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List of works by Erik V Van der Eycken

A Gold(I)-Catalyzed Hydroamination/Cycloisomerization Cascade: Concise Synthesis of (±)-seco-Antofine and (±)-Septicine

scientific article published on 13 October 2020

A Gold-Catalyzed Domino Cyclization Enabling Rapid Construction of Diverse Polyheterocyclic Frameworks

scientific article

A Lewis Base Catalysis Approach for the Photoredox Activation of Boronic Acids and Esters.

scientific article published on 11 October 2017

A chromone analog inhibits TNF-alpha induced expression of cell adhesion molecules on human endothelial cells via blocking NF-kappaB activation

scientific article published on 12 February 2007

A divergent synthesis of substituted 2-aminoimidazoles from 2-aminopyrimidines

scientific article published on 26 July 2008

A gold-triggered dearomative spirocarbocyclization/Diels-Alder reaction cascade towards diverse bridged N-heterocycles

scientific article published on 01 November 2019

A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: synthesis and biological evaluation.

scientific article published on 22 March 2011

A new colorimetric test for solid-phase amines and thiols

scientific article published on 11 June 2008

A novel and versatile entry to asymmetrically substituted pyrazines

scientific article

A walk around the A3-coupling

scientific article published on 15 March 2012

Access to Polycyclic Azepino[5,4,3-cd]indoles via a Gold-Catalyzed Post-Ugi Dearomatization Cascade

scientific article published on 17 November 2020

Aldehydes: magnificent acyl equivalents for direct acylation

scientific article published on 01 October 2020

An antibiofilm coating of 5-aryl-2-aminoimidazole covalently attached to a titanium surface

scientific article published on 13 December 2018

Anti-inflammatory and antioxidant properties of Piper species: a perspective from screening to molecular mechanisms.

scientific article

Arylalkyl Ketones, Benzophenones, Desoxybenzoins and Chalcones Inhibit TNF‐α Induced Expression of ICAM‐1: Structure‐Activity Analysis ⬇️

scientific article published on December 20, 2011

C-N bond forming cross-coupling reactions: an overview

scientific article published on 30 September 2013

Chemo- and Regioselective Catalyst-Controlled Carbocyclization of Alkynyl Ketones: Rapid Synthesis of 1-Indanones and 1-Naphthols

scientific article published on 10 May 2019

Click chemistry under non-classical reaction conditions.

scientific article published on 27 July 2009

Combining the Ugi-azide multicomponent reaction and rhodium(III)-catalyzed annulation for the synthesis of tetrazole-isoquinolone/pyridone hybrids

scientific article published on 16 October 2019

Concise and diversity-oriented route toward polysubstituted 2-aminoimidazole alkaloids and their analogues.

scientific article published on December 2010

Copper‐Catalyzed Direct Secondary and Tertiary CH Alkylation of Azoles through a Heteroarene–Amine–Aldehyde/Ketone Coupling Reaction ⬇️

scientific article published on January 22, 2013

CuICuII and AgIp-isocyanobenzoates as novel 1D semiconducting coordination oligomers

scientific article published on 27 August 2020

DBU-Catalyzed Alkyne-Imidate Cyclization toward 1-Alkoxypyrazino[1,2- a]indole Synthesis

scientific article published on 19 July 2018

Development of a new microwave-assisted cleavable backbone amide linker (BAL): a comparative study

scientific article published on 19 November 2009

Developments in direct C-H arylation of (hetero)arenes under microwave irradiation.

scientific article published on 4 January 2013

Direct Heteroarylation of Tautomerizable Heterocycles into Unsymmetrical and Symmetrical Biheterocycles via Pd/Cu-Catalyzed Phosphonium Coupling ⬇️

scientific article published on March 14, 2012

Diversity oriented microwave-assisted synthesis of (-)-steganacin aza-analogues.

scientific article published on 28 August 2008

Doebner-type pyrazolopyridine carboxylic acids in an Ugi four-component reaction

scientific article published on 12 June 2019

Domino Carbopalladation/C-H Functionalization Sequence: An Expedient Synthesis of Bis-Heteroaryls through Transient Alkyl/Vinyl-Palladium Species Capture

scientific article published on 20 November 2015

Enhancing the anti-biofilm activity of 5-aryl-2-aminoimidazoles through nature inspired dimerisation

scientific article published on 31 January 2018

Evaluation of the antibacterial and antibiofilm activities of novel CRAMP-vancomycin conjugates with diverse linkers.

scientific article

Evaluation of the toxicity of 5-aryl-2-aminoimidazole-based biofilm inhibitors against eukaryotic cell lines, bone cells and the nematode Caenorhabditis elegans.

scientific article

Facile access to functionalized spiro[indoline-3,2'-pyrrole]-2,5'-diones via post-Ugi domino Buchwald-Hartwig/Michael reaction

scientific article

Facile construction of diverse polyheterocyclic scaffolds via gold-catalysed dearomative spirocyclization/1,6-addition cascade

scientific article published on 01 June 2019

Gold-Catalyzed Post-Ugi Ipso-Cyclization with Switchable Diastereoselectivity

scientific article published on 11 July 2018

Gold-catalyzed diastereoselective domino dearomatization/ipso-cyclization/aza-Michael sequence: a facile access to diverse fused azaspiro tetracyclic scaffolds

scientific article published in June 2017

Gold-catalyzed post-MCR transformations towards complex (poly)heterocycles

scientific article published on 28 August 2018

Gold-catalyzed post-Ugi alkyne hydroarylation for the synthesis of 2-quinolones

scientific article published on 04 October 2018

Heck-Suzuki Tandem Reaction for the Synthesis of 3-Benzazepines

scientific article published on 12 June 2015

High-speed microwave-promoted hetero-Diels-Alder reactions of 2(1H)-pyrazinones in ionic liquid doped solvents

scientific article published in November 2002

Hypervalent Iodine(III)-Mediated Cascade Cyclization of Propargylguanidines and Total Syntheses of Kealiinine B and C.

scientific article published on 29 March 2017

Identification of small peptides inhibiting the integrase-LEDGF/p75 interaction through targeting the cellular co-factor

scientific article published on 27 August 2013

Inhibiting bacterial cooperation is an evolutionarily robust anti-biofilm strategy

scientific article published on 09 January 2020

Iron(II)-Catalyzed Heck-Type Coupling of Vinylarenes with Alkyl Iodides

scientific article published on 22 January 2019

Iterative Chemical Engineering of Vancomycin Leads to Novel Vancomycin Analogs With a High in Vitro Therapeutic Index.

scientific article published on 7 June 2018

Metal-Free Dearomatization: Direct Access to Spiroindol(en)ines in Batch and Continuous-Flow

scientific article published on 21 January 2019

Metal-mediated post-Ugi transformations for the construction of diverse heterocyclic scaffolds

scientific article published on 05 February 2015

Microwave-Assisted Copper-Catalyzed Oxidative Cyclization of Acrylamides with Non-Activated Ketones

scientific article published on 12 February 2016

Microwave-assisted Cu(I)-catalyzed, three-component synthesis of 2-(4-((1-phenyl-1H-1,2,3-triazol-4-yl)methoxy)phenyl)-1H-benzo[d]imidazoles

scientific article published on 24 June 2014

Microwave-assisted C–C bond forming cross-coupling reactions: an overview ⬇️

scientific article published on June 30, 2011

Microwave-assisted cycloaddition reactions

scientific article published on December 2009

Microwave-assisted one-pot synthesis and anti-biofilm activity of 2-amino-1H-imidazole/triazole conjugates

scientific article published on 24 April 2014

Microwave-assisted synthesis of a novel class of imidazolylthiazolidin-4-ones and evaluation of its biological activities.

scientific article

Microwave-assisted synthesis of medium-sized heterocycles

scientific article published on 27 October 2011

Microwave-enhanced transition metal-catalyzed decoration of 2(1H)-pyrazinone scaffolds

scientific article published in January 2003

Modular Access to Diverse Bridged Indole Alkaloid Mimics via a Gold-Triggered Cascade Dearomative Spirocarbocyclization/[4 + 2] Cycloaddition Sequence

scientific article published on 05 June 2019

Modulation of the Substitution Pattern of 5-Aryl-2-Aminoimidazoles Allows Fine-Tuning of Their Antibiofilm Activity Spectrum and Toxicity.

scientific article published on 22 August 2016

New tricks of well-known aminoazoles in isocyanide-based multicomponent reactions and antibacterial activity of the compounds synthesized.

scientific article

Novel (2-amino-4-arylimidazolyl)propanoic acids and pyrrolo[1,2-c]imidazoles via the domino reactions of 2-amino-4-arylimidazoles with carbonyl and methylene active compounds

scientific article published on 06 May 2019

One-pot microwave-assisted protocol for the synthesis of substituted 2-amino-1H-imidazoles ⬇️

scientific article published on August 26, 2010

Pd-catalyzed Csp(2) -H functionalization of heteroarenes via isocyanide insertion: concise synthesis of di-(hetero)aryl ketones and di-(hetero)aryl alkylamines

scientific article published on 6 February 2015

Pd/Cu-Catalyzed C–H Arylation of 1,3,4-Thiadiazoles with (Hetero)aryl Iodides, Bromides, and Triflates ⬇️

scientific article published on September 21, 2012

Peptide macrocyclization by transition metal catalysis

scientific article published on 01 April 2020

Photoredox-Catalyzed Hydrosulfonylation of Arylallenes

scientific article published on 06 January 2020

Polysubstituted 2-aminoimidazoles as anti-biofilm and antiproliferative agents: Discovery of potent lead.

scientific article published on 24 June 2017

Post-Ugi Cyclization for the Construction of Diverse Heterocyclic Compounds: Recent Updates

scientific article published on 20 November 2018

Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines

scientific article

Reactions of secondary propargylamines with heteroallenes for the synthesis of diverse heterocycles

scientific article published on 16 March 2018

Recent Advances in Phthalan and Coumaran Chemistry

scientific article published on 23 November 2018

Recent advances in spirocyclization of indole derivatives.

scientific article published on 10 April 2018

Retraction of "Iron-Catalyzed Three-Component Reaction: Synthesis of Fluoroalkylated 2 H-Azirines"

scientific article published on 21 November 2018

Rhodium(iii)-catalyzed intramolecular annulation through C-H activation: concise synthesis of rosettacin and oxypalmatime.

scientific article published on 28 September 2017

Ruthenium-catalysed one-pot regio- and diastereoselective synthesis of pyrrolo[1,2-a]indoles via cascade C-H functionalization/annulation

scientific article published on 18 September 2017

Sequential and direct multicomponent reaction (MCR)-based dearomatization strategies

scientific article published on 20 October 2020

Smart Metal-Organic Framework Coatings: Triggered Antibiofilm Compound Release

scientific article published on 12 January 2017

Solid-phase synthesis of the 2(1H)-pyrazinone scaffold: a new approach toward diversely substituted heterocycles

scientific article

Structure-activity relationship of 2-hydroxy-2-aryl-2,3-dihydro-imidazo[1,2-a]pyrimidinium salts and 2N-substituted 4(5)-aryl-2-amino-1H-imidazoles as inhibitors of biofilm formation by Salmonella Typhimurium and Pseudomonas aeruginosa.

scientific article

Structure-activity relationship of 4(5)-aryl-2-amino-1H-imidazoles, N1-substituted 2-aminoimidazoles and imidazo[1,2-a]pyrimidinium salts as inhibitors of biofilm formation by Salmonella typhimurium and Pseudomonas aeruginosa.

scientific article published on 20 December 2010

Suzuki-Miyaura and Stille reactions as key steps in the synthesis of diversely functionalized Amaryllidaceae alkaloid analogs bearing a 5,6,7,8-tetrahydrobenzo[c,e]azocine skeleton

scientific article published in November 2007

Switching the regioselectivity via indium(III) and gold(I) catalysis: a post-Ugi intramolecular hydroarylation to azepino- and azocino-[c,d]indolones.

scientific article published in August 2013

Synthesis and HIV-1 RT inhibitory action of novel (4/6-substituted benzo[d]thiazol -2-yl)thiazolidin-4-ones. Divergence from the non-competitive inhibition mechanism

scientific article published in March 2012

Synthesis and anti-inflammatory activity evaluation of novel chroman derivatives

scientific article published in 2020

Synthesis and anti-inflammatory activity evaluation of novel triazolyl-isatin hybrids.

scientific article published on 5 May 2016

Synthesis and fungicidal activity of 3,5-dichloropyrazin-2(1H)-one derivatives.

scientific article published on 13 June 2009

Synthesis of 1-(-methoxyphenyl)tetrazolyl-Substituted 1,2,3,4-Tetrahydroisoquinolines and Their Transformations Involving Activated Alkynes

scientific article published on 17 November 2018

Synthesis of Differentially Substituted 2-Aminoimidazolidines via a Microwave-Assisted Tandem Staudinger/Aza-Wittig Cyclization ⬇️

scientific article published on May 14, 2013

Synthesis of Pyrrolo[1,2-b]isoquinolines via Gold(I)-Catalyzed Cyclization/Enyne Cycloisomerization/1,2-Migration Cascade

scientific article published on 10 August 2020

Synthetic Access to Secondary Propargylamines via a Copper-Catalyzed Oxidative Deamination/Alkynylation Cascade

scientific article published on 07 August 2019

The application of "click chemistry" for the decoration of 2(1H)-pyrazinone scaffold: generation of templates.

scientific article published in May 2005

Three-Component Reaction of 3-Arylidene-3H-Indolium Salts, Isocyanides, and Alcohols

scientific article published on 16 May 2019

Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives

scientific article

Transition metal-catalyzed C-C bond formation via C-S bond cleavage: an overview

scientific article published on June 2013

Transition metal-catalyzed orthogonal solid-phase decoration of the 2(1H)-pyrazinone scaffold using a sulfur linker

scientific article

Tunability of Size and Magnetic Moment of Iron Oxide Nanoparticles Synthesized by Forced Hydrolysis

scientific article published on 8 July 2016

Unprecedented Cu(I)-catalyzed microwave-assisted three-component coupling of a ketone, an alkyne, and a primary amine.

scientific article published in June 2010

Validation of an ultra-high-performance liquid chromatography-mass spectrometry method for the quantification of cysteinylated aldehydes and application to malt and beer samples

scientific article published on 20 August 2019

Visible light-mediated chemistry of indoles and related heterocycles

scientific article published on 01 August 2019

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