List of works - Terrence R Burke

A novel macrocyclic tetrapeptide mimetic that exhibits low-picomolar Grb2 SH2 domain-binding affinity ⬇️

scientific article published on October 17, 2003

An NMR strategy for fragment-based ligand screening utilizing a paramagnetic lanthanide probe ⬇️

scientific article published on September 17, 2011

Application of a water-soluble pyridyl disulfide amine linker for use in Cu-free click bioconjugation ⬇️

scientific article published on August 17, 2011

Aromatic hydroxylation of beta-adrenergic antagonists. 4- and 5-hydroxylation of 1-(isopropylamino)-3-[2-(allyloxy)phenoxy]-2-propanol (oxprenolol)

scientific article published on December 1, 1978

Aromatic hydroxylation of beta-adrenergic antagonists. Formation of 4'- and 5'-hydroxy-1-(isopropylamino)-3-[2'-allyloxy)phenoxy]-2-propanol from oxprenolol

scientific article published on 01 September 1979

Authentic HIV-1 Integrase Inhibitors ⬇️

scientific article published on July 1, 2010

Calcium ion-dependent covalent modification of calmodulin with norchlorpromazine isothiocyanate ⬇️

scientific article published on November 22, 1983

High-Resolution Structure of the Yersinia pestis Protein Tyrosine Phosphatase YopH in Complex with a Phosphotyrosyl Mimetic-Containing Hexapeptide ⬇️

scientific article published on November 18, 2003

Identification of High Affinity Polo-like Kinase 1 (Plk1) Polo-box Domain Binding Peptides Using Oxime-Based Diversification ⬇️

scientific article published on February 14, 2012

Identification of a Mr 58 000 glycoprotein subunit of the opiate receptor ⬇️

scientific article published on December 13, 1982

Ionic conditions differentially affect 3H-DADL binding to type-I and type-II opiate delta receptors in vitro ⬇️

scientific article published on May 1, 1984

Irreversible Ligands with High Selectivity Toward δ and μ Opiate Receptors ⬇️

scientific article published on April 15, 1983

MK-0536 Inhibits HIV-1 Integrases Resistant to Raltegravir ⬇️

scientific article published on August 29, 2011

Metabolism of .beta.-adrenergic antagonists. Evidence for an arene oxide-NIH shift pathway in the aromatic hydroxylation of oxprenolol ⬇️

scientific article published on 01 September 1979

Morphine noncompetitively inhibits [3H]leucine enkephalin binding to membranes lacking type-II delta binding sites: Evidence for a two-site allosteric model ⬇️

scientific article published on May 1, 1984

Oxime-based linker libraries as a general approach for the rapid generation and screening of multidentate inhibitors ⬇️

scientific article published on March 15, 2012

Oxime‐Based Click Chemistry in the Development of 3‐Isoxazolecarboxylic Acid Containing Inhibitors of Yersinia pestis Protein Tyrosine Phosphatase, YopH ⬇️

scientific article published on June 10, 2011

Peptoid–Peptide Hybrid Ligands Targeting the Polo Box Domain of Polo‐Like Kinase 1 ⬇️

scientific article published on May 8, 2012

Phosphotyrosyl peptides and analogues as substrates and inhibitors of purple acid phosphatases

scientific article published in April 2004

Potent Inhibition of Insulin Receptor Dephosphorylation by a Hexamer Peptide Containing the Phosphotyrosyl Mimetic F2Pmp ⬇️

scientific article published on October 14, 1994

Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for .mu. or .delta. opiate receptors ⬇️

scientific article published on December 1, 1984

S-[18 F]Acetylcyclofoxy: a useful probe for the visualization of opiate receptors in living animals ⬇️

scientific article published on November 19, 1984

Salicylhydrazine-Containing Inhibitors of HIV-1 Integrase: Implication for a Selective Chelation in the Integrase Active Site ⬇️

scientific article published on August 13, 1998

Samarium Iodide-Mediated Reformatsky Reactions for the Stereoselective Preparation of β-Hydroxy-γ-amino Acids: Synthesis of Isostatine and Dolaisoleucine ⬇️

scientific article published on December 14, 2011

Site-Specific Lysine Arylation as an Alternative Bioconjugation Strategy for Chemically Programmed Antibodies and Antibody-Drug Conjugates

scientific article published on 01 November 2019

Structural basis for strand-transfer inhibitor binding to HIV intasomes

scientific article

Structural basis for the inhibition of HTLV-1 integration inferred from cryo-EM deltaretroviral intasome structures

scientific article published on 17 August 2021

Structure of the catalytic domain of avian sarcoma virus integrase with a bound HIV-1 integrase-targeted inhibitor ⬇️

scientific article published on April 28, 1998

Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors.

scientific article published on 24 July 2017

Synthesis and pharmacological characterization of (.+-.)-5,9.alpha.-dimethyl-2-[2-(4-fluorophenyl)ethyl]-2'-hydroxy-6,7-benzomorphan (fluorophen), a ligand suitable for visualization of opiate receptors in vivo ⬇️

scientific article published on November 1, 1983

Synthesis of 4'- and 5'-hydroxyoxprenolol: pharmacologically active ring-hydroxylated metabolites of oxprenolol ⬇️

scientific article published on December 1, 1979

Synthesis, configuration, and evaluation of two conformationally restrained analogs of phencyclidine ⬇️

scientific article published on August 1, 1988

The Stereoselective Disposition of Disopyramide in the Dog ⬇️

scientific article published on November 1, 1980

Tritiated-6-beta-fluoro-6-desoxy-oxymorphone: A highly selective ligand for the opiate mu receptor whose binding is characterized by low nonspecific binding ⬇️

scientific article published on June 1, 1984

Uncoupling the Folding-Function Paradigm of Lytic Peptides to Deliver Impermeable Inhibitors of Intracellular Protein-Protein Interactions

scientific article published on 11 November 2020

Utilization of Nitrophenylphosphates and Oxime-Based Ligation for the Development of Nanomolar Affinity Inhibitors of the Yersinia pestis Outer Protein H (YopH) Phosphatase ⬇️

scientific article published on March 28, 2011

Yersinia pestis and Approaches to Targeting its Outer Protein H Protein-Tyrosine Phosphatase (YopH) ⬇️

scientific article published on January 1, 2012

List of works by Terrence R Burke