9 October 2015

Discovery and SAR of a novel series of metabotropic glutamate receptor 5 positive allosteric modulators with high ligand efficiency

scientific article

Evaluation of 1,2,3-Triazoles as Amide Bioisosteres In Cystic Fibrosis Transmembrane Conductance Regulator Modulators VX-770 and VX-809

scientific article published on 11 February 2019

Exploration of allosteric agonism structure-activity relationships within an acetylene series of metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulators (PAMs): discovery of 5-((3-fluorophenyl)ethynyl)-N-(3-methyloxetan-3-yl)picolin

scientific article

From Highly Enantioselective Catalytic Reaction of 1,3-Diynes with Aldehydes to Facile Asymmetric Synthesis of Polycyclic Compounds ⬇️

scientific article published on July 11, 2011

Heterotropic activation of the midazolam hydroxylase activity of CYP3A by a positive allosteric modulator of mGlu5: in vitro to in vivo translation and potential impact on clinically relevant drug-drug interactions

scientific article published on 03 September 2013

Reverse the Diastereoselectivity of the Rh(I)-Catalyzed Pauson-Khand Cycloaddition ⬇️

scientific article published on July 18, 2011

Study of the Fluorescent Properties of Partially Hydrogenated 1,1′-Bi-2-naphthol-amine Molecules and Their Use for Enantioselective Fluorescent Recognition ⬇️

scientific article published on March 24, 2011

Targeting selective activation of M(1) for the treatment of Alzheimer's disease: further chemical optimization and pharmacological characterization of the M(1) positive allosteric modulator ML169.

scientific article

Tetrahydronaphthyridine and dihydronaphthyridinone ethers as positive allosteric modulators of the metabotropic glutamate receptor 5 (mGlu₅).

scientific article

Total Synthesis of Stemaphylline N‐Oxide and Related C9a‐Epimeric Analogues ⬇️

scientific article published on August 16, 2013

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