List of works by William J Zuercher

1,2,6-Thiadiazinones as Novel Narrow Spectrum Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CaMKK2) Inhibitors.

scientific article

A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation

scientific article published on 20 November 2020

A public-private partnership to unlock the untargeted kinome

scientific article published in January 2013

A trust approach for sharing research reagents.

scientific article published on May 2017

An in silico screen and structural analysis identifies bacterial kinase inhibitors which act with β-lactams to inhibit mycobacterial growth

scientific article published on 18 October 2018

CDK12 inhibition reduces abnormalities in cells from patients with myotonic dystrophy and in a mouse model

scientific article published on 01 April 2020

CaMKK2 in myeloid cells is a key regulator of the immune-suppressive microenvironment in breast cancer

scientific article published on 04 June 2019

Comprehensive characterization of the Published Kinase Inhibitor Set

scientific article

Covalent inhibitors of EGFR family protein kinases induce degradation of human Tribbles 2 (TRIB2) pseudokinase in cancer cells.

scientific article published on 25 September 2018

Design and Analysis of the 4-Anilinoquin(az)oline Kinase Inhibition Profiles of GAK/SLK/STK10 Using Quantitative Structure-Activity Relationships

scientific article published on 26 November 2019

Design of a Cyclin G Associated Kinase (GAK)/Epidermal Growth Factor Receptor (EGFR) Inhibitor Set to Interrogate the Relationship of EGFR and GAK in Chordoma

scientific article published on 19 April 2019

Donated chemical probes for open science.

scientific article published on 20 April 2018

Erratum: Corrigendum: The promise and peril of chemical probes

scientific article published in November 2015

Gram-scale synthesis of FICZ, a photoreactive endogenous ligand of the aryl hydrocarbon receptor

scientific article published on 10 July 2019

Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase.

scientific article

Identification of lead anti-human cytomegalovirus compounds targeting MAP4K4 via machine learning analysis of kinase inhibitor screening data

scientific article published in PLoS ONE

New Insights into 4-Anilinoquinazolines as Inhibitors of Cardiac Troponin I-Interacting Kinase (TNNi3K)

scientific article published on 07 April 2020

New tools for carbohydrate sulfation analysis: heparan sulfate 2--sulfotransferase (HS2ST) is a target for small-molecule protein kinase inhibitors

article

New tools for evaluating protein tyrosine sulfation: tyrosylprotein sulfotransferases (TPSTs) are novel targets for RAF protein kinase inhibitors

article

Quinazoline-Based Antivirulence Compounds Selectively Target Salmonella PhoP/PhoQ Signal Transduction System

scientific article published on 20 December 2019

Repurposing Eukaryotic Kinase Inhibitors as Colistin Adjuvants in Gram-Negative Bacteria

scientific article published on 04 September 2019

SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK)

scientific article published on 26 February 2019

The Intersection of Structural and Chemical Biology - An Essential Synergy

scientific article

The promise and peril of chemical probes

scientific article

Towards the Development of an In vivo Chemical Probe for Cyclin G Associated Kinase (GAK)

scientific article published on 06 November 2019

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