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List of works by Robert N Young

5 Discovery of Montelukast: a Once-a-Day Oral Antagonist of Leukotriene D4 for the Treatment of Chronic Asthma

scientific article published on January 1, 2001

A new quinoline-based chemical probe inhibits the autophagy-related cysteine protease ATG4B

scientific article published in Scientific Reports

Cheminformatics-Driven Discovery of Selective, Nanomolar Inhibitors for Staphylococcal Pyruvate Kinase ⬇️

scientific article published on November 21, 2011

Design and synthesis of novel bone-targeting dual-action pro-drugs for the treatment and reversal of osteoporosis ⬇️

scientific article published on January 31, 2012

Design, Synthesis, and Pharmacokinetics of a Bone-Targeting Dual-Action Prodrug for the Treatment of Osteoporosis.

scientific article

Determination of the rat in vivo pharmacokinetic profile of a bone-targeting dual-action pro-drug for treatment of osteoporosis

scientific article published on 15 May 2015

Development of 2,3-dihydro-6-(3-phenoxypropyl)-2-(2-phenylethyl)-5-benzofuranol (L-670,630) as a potent and orally active inhibitor of 5-lipoxygenase

scientific article published on April 3, 1992

Development of fluorescent peptide substrates and assays for the key autophagy-initiating cysteine protease enzyme, ATG4B.

scientific article published on 28 April 2015

Development of fluorescent substrates and assays for the key autophagy-related cysteine protease enzyme, ATG4B.

scientific article published on April 2014

Difluoroethylamines as an amide isostere in inhibitors of cathepsin K ⬇️

scientific article published on December 19, 2010

Discovery and optimization of a new class of pyruvate kinase inhibitors as potential therapeutics for the treatment of methicillin-resistant Staphylococcus aureus infections

scientific article published on 24 January 2014

Discovery of MK-0952, a selective PDE4 inhibitor for the treatment of long-term memory loss and mild cognitive impairment ⬇️

scientific article published on September 21, 2010

Erratum: Corrigendum: The promise and peril of chemical probes

scientific article published in November 2015

Inhibition of Autophagosome Formation by the Benzoporphyrin Derivative Verteporfin ⬇️

scientific article published on December 30, 2010

Optimization and structure–activity relationships of a series of potent inhibitors of methicillin-resistant Staphylococcus aureus (MRSA) pyruvate kinase as novel antimicrobial agents ⬇️

scientific article published on October 17, 2012

Precision autophagy: Will the next wave of selective autophagy markers and specific autophagy inhibitors feed clinical pipelines?

scientific article

Preparation and analgesic properties of amino acid derivatives of (-)-5,9.alpha.-diethyl-2'-hydroxybenzomorphan ⬇️

scientific article published on 01 November 1981

Stereoselective Total Synthesis of (±)-Thielocin Alβ ⬇️

scientific article published on November 21, 2001

Substituted (Pyridylmethoxy)naphthalenes as Potent and Orally Active 5-Lipoxygenase Inhibitors: Synthesis, Biological Profile, and Pharmacokinetics of L-739,010 ⬇️

scientific article published on August 29, 1997

Substituted 2-Pyridinemethanol derivatives as potent and selective phosphodiesterase-4 inhibitors ⬇️

scientific article published on June 2, 2003

Targeting the Binding Function 3 (BF3) Site of the Androgen Receptor Through Virtual Screening. 2. Development of 2-((2-phenoxyethyl) thio)-1H-benzimidazole Derivatives ⬇️

scientific article published on January 18, 2013

The promise and peril of chemical probes

scientific article

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