List of works - Evi Kostenis

3-(2-Carboxyethyl)indole-2-carboxylic Acid Derivatives: Structural Requirements and Properties of Potent Agonists of the Orphan G Protein-Coupled Receptor GPR17

scientific article published on 05 September 2018

A MassQL-Integrated Molecular Networking Approach for the Discovery and Substructure Annotation of Bioactive Cyclic Peptides

Author Correction: Chemokine receptor trafficking coordinates neutrophil clustering and dispersal at wounds in zebrafish

scientific article published on 21 January 2020

BIM-46174 fragments as potential ligands of G proteins

scientific article published on 21 August 2019

Chemokine receptor trafficking coordinates neutrophil clustering and dispersal at wounds in zebrafish

scientific article published on 14 November 2019

Deciphering Specificity Determinants for FR900359-Derived Gq α Inhibitors Based on Computational and Structure-Activity Studies

scientific article published on 03 July 2018

Delineation of molecular determinants for FR900359 inhibition of Gq/11 unlocks inhibition of Gαs

scientific article published on 04 August 2020

Direct targeting of Gαq and Gα11 oncoproteins in cancer cells

scientific article published on 19 March 2019

FZD5 is a Gαq-coupled receptor that exhibits the functional hallmarks of prototypical GPCRs

scientific article published on 04 December 2018

Feature-Based Molecular Networking for the Targeted Identification of G<sub>q</sub>-Inhibiting FR900359 Derivatives

scientific article published in July 2021

Gq/11-dependent regulation of endosomal cAMP generation by parathyroid hormone class B GPCR

scientific article published on 17 March 2020

Gβγ signaling to the chemotactic effector P-REX1 and mammalian cell migration is directly regulated by Gαq and Gα13 proteins

scientific article published on 16 November 2018

Heterotrimeric Gq proteins as therapeutic targets?

scientific article published on 02 March 2020

Impaired endothelium-mediated cerebrovascular reactivity promotes anxiety and respiration disorders in mice

scientific article published on 02 January 2020

Rational design of a heterotrimeric G protein α subunit with artificial inhibitor sensitivity

scientific article published on 11 February 2019

Selective optogenetic control of G<sub>q</sub> signaling using human Neuropsin

scientific article published on 01 April 2022

Targeted inhibition of Gq signaling induces airway relaxation in mouse models of asthma

scientific article published in September 2017

The atypical chemokine receptor ACKR3/CXCR7 is a broad-spectrum scavenger for opioid peptides

scientific article published on 19 June 2020

Thioesterase-mediated side chain transesterification generates potent Gq signaling inhibitor FR900359

scientific article published on 08 January 2021

List of works by Evi Kostenis