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List of works by Suresh V Ambudkar

A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein

scientific article published on 12 September 2019

ABC-transporter upregulation mediates resistance to the CDK7 inhibitors THZ1 and ICEC0942

scientific article published on 17 September 2019

ATP-dependent thermostabilization of human P-glycoprotein (ABCB1) is blocked by modulators

scientific article published on 27 November 2019

Comprehensive Synthesis of Amino Acid-Derived Thiazole Peptidomimetic Analogues to Understand the Enigmatic Drug/Substrate-Binding Site of P-Glycoprotein

scientific article

Evidence for the critical role of transmembrane helices 1 and 7 in substrate transport by human P-glycoprotein (ABCB1)

scientific article published in PLoS ONE

Mapping discontinuous epitopes for MRK-16, UIC2 and 4E3 antibodies to extracellular loops 1 and 4 of human P-glycoprotein

scientific article published in Scientific Reports

Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles

scientific article published on 19 January 2021

Multidrug transporters: recent insights from cryo-electron microscopy-derived atomic structures and animal models

scientific article published on 13 January 2020

Nonsynonymous Mutations in Linker-2 of the Pdr5 Multidrug Transporter Identify a New RNA Stability Element

scientific article published on 07 January 2020

P-glycoprotein Mediates Resistance to the Anaplastic Lymphoma Kinase Inhiitor Ensartinib in Cancer Cells

scientific article published on 09 May 2022

Reversing the direction of drug transport mediated by the human multidrug transporter P-glycoprotein

scientific article published on 09 November 2020

Synthetic Analogs of Curcumin Modulate the Function of Multidrug Resistance-Linked ATP-Binding Cassette Transporter ABCG2.

scientific article published on 13 September 2017

Tivantinib, A c-Met Inhibitor in Clinical Trials, Is Susceptible to ABCG2-Mediated Drug Resistance

scientific article published on 12 January 2020