List of works - Sungwoo Hong

A Pd-catalyzed one-pot dehydrogenative aromatization and ortho-functionalization sequence of N-acetyl enamides

scientific article published on 13 February 2014

A copper-mediated cross-coupling approach for the synthesis of 3-heteroaryl quinolone and related analogues

scientific article published on 26 June 2014

A facile route to isoflavone quinones via the direct cross-coupling of chromones and quinones

scientific article published on 11 June 2012

A novel PI3K inhibitor alleviates fibrotic responses in fibroblasts derived from Peyronie's plaques

scientific article published on 16 April 2013

A novel imidazopyridine PI3K inhibitor with anticancer activity in non-small cell lung cancer cells

scientific article published on 27 May 2013

A novel imidazopyridine analogue as a phosphatidylinositol 3-kinase inhibitor against human breast cancer

scientific article

A novel imidazopyridine derivative, HS-106, induces apoptosis of breast cancer cells and represses angiogenesis by targeting the PI3K/mTOR pathway

scientific article

AgSbF₆-controlled diastereodivergence in alkyne hydroarylation: facile access to Z- and E-alkenyl arenes

scientific article published on 01 July 2014

Allylic Acetals as Acrolein Oxonium Precursors in Tandem C-H Allylation and [3+2] Dipolar Cycloaddition

scientific article published on 03 June 2019

Aminoglycoside antibiotics bind to the influenza A virus RNA promoter.

scientific article published on 19 September 2012

Anti-cancer effect of HS-345, a new tropomyosin-related kinase A inhibitor, on human pancreatic cancer

scientific article published on 13 April 2013

Anti-cancer effects of a novel compound HS-113 on cell growth, apoptosis, and angiogenesis in human hepatocellular carcinoma cells.

scientific article published on 3 April 2011

Anticancer activity of HS-527, a novel inhibitor targeting PI3-kinase in human pancreatic cancer cells

scientific article

Application of Fragment-Based de Novo Design to the Discovery of Selective Picomolar Inhibitors of Glycogen Synthase Kinase-3 Beta

scientific article published on 27 September 2016

Asymmetric C-H functionalization of cyclopropanes using an isoleucine-NH2 bidentate directing group

scientific article published on 16 April 2015

C2-Selective C-H Methylation of Heterocyclic N-Oxides with Sulfonium Ylides

scientific article published on 09 November 2020

Catalyst Controlled Divergent C4/C8 Site-Selective C-H Arylation of Isoquinolones

scientific article published on 28 July 2015

Computational design and discovery of nanomolar inhibitors of IκB kinase β.

scientific article published on 2 January 2015

Construction of an advanced tetracyclic intermediate for total synthesis of the marine alkaloid sarain A

scientific article (publication date: 3 March 2006)

Correction to Identification of 4-Phenoxyquinoline Based Inhibitors for L1196M Mutant of Anaplastic Lymphoma Kinase by Structure-Based Design.

scientific article published on 22 February 2018

Design and synthesis of imidazopyridine analogues as inhibitors of phosphoinositide 3-kinase signaling and angiogenesis

scientific article published on 9 March 2011

Design, synthesis, and evaluation of 3,5-disubstituted 7-azaindoles as Trk inhibitors with anticancer and antiangiogenic activities

scientific article published on 18 May 2012

Development and biological evaluation of potent and selective c-KIT(D816V) inhibitors

scientific article

Development of new fluorescent xanthines as kinase inhibitors

scientific article

Direct C-H cross-coupling approach to heteroaryl coumarins

scientific article published on 22 February 2012

Direct Phosphonation of Quinolinones and Coumarins Driven by the Photochemical Activity of Substrates and Products

scientific article published on 02 March 2017

Discovery of EGF Receptor Inhibitors That Are Selective for the d746-750/T790M/C797S Mutant through Structure-Based de Novo Design.

scientific article published on 22 May 2017

Discovery of Low Micromolar Dual Inhibitors for Wild Type and L1196M Mutant of Anaplastic Lymphoma Kinase through Structure-Based Virtual Screening

scientific article

Discovery of MEK/PI3K dual inhibitor via structure-based virtual screening.

scientific article

Discovery of fluorescent 3-heteroarylcoumarin derivatives as novel inhibitors of anaplastic lymphoma kinase

scientific article published on 01 December 2018

Discovery of new aminopyrimidine-based phosphoinositide 3-kinase beta (PI3Kβ) inhibitors with selectivity over PI3Kα.

scientific article

Discovery of new azaindole-based PI3Kα inhibitors: Apoptotic and antiangiogenic effect on cancer cells ⬇️

scientific article published on October 26, 2010

Discovery of new benzothiazole-based inhibitors of breakpoint cluster region-Abelson kinase including the T315I mutant.

scientific article published on 19 April 2013

Discovery of picomolar ABL kinase inhibitors equipotent for wild type and T315I mutant via structure-based de novo design

scientific article published on 24 May 2013

Discovery of wrightiadione as a novel template for the TrkA kinase inhibitors

scientific article

Efficient synthesis of frutinone A and its derivatives through palladium-catalyzed C - H activation/carbonylation.

scientific article published on 22 September 2014

Fascaplysin Exerts Anti-Cancer Effects through the Downregulation of Survivin and HIF-1α and Inhibition of VEGFR2 and TRKA.

scientific article published on 29 September 2017

Fluorescent phosphoinositide 3-kinase inhibitors suitable for monitoring of intracellular distribution

scientific article published on 15 March 2011

Frontispiece: Visible‐Light‐Induced Cysteine‐Specific Bioconjugation: Biocompatible Thiol–Ene Click Chemistry

scientific article published in 2020

Frontispiz: Visible‐Light‐Induced Cysteine‐Specific Bioconjugation: Biocompatible Thiol–Ene Click Chemistry

scientific article published in 2020

Functionalization of Pyridinium Derivatives with 1,4-Dihydropyridines Enabled by Photoinduced Charge Transfer

scientific article published on 26 October 2020

HS-104, a PI3K inhibitor, enhances the anticancer efficacy of gemcitabine in pancreatic cancer.

scientific article

HS-116, a novel phosphatidylinositol 3-kinase inhibitor induces apoptosis and suppresses angiogenesis of hepatocellular carcinoma through inhibition of the PI3K/AKT/mTOR pathway

scientific article

HS-133, a novel fluorescent phosphatidylinositol 3-kinase inhibitor as a potential imaging and anticancer agent for targeted therapy

scientific article

HS-1371, a novel kinase inhibitor of RIP3-mediated necroptosis

scholarly article by Han-Hee Park published in September 2018

HS-173 as a novel inducer of RIP3-dependent necroptosis in lung cancer

scientific article published on 21 December 2018

HS-173, a novel PI3K inhibitor suppresses EMT and metastasis in pancreatic cancer

scientific article published on 25 October 2016

HS-173, a novel PI3K inhibitor, attenuates the activation of hepatic stellate cells in liver fibrosis

scientific article published on 11 December 2013

HS-173, a novel phosphatidylinositol 3-kinase (PI3K) inhibitor, has anti-tumor activity through promoting apoptosis and inhibiting angiogenesis

scientific article published on 26 August 2012

HS-438, a new inhibitor of imatinib-resistant BCR-ABL T315I mutation in chronic myeloid leukemia

scientific article published on 18 March 2014

HS-543 induces apoptosis of Imatinib-resistant chronic myelogenous leukemia with T315I mutation

scientific article

HS‑146, a novel phosphoinositide 3‑kinase α inhibitor, induces the apoptosis and inhibits the metastatic ability of human breast cancer cells

scientific article published on 19 March 2020

High-throughput chemical screening to discover new modulators of microRNA expression in living cells by using graphene-based biosensor.

scientific article published on 30 July 2018

IPD-196, a novel phosphatidylinositol 3-kinase inhibitor with potent anticancer activity against hepatocellular carcinoma

scientific article published on 8 November 2012

Identification of 4-Phenoxyquinoline Based Inhibitors for L1196M Mutant of Anaplastic Lymphoma Kinase by Structure-Based Design.

scientific article published in November 2017

Identification of common inhibitors of wild-type and T315I mutant of BCR-ABL through the parallel structure-based virtual screening.

scientific article

Identification of lead small molecule inhibitors of glycogen synthase kinase-3 beta using a fragment-linking strategy

scientific article published on 22 October 2016

Identification of novel BRAF kinase inhibitors with structure-based virtual screening

scientific article published on 08 August 2011

Identification of novel inhibitors of tropomyosin-related kinase A through the structure-based virtual screening with homology-modeled protein structure

scientific article

Identification of β-Lapachone Analogs as Novel MALT1 Inhibitors To Treat an Aggressive Subtype of Diffuse Large B-Cell Lymphoma

scientific article published on 23 October 2015

Induction of apoptosis and suppression of angiogenesis of hepatocellular carcinoma by HS-159, a novel phosphatidylinositol 3-kinase inhibitor

scientific article published on 22 April 2013

Kinase and GPCR polypharmacological approach for the identification of efficient anticancer medicines

scientific article published on 01 October 2020

Metal-Free, Visible-Light-Induced Remote C(sp3)-H Pyridylation via Radical Translocation of N-Alkoxypyridinium Salts

scientific article published on 23 October 2018

NiH-Catalyzed Proximal-Selective Hydroamination of Unactivated Alkenes

scientific article published on 18 November 2020

Nocodazole is a high-affinity ligand for the cancer-related kinases ABL, c-KIT, BRAF, and MEK.

scientific article published on 14 October 2011

One-pot catalysis of dehydrogenation of cyclohexanones to phenols and oxidative Heck coupling: expedient synthesis of coumarins

scientific article published on 3 April 2013

Optimization and biological evaluation of aminopyrimidine-based IκB kinase β inhibitors with potent anti-inflammatory effects

scientific article published in August 2016

Palladium(II)-Catalyzed Tandem Synthesis of Acenes Using Carboxylic Acids as Traceless Directing Groups

scientific article published on 31 May 2016

Palladium(II)-catalyzed direct intermolecular alkenylation of chromones

scientific article published on 28 July 2011

Palladium-Catalyzed Divergent Arylation of Triazolopyridines: A Computational Study

scientific article published on 20 June 2018

Palladium-catalyzed dehydrogenation/oxidative cross-coupling sequence of β-heteroatom-substituted ketones

scientific article published on 04 October 2012

Photocatalytic Vicinal Aminopyridylation of Methyl Ketones by a Double Umpolung Strategy

scientific article published on 30 June 2020

Photochemical Carbopyridylation of Alkenes Using N-Alkenoxypyridinium Salts as Bifunctional Reagents

scientific article published on 12 December 2019

Rational Computational Design of Fourth-Generation EGFR Inhibitors to Combat Drug-Resistant Non-Small Cell Lung Cancer

scientific article published on 07 December 2020

Reactivity of Morita-Baylis-Hillman Adducts in C-H Functionalization of (Hetero)aryl Nitrones: Access to Bridged Cycles and Carbazoles

scientific article published on 26 July 2018

Regiodivergent Ring-Opening Cross-Coupling of Vinyl Aziridines with Phosphorus Nucleophiles: Access to Phosphorus-Containing Amino Acid Derivatives

scientific article published on 02 November 2018

Regioselective C-H Functionalization of Heteroarene N-Oxides Enabled by a Traceless Nucleophile

scientific article published on 04 September 2020

Regioselective palladium-catalyzed direct cross-coupling of coumarins with simple arenes

scientific article published on 01 October 2012

Regioselective palladium-catalyzed olefination of coumarins via aerobic oxidative Heck reactions

scientific article published on 21 November 2012

Rh(III) and Ru(II)-catalyzed site-selective C-H alkynylation of quinolones

scientific article published on 30 March 2015

Rh(III)-catalyzed direct C-H/C-H cross-coupling of quinones with arenes assisted by a directing group: identification of carbazole quinones as GSKβ inhibitors

scientific article published on April 2015

Rh(iii)-catalyzed 7-azaindole synthesis via C-H activation/annulative coupling of aminopyridines with alkynes

scientific article published on 01 June 2015

Ru(II)-Catalyzed Site-Selective Hydroxylation of Flavone and Chromone Derivatives: The Importance of the 5-Hydroxyl Motif for the Inhibition of Aurora Kinases.

scientific article

Selective and potent small-molecule inhibitors of PI3Ks

scientific article

Selectivity enhancement arising from interactions at the PI3K unique pocket.

scientific article

Site-Selective 1,1-Difunctionalization of Unactivated Alkenes Enabled by Cationic Palladium Catalysis

scientific article published on 12 June 2019

Site-Selective Functionalization of Pyridinium Derivatives via Visible-Light-Driven Photocatalysis with Quinolinone

scientific article published on 03 June 2019

Stereoselective construction of sterically hindered oxaspirocycles via chiral bidentate directing group-mediated C(sp3)-O bond formation.

scientific article published on 27 November 2017

Strategic Approach to the Metamorphosis of γ-Lactones to NH γ-Lactams via Reductive Cleavage and C-H Amidation

scientific article published on 16 August 2019

Strategies to overcome acquired resistances conferred by mutations in the kinase domain of EGFR.

scientific article published on 19 May 2016

Structure-based de novo design and biochemical evaluation of novel BRAF kinase inhibitors.

scientific article

Structure-based de novo design and identification of D816V mutant-selective c-KIT inhibitors.

scientific article published in July 2014

Structure-based de novo design and synthesis of aminothiazole-based p38 MAP kinase inhibitors.

scientific article

Structure-based design of flavone-based inhibitors of wild-type and T315I mutant of ABL.

scientific article published on 6 June 2013

Structure-based virtual screening approach to the discovery of p38 MAP kinase inhibitors

scientific article published on 02 February 2012

Structure-based virtual screening approach to the discovery of phosphoinositide 3-kinase alpha inhibitors

scientific article published on 26 February 2011

Suppression of tumor proliferation and angiogenesis of hepatocellular carcinoma by HS-104, a novel phosphoinositide 3-kinase inhibitor

scientific article published on 15 August 2012

Synergistic anticancer activity of HS-173, a novel PI3K inhibitor in combination with Sorafenib against pancreatic cancer cells

scientific article published on 20 January 2013

Synergistic effect of graphene oxide/MWCNT films in laser desorption/ionization mass spectrometry of small molecules and tissue imaging

scientific article

Synthesis of Gemcitabine-Threonine Amide Prodrug Effective on Pancreatic Cancer Cells with Improved Pharmacokinetic Properties

scientific article published on 11 October 2018

Synthesis of heterocyclic-fused benzofurans via C-H functionalization of flavones and coumarins

scientific article published on September 2013

Synthesis of heterocyclic-fused benzopyrans via the Pd(II)-catalyzed C-H alkenylation/C-O cyclization of flavones and coumarins

scientific article published on 17 April 2014

Synthetic approach to flavanones and flavones via ligand-free palladium(II)-catalyzed conjugate addition of arylboronic acids to chromones

scientific article published on 01 September 2012

Systematic Computational Design and Identification of Low Picomolar Inhibitors of Aurora Kinase A.

scientific article

Tandem Dehydrogenation/Oxidation/Oxidative Cyclization Approach to Wrightiadione and Its Derivatives

scientific article

The effect of HS-111, a novel thiazolamine derivative, on apoptosis and angiogenesis of hepatocellular carcinoma cells

scientific article published on March 2012

Total synthesis of the Securinega alkaloid (-)-secu'amamine A.

scientific article published on 21 May 2008

Unraveling innate substrate control in site-selective palladium-catalyzed C-H heterocycle functionalization.

scientific article published on 8 March 2016

Virtual screening and biochemical evaluation to identify new inhibitors of mammalian target of rapamycin (mTOR).

scientific article

Visible Light-Driven C4-Selective Alkylation of Pyridinium Derivatives with Alkyl Bromides

scientific article published on 12 June 2020

Visible light induced alkene aminopyridylation using N-aminopyridinium salts as bifunctional reagents

scientific article published on 11 September 2019

Visible-Light Excitation of Quinolinone-Containing Substrates Enables Divergent Radical Cyclizations

scientific article published on 22 April 2019

Visible-Light-Enabled Ortho-Selective Aminopyridylation of Alkenes with N-Aminopyridinium Ylides

scientific article published on 02 July 2020

Visible-Light-Enabled Trifluoromethylative Pyridylation of Alkenes from Pyridines and Triflic Anhydride

scientific article published on 05 May 2020

Visible-Light-Induced 1,3-Aminopyridylation of [1.1.1]Propellane with N-Aminopyridinium Salts

scientific article published on 06 January 2021

Visible-Light-Induced C-O Bond Formation for the Construction of Five- and Six-Membered Cyclic Ethers and Lactones

scientific article published on 14 November 2018

Visible-Light-Induced Cysteine-Specific Bioconjugation: Biocompatible Thiol-Ene Click Chemistry

scientific article published on 31 August 2020

Visible-Light-Induced Remote C(sp3)-H Pyridylation of Sulfonamides and Carboxamides

scientific article published on 18 November 2019

Visible-Light-Induced ortho-Selective Migration on Pyridyl Ring: Trifluoromethylative Pyridylation of Unactivated Alkenes

scientific article published on 15 November 2019

Visible-Light-Photocatalyzed Synthesis of Phenanthridinones and Quinolinones via Direct Oxidative C-H Amidation.

scientific article published on 14 December 2017

Visible‐Light‐Induced Cysteine‐Specific Bioconjugation: Biocompatible Thiol–Ene Click Chemistry

scientific article published in 2020

List of works by Sungwoo Hong

A Pd-catalyzed one-pot dehydrogenative aromatization and ortho-functionalization sequence of N-acetyl enamides

A copper-mediated cross-coupling approach for the synthesis of 3-heteroaryl quinolone and related analogues

A facile route to isoflavone quinones via the direct cross-coupling of chromones and quinones

A novel PI3K inhibitor alleviates fibrotic responses in fibroblasts derived from Peyronie's plaques

A novel imidazopyridine PI3K inhibitor with anticancer activity in non-small cell lung cancer cells

A novel imidazopyridine analogue as a phosphatidylinositol 3-kinase inhibitor against human breast cancer

A novel imidazopyridine derivative, HS-106, induces apoptosis of breast cancer cells and represses angiogenesis by targeting the PI3K/mTOR pathway

AgSbF₆-controlled diastereodivergence in alkyne hydroarylation: facile access to Z- and E-alkenyl arenes

Allylic Acetals as Acrolein Oxonium Precursors in Tandem C-H Allylation and [3+2] Dipolar Cycloaddition

Aminoglycoside antibiotics bind to the influenza A virus RNA promoter.

Anti-cancer effect of HS-345, a new tropomyosin-related kinase A inhibitor, on human pancreatic cancer

Anti-cancer effects of a novel compound HS-113 on cell growth, apoptosis, and angiogenesis in human hepatocellular carcinoma cells.

Anticancer activity of HS-527, a novel inhibitor targeting PI3-kinase in human pancreatic cancer cells

Application of Fragment-Based de Novo Design to the Discovery of Selective Picomolar Inhibitors of Glycogen Synthase Kinase-3 Beta

Asymmetric C-H functionalization of cyclopropanes using an isoleucine-NH2 bidentate directing group

C2-Selective C-H Methylation of Heterocyclic N-Oxides with Sulfonium Ylides

Catalyst Controlled Divergent C4/C8 Site-Selective C-H Arylation of Isoquinolones

Computational design and discovery of nanomolar inhibitors of IκB kinase β.

Construction of an advanced tetracyclic intermediate for total synthesis of the marine alkaloid sarain A

Correction to Identification of 4-Phenoxyquinoline Based Inhibitors for L1196M Mutant of Anaplastic Lymphoma Kinase by Structure-Based Design.

Design and synthesis of imidazopyridine analogues as inhibitors of phosphoinositide 3-kinase signaling and angiogenesis

Design, synthesis, and evaluation of 3,5-disubstituted 7-azaindoles as Trk inhibitors with anticancer and antiangiogenic activities

Development and biological evaluation of potent and selective c-KIT(D816V) inhibitors

Development of new fluorescent xanthines as kinase inhibitors

Direct C-H cross-coupling approach to heteroaryl coumarins

Direct Phosphonation of Quinolinones and Coumarins Driven by the Photochemical Activity of Substrates and Products

Discovery of EGF Receptor Inhibitors That Are Selective for the d746-750/T790M/C797S Mutant through Structure-Based de Novo Design.

Discovery of Low Micromolar Dual Inhibitors for Wild Type and L1196M Mutant of Anaplastic Lymphoma Kinase through Structure-Based Virtual Screening

Discovery of MEK/PI3K dual inhibitor via structure-based virtual screening.

Discovery of fluorescent 3-heteroarylcoumarin derivatives as novel inhibitors of anaplastic lymphoma kinase

Discovery of new aminopyrimidine-based phosphoinositide 3-kinase beta (PI3Kβ) inhibitors with selectivity over PI3Kα.

Discovery of new azaindole-based PI3Kα inhibitors: Apoptotic and antiangiogenic effect on cancer cells ⬇️

Discovery of new benzothiazole-based inhibitors of breakpoint cluster region-Abelson kinase including the T315I mutant.

Discovery of picomolar ABL kinase inhibitors equipotent for wild type and T315I mutant via structure-based de novo design

Discovery of wrightiadione as a novel template for the TrkA kinase inhibitors

Efficient synthesis of frutinone A and its derivatives through palladium-catalyzed C - H activation/carbonylation.

Fascaplysin Exerts Anti-Cancer Effects through the Downregulation of Survivin and HIF-1α and Inhibition of VEGFR2 and TRKA.

Fluorescent phosphoinositide 3-kinase inhibitors suitable for monitoring of intracellular distribution

Frontispiece: Visible‐Light‐Induced Cysteine‐Specific Bioconjugation: Biocompatible Thiol–Ene Click Chemistry

Frontispiz: Visible‐Light‐Induced Cysteine‐Specific Bioconjugation: Biocompatible Thiol–Ene Click Chemistry

Functionalization of Pyridinium Derivatives with 1,4-Dihydropyridines Enabled by Photoinduced Charge Transfer

HS-104, a PI3K inhibitor, enhances the anticancer efficacy of gemcitabine in pancreatic cancer.

HS-116, a novel phosphatidylinositol 3-kinase inhibitor induces apoptosis and suppresses angiogenesis of hepatocellular carcinoma through inhibition of the PI3K/AKT/mTOR pathway

HS-133, a novel fluorescent phosphatidylinositol 3-kinase inhibitor as a potential imaging and anticancer agent for targeted therapy

HS-1371, a novel kinase inhibitor of RIP3-mediated necroptosis

HS-173 as a novel inducer of RIP3-dependent necroptosis in lung cancer

HS-173, a novel PI3K inhibitor suppresses EMT and metastasis in pancreatic cancer

HS-173, a novel PI3K inhibitor, attenuates the activation of hepatic stellate cells in liver fibrosis

HS-173, a novel phosphatidylinositol 3-kinase (PI3K) inhibitor, has anti-tumor activity through promoting apoptosis and inhibiting angiogenesis

HS-438, a new inhibitor of imatinib-resistant BCR-ABL T315I mutation in chronic myeloid leukemia

HS-543 induces apoptosis of Imatinib-resistant chronic myelogenous leukemia with T315I mutation

HS‑146, a novel phosphoinositide 3‑kinase α inhibitor, induces the apoptosis and inhibits the metastatic ability of human breast cancer cells

High-throughput chemical screening to discover new modulators of microRNA expression in living cells by using graphene-based biosensor.

IPD-196, a novel phosphatidylinositol 3-kinase inhibitor with potent anticancer activity against hepatocellular carcinoma

Identification of 4-Phenoxyquinoline Based Inhibitors for L1196M Mutant of Anaplastic Lymphoma Kinase by Structure-Based Design.

Identification of common inhibitors of wild-type and T315I mutant of BCR-ABL through the parallel structure-based virtual screening.

Identification of lead small molecule inhibitors of glycogen synthase kinase-3 beta using a fragment-linking strategy

Identification of novel BRAF kinase inhibitors with structure-based virtual screening

Identification of novel inhibitors of tropomyosin-related kinase A through the structure-based virtual screening with homology-modeled protein structure

Identification of β-Lapachone Analogs as Novel MALT1 Inhibitors To Treat an Aggressive Subtype of Diffuse Large B-Cell Lymphoma

Induction of apoptosis and suppression of angiogenesis of hepatocellular carcinoma by HS-159, a novel phosphatidylinositol 3-kinase inhibitor

Kinase and GPCR polypharmacological approach for the identification of efficient anticancer medicines

Metal-Free, Visible-Light-Induced Remote C(sp3)-H Pyridylation via Radical Translocation of N-Alkoxypyridinium Salts

NiH-Catalyzed Proximal-Selective Hydroamination of Unactivated Alkenes

Nocodazole is a high-affinity ligand for the cancer-related kinases ABL, c-KIT, BRAF, and MEK.

One-pot catalysis of dehydrogenation of cyclohexanones to phenols and oxidative Heck coupling: expedient synthesis of coumarins

Optimization and biological evaluation of aminopyrimidine-based IκB kinase β inhibitors with potent anti-inflammatory effects

Palladium(II)-Catalyzed Tandem Synthesis of Acenes Using Carboxylic Acids as Traceless Directing Groups

Palladium(II)-catalyzed direct intermolecular alkenylation of chromones

Palladium-Catalyzed Divergent Arylation of Triazolopyridines: A Computational Study

Palladium-catalyzed dehydrogenation/oxidative cross-coupling sequence of β-heteroatom-substituted ketones

Photocatalytic Vicinal Aminopyridylation of Methyl Ketones by a Double Umpolung Strategy

Photochemical Carbopyridylation of Alkenes Using N-Alkenoxypyridinium Salts as Bifunctional Reagents

Rational Computational Design of Fourth-Generation EGFR Inhibitors to Combat Drug-Resistant Non-Small Cell Lung Cancer

Reactivity of Morita-Baylis-Hillman Adducts in C-H Functionalization of (Hetero)aryl Nitrones: Access to Bridged Cycles and Carbazoles

Regiodivergent Ring-Opening Cross-Coupling of Vinyl Aziridines with Phosphorus Nucleophiles: Access to Phosphorus-Containing Amino Acid Derivatives

Regioselective C-H Functionalization of Heteroarene N-Oxides Enabled by a Traceless Nucleophile

Regioselective palladium-catalyzed direct cross-coupling of coumarins with simple arenes

Regioselective palladium-catalyzed olefination of coumarins via aerobic oxidative Heck reactions