List of works - Douglas J Kojetin

1H, 13C and 15N chemical shift assignments for the human Pitx2 homeodomain in complex with a 22-base hairpin DNA ⬇️

scientific article published on August 5, 2011

A molecular switch regulating transcriptional repression and activation of PPARγ

scientific article published on 19 February 2020

A structural mechanism for directing corepressor-selective inverse agonism of PPARγ

scientific article published in Nature Communications

Assessment of NR4A Ligands That Directly Bind and Modulate the Orphan Nuclear Receptor Nurr1

scientific article published on 08 December 2020

CAR directs T cell adaptation to bile acids in the small intestine

scientific article published on 07 April 2021

Characterization of the Core Mammalian Clock Component, NPAS2, as a REV-ERBα/RORα Target Gene ⬇️

scientific article published on September 3, 2010

Chemical systems biology reveals mechanisms of glucocorticoid receptor signaling

scientific article published on 28 January 2021

Cooperative cobinding of synthetic and natural ligands to the nuclear receptor PPARγ

scientific article published on 21 December 2018

DNA binding alters coactivator interaction surfaces of the intact VDR–RXR complex ⬇️

scientific article published on April 10, 2011

Defining a conformational ensemble that directs activation of PPARγ.

scientific article

Modification of the Orthosteric PPARγ Covalent Antagonist Scaffold Yields an Improved Dual-Site Allosteric Inhibitor.

scientific article published on 06 February 2017

Observing selected domains in multi-domain proteins via sortase-mediated ligation and NMR spectroscopy ⬇️

scientific article published on December 29, 2010

Regulation of p53 Stability and Apoptosis by a ROR Agonist ⬇️

scientific article published on April 11, 2012

Small Molecule Modulation of Nuclear Receptor Conformational Dynamics: Implications for Function and Drug Discovery ⬇️

scientific article published on August 6, 2012

Structural Basis of Altered Potency and Efficacy Displayed by a Major in Vivo Metabolite of the Antidiabetic PPARγ Drug Pioglitazone

scientific article published on 07 February 2019

Structural organization of a major neuronal G protein regulator, the RGS7-Gβ5-R7BP complex

scientific article published on 12 December 2018

Sub‐classification of response regulators using the surface characteristics of their receiver domains ⬇️

scientific article published on November 20, 2003

The REV-ERBs and RORs: Molecular Links Between Circadian Rhythms and Lipid Homeostasis ⬇️

scientific article published on April 1, 2011

List of works by Douglas J Kojetin