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List of works by Paul Bamborough

A Chemical Probe for the ATAD2 Bromodomain

scientific article

A Qualified Success: Discovery of a New Series of ATAD2 Bromodomain Inhibitors with a Novel Binding Mode Using High-Throughput Screening and Hit Qualification

scientific article published on 09 August 2019

Aiming to Miss a Moving Target: Bromo and Extra Terminal Domain (BET) Selectivity in Constrained ATAD2 Inhibitors

article

CDK12 inhibition reduces abnormalities in cells from patients with myotonic dystrophy and in a mouse model

scientific article published on 01 April 2020

Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening

scientific article published on 06 January 2020

Selective targeting of BD1 and BD2 of the BET proteins in cancer and immuno-inflammation

scientific article

Structure-Based Design of a Bromodomain and Extraterminal Domain (BET) Inhibitor Selective for the N-Terminal Bromodomains That Retains an Anti-inflammatory and Antiproliferative Phenotype

scientific article published on 03 August 2020

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