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List of works by Jesús Alcázar

Alcohol-alcohol cross-coupling enabled by S <sub>H</sub> 2 radical sorting

scientific article published on 21 March 2024

Discovery of VU0409551/JNJ-46778212: An mGlu5 Positive Allosteric Modulator Clinical Candidate Targeting Schizophrenia

scientific article published on 20 May 2015

Flow chemistry as a tool to access novel chemical space for drug discovery

scientific article published on 21 August 2020

Formation of quaternary carbons through cobalt-catalyzed C(sp3)-C(sp3) Negishi cross-coupling

scientific article published on 18 June 2020

Grignard Reagents on a Tab: Direct Magnesium Insertion under Flow Conditions

scientific article published on 28 June 2017

On-demand synthesis of organozinc halides under continuous flow conditions.

scientific article

Photoinduced Palladium-Catalyzed Negishi Cross-Couplings Enabled by the Visible-Light Absorption of Palladium-Zinc Complexes

scientific article published on 10 September 2018

Preliminary investigation of 6,7-dihydropyrazolo[1,5-a]pyrazin-4-one derivatives as a novel series of mGlu5 receptor positive allosteric modulators with efficacy in preclinical models of schizophrenia

scientific article published on 28 November 2015

Recent Applications of Microwave Irradiation to Medicinal Chemistry

scientific article published on February 1, 2010

Scalability of Visible-Light-Induced Nickel Negishi Reactions: A Combination of Flow Photochemistry, Use of Solid Reagents, and In-Line NMR Monitoring

scientific article published on 26 October 2018

Selective Synthesis of 2-, 4-, and 5-Cyano Substituted Imidazoles from Imidazole N-Oxides and Trimethylsilyl Cyanide

scientific article published on 01 October 1996

Synthesis and structure–activity relationship of 2-(aminoalkyl)-2,3,3a,8-tetrahydrodibenzo[c,f]isoxazolo[2,3-a]azepine derivatives: a novel series of 5-HT2A/2C receptor antagonists. Part 1

scientific article published on January 21, 2002

Synthesis, In Vivo Occupancy, and Radiolabeling of Potent Phosphodiesterase Subtype-10 Inhibitors as Candidates for Positron Emission Tomography Imaging

scientific article published on August 2, 2011

Visible-Light-Induced Nickel-Catalyzed Negishi Cross-Couplings by Exogenous-Photosensitizer-Free Photocatalysis.

scientific article published on 22 March 2018