List of works - Philippe Sarret

Apelin-13 in septic shock: effective in supporting hemodynamics in sheep but compromised by enzymatic breakdown in patients

scientific article published on 23 November 2021

Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists

scientific article published on 27 November 2019

Epithelial BMP signaling is required for proper specification of epithelial cell lineages and gastric endocrine cells ⬇️

scientific article published on March 17, 2011

Immunohistochemical distribution of NTS2 neurotensin receptors in the rat central nervous system ⬇️

scientific article published on July 7, 2003

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

scientific article published on 21 October 2019

Postnatal administration of IL-1Ra exerts neuroprotective effects following perinatal inflammation and/or hypoxic-ischemic injuries ⬇️

scientific article published on September 13, 2012

Regional and cellular distribution of low affinity neurotensin receptor mRNA in adult and developing mouse brain ⬇️

scientific article published on May 11, 1998

Regional and subcellular distribution of the receptor‐targeting protein PIST in the rat central nervous system ⬇️

scientific article published on April 1, 2012

Spinal NTS2 receptor activation reverses signs of neuropathic pain

scientific article published on 11 June 2013

Stereoselective Synthesis of β-(5-Arylthiazolyl) α-Amino Acids and Use in Neurotensin Analogues

Structural insights on ligand recognition at the human leukotriene B4 receptor 1

scientific article published on 20 May 2021

Structure-Activity Relationship and Bioactivity of Short Analogues of ELABELA as Agonists of the Apelin Receptor

scientific article published on 22 December 2020

Structure-based mechanism of cysteinyl leukotriene receptor inhibition by antiasthmatic drugs

scientific article published on 09 October 2019

Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues.

scientific article published on 8 September 2015

The P2Y6 receptor signals through Gαq /Ca2+ /PKCα and Gα13 /ROCK pathways to drive the formation of membrane protrusions and dictate cell migration

scientific article published on 18 May 2020

Use of Molecular Modeling to Design Selective NTS2 Neurotensin Analogues.

scientific article published on 3 April 2017

Use of a non-invasive brain penetrating peptide-drug conjugate strategy to improve the delivery of opioid pain relief medications to the brain

scientific article published on 23 April 2020

List of works by Philippe Sarret