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List of works by Holger Stark

Antinociceptive effects of novel histamine H3 R and H4 R receptor antagonists and their influence on morphine analgesia of neuropathic pain in the mouse.

scientific article published on 27 February 2018

Binding kinetics of cariprazine and aripiprazole at the dopamine D receptor

scientific article published in Scientific Reports

Biphenylalkoxyamine Derivatives-Histamine H Receptor Ligands with Butyrylcholinesterase Inhibitory Activity

scientific article published on 11 June 2021

From medicinal plant extracts to defined chemical compounds targeting the histamine H4 receptor: Curcuma longa in the treatment of inflammation.

scientific article published on 24 June 2017

Guanidine Derivatives: How Simple Structural Modification of Histamine H<sub>3</sub>R Antagonists Has Led to the Discovery of Potent Muscarinic M<sub>2</sub>R/M<sub>4</sub>R Antagonists

scientific article published on 08 June 2021

Histamine H3 receptor ligands by hybrid virtual screening, docking, molecular dynamics simulations, and investigation of their biological effects

scientific article published on 24 January 2019

Human β-Defensin 2 Expression in Oral Epithelium: Potential Therapeutic Targets in Oral Lichen Planus ⬇️

scientific article published on 10 April 2019

In silico and in vitro studies of two non-imidazole multiple targeting agents at histamine H3 receptors and cholinesterase enzymes

scientific article published on 12 November 2019

Morpholino Analogues of Fingolimod as Novel and Selective S1P1 Ligands with In Vivo Efficacy in a Mouse Model of Experimental Antigen-Induced Encephalomyelitis

scientific article published on 04 September 2020

Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H3 R Antagonism for Neurodegenerative Diseases.

scientific article published in September 2017

Reversible Small Molecule Inhibitors of MAO A and MAO B with Anilide Motifs

scientific article published on 28 January 2020

Role of Histamine H₃ Receptor Antagonists on Intraocular Pressure Reduction in Rabbit Models of Transient Ocular Hypertension and Glaucoma

scientific article published on 24 February 2019

Simultaneous Blockade of Histamine H3 Receptors and Inhibition of Acetylcholine Esterase Alleviate Autistic-Like Behaviors in BTBR T+ tf/J Mouse Model of Autism

scientific article published on 28 August 2020

Studies on Anticonvulsant Effects of Novel Histamine H3R Antagonists in Electrically and Chemically Induced Seizures in Rats

scientific article published on 29 October 2018

Substituted Purines as High-Affinity Histamine H<sub>3</sub> Receptor Ligands

scientific article published on 04 May 2022

The Dual-Active Histamine H3 Receptor Antagonist and Acetylcholine Esterase Inhibitor E100 Alleviates Autistic-Like Behaviors and Oxidative Stress in Valproic Acid Induced Autism in Mice

scientific article published on 03 June 2020

The chemical probe - scopes, limitations and challenges

scientific article published on 19 June 2020

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