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List of works by Salvatore Santamaria

ADAMTS-5: A difficult teenager turning 20

scientific article published on 27 March 2020

Arylsulfonamide inhibitors of aggrecanases as potential therapeutic agents for osteoarthritis: synthesis and biological evaluation

scientific article

Design, Synthesis, Biological Evaluation, and NMR Studies of a New Series of Arylsulfones As Selective and Potent Matrix Metalloproteinase-12 Inhibitors

article by Elisa Nuti et al published 22 October 2009 in Journal of Medicinal Chemistry

Identification of novel molecular scaffolds for the design of MMP-13 inhibitors: A first round of lead optimization

article

Monoclonal antibodies against metzincin targets.

scientific article published on 27 February 2018

N-O-Isopropyl Sulfonamido-Based Hydroxamates: Design, Synthesis and Biological Evaluation of Selective Matrix Metalloproteinase-13 Inhibitors as Potential Therapeutic Agents for Osteoarthritis

article

N-O-Isopropyl sulfonamido-based hydroxamates: Kinetic characterisation of a series of MMP-12/MMP-13 dual target inhibitors

scientific article published in 2012

Novel 1-hydroxypiperazine-2,6-diones as new leads in the inhibition of metalloproteinases.

scientific article published on 17 November 2011

Novel folate-hydroxamate based antimetabolites: synthesis and biological evaluation

scientific article published on July 2011

Potent arylsulfonamide inhibitors of tumor necrosis factor-alpha converting enzyme able to reduce activated leukocyte cell adhesion molecule shedding in cancer cell models

scientific article

Proteomic discovery of substrates of the cardiovascular protease ADAMTS7

scientific article published on 29 March 2019

Selective arylsulfonamide inhibitors of ADAM-17: hit optimization and activity in ovarian cancer cell models

scientific article published on 4 October 2013

Synthesis and biological evaluation in U87MG glioma cells of (ethynylthiophene)sulfonamido-based hydroxamates as matrix metalloproteinase inhibitors

scientific article published on 2 April 2011