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List of works by Mario van der Stelt

ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction

scientific article published on 01 October 2019

ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction

scientific article published on 07 November 2019

Activity-Based Protein Profiling Delivers Selective Drug Candidate ABX-1431, a Monoacylglycerol Lipase Inhibitor, To Control Lipid Metabolism in Neurological Disorders

article

Activity-Based Protein Profiling Identifies α-Ketoamides as Inhibitors for Phospholipase A2 Group XVI

scientific article published on 18 January 2019

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.

scientific article

Chemical genetics strategy to profile kinase target engagement reveals role of FES in neutrophil phagocytosis

scientific article published on 25 June 2020

Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice

scientific article published on 11 May 2020

Drug Discovery Maps, a machine learning model, visualizes and predicts kinome-inhibitor interaction landscapes

scientific article published on 08 November 2018

STA-55, an Easily Accessible, Broad-Spectrum, Activity-Based Aldehyde Dehydrogenase Probe

scientific article published on 27 January 2020

Structure Kinetics Relationships and Molecular Dynamics Show Crucial Role for Heterocycle Leaving Group in Irreversible Diacylglycerol Lipase Inhibitors

scientific article published on 30 August 2019

Structure-Activity Relationship Studies of α-Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family

scientific article published on 13 August 2020