List of works - Paola B Arimondo

Assembly of the Entire Carbon Backbone of a Stereoisomer of the Antitumor Marine Natural Product Hemicalide

scientific article published on 25 January 2019

Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic 'writers'

scientific article published on 17 September 2020

Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs

scientific article published on 06 April 2020

C5-DNA methyltransferase inhibitors: from screening to effects on zebrafish embryo development.

scientific article

Demethylation by low-dose 5-aza-2'-deoxycytidine impairs 3D melanoma invasion partially through miR-199a-3p expression revealing the role of this miR in melanoma

scientific article published on 16 January 2019

Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation

scientific article published in March 2014

Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors

scientific article published on 01 June 2018

Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells

scientific article published on 06 May 2019

Identification of novel inhibitors of DNA methylation by screening of a chemical library.

scientific article

Mechanistic insights on the inhibition of c5 DNA methyltransferases by zebularine

scientific article

Properly substituted analogues of BIX-01294 lose inhibition of G9a histone methyltransferase and gain selective anti-DNA methyltransferase 3A activity

scientific article

Rapid synthesis of new DNMT inhibitors derivatives of procainamide

scientific article

Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells.

scientific article

Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells

scientific article published on 15 January 2014

Synthesis and evaluation of analogues of N-phthaloyl-l-tryptophan (RG108) as inhibitors of DNA methyltransferase 1.

scientific article published on 9 January 2014

The DNMT3A R882H mutant displays altered flanking sequence preferences.

scientific article published on 6 March 2018

The past and presence of gene targeting: from chemicals and DNA via proteins to RNA.

scientific article published in June 2018

Wandering along the epigenetic timeline

scientific article published on 02 July 2020

List of works by Paola B Arimondo

Assembly of the Entire Carbon Backbone of a Stereoisomer of the Antitumor Marine Natural Product Hemicalide

Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic 'writers'

Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs

C5-DNA methyltransferase inhibitors: from screening to effects on zebrafish embryo development.

Demethylation by low-dose 5-aza-2'-deoxycytidine impairs 3D melanoma invasion partially through miR-199a-3p expression revealing the role of this miR in melanoma

Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation

Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors

Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells

Identification of novel inhibitors of DNA methylation by screening of a chemical library.

Mechanistic insights on the inhibition of c5 DNA methyltransferases by zebularine

Properly substituted analogues of BIX-01294 lose inhibition of G9a histone methyltransferase and gain selective anti-DNA methyltransferase 3A activity

Rapid synthesis of new DNMT inhibitors derivatives of procainamide

Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells.

Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells

Synthesis and evaluation of analogues of N-phthaloyl-l-tryptophan (RG108) as inhibitors of DNA methyltransferase 1.

The DNMT3A R882H mutant displays altered flanking sequence preferences.

The past and presence of gene targeting: from chemicals and DNA via proteins to RNA.

Wandering along the epigenetic timeline