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List of works by Hiroaki Ohno

A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase ⬇️

scientific article published on July 7, 2011

Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants

article

Affinity-based screening of MDM2/MDMX–p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors ⬇️

scientific article published on May 15, 2013

Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group

scientific article published on 13 October 2009

Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins

scientific article published on 15 September 2009

Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles

scientific article

Construction of Quaternary Carbon Stereocenter of α-Tertiary Amine through Remote C-H Functionalization of Tris Derivatives: Enantioselective Total Synthesis of Myriocin

scientific article published on 09 July 2019

Construction of the Pyrrolo[2,3-d]carbazole Core of Spiroindoline Alkaloids by Gold-Catalyzed Cascade Cyclization of Ynamide

scientific article published on 17 June 2019

Correction to Construction of the Pyrrolo[2,3-d]carbazole Core of Spiroindoline Alkaloids by Gold-Catalyzed Cascade Cyclization of Ynamide

scientific article published on 13 February 2020

Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182.

scientific article published on 16 January 2013

Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus

scientific article published on 6 June 2009

Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity

scientific article published on 16 January 2008

Development and application of fluorescent SDF-1 derivatives

scientific article published on May 2012

Development of Aziridination and Azetizination Reactions of Amino Allenes Using a Palladium Catalyst ⬇️

scientific article published on October 1, 2001

Development of Mirror-Image Screening Systems for XIAP BIR3 Domain Inhibitors

scientific article published on 17 April 2019

Development of a novel fusion inhibitor against T-20-resistant HIV-1.

scientific article published in January 2009

Direct synthesis of aryl-annulated [c]carbazoles by gold(i)-catalysed cascade reaction of azide-diynes and arenes

scientific article published on 10 September 2018

Double CH Functionalization in Sequential Order: Direct Synthesis of Polycyclic Compounds by a Palladium‐Catalyzed CH Alkenylation–Arylation Cascade ⬇️

scientific article published on March 15, 2012

Enhanced Plasmid DNA Transfer into Tumor Cells by Nanoparticle Composed of Cholesteryl Triamine and Diamine ⬇️

scientific article published on January 1, 2013

First Palladium-Catalyzed Aziridination Reaction of Amino Allenes ⬇️

scientific article published on April 30, 1999

Gold(I)-Catalyzed Cascade Cyclization Reactions of Allenynes for the Synthesis of Fused Cyclopropanes and Acenaphthenes

scientific article published on 06 May 2019

Gold(I)-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring-Fused Indoles and Propellane-Type Indolines

scientific article published on 22 January 2020

Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds

scientific article published on 23 July 2018

Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold.

scientific article

Gold-Catalyzed Three-Component Annulation: Efficient Synthesis of Highly Functionalized Dihydropyrazoles from Alkynes, Hydrazines, and Aldehydes or Ketones ⬇️

scientific article published on December 16, 2011

Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold

scientific article published on 16 February 2015

Identification of minimal sequence for HIV-1 fusion inhibitors

scientific article published on 10 September 2008

Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach

scientific article published on 29 May 2008

Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds

scientific article published on April 2015

Maternal gut microbiota in pregnancy influences offspring metabolic phenotype in mice

scientific article published on 01 February 2020

Palladium(0)-Catalyzed Isomerization Reactions of Aziridines Bearing an α,β-Unsaturated Ester Group: A Thermodynamic Preference for Chiral Alkyl (2E)-4,5-cis-4,5-Epimino-N-(alkyl- or arylsulfonyl) 2-Enoates over the Other Three Stereoisomers ⬇️

scientific article published on 01 May 1997

Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: synthesis and bioevaluation of alpha-helical anti-HIV peptide analogues

scientific article

Potent CXCR4 antagonists containing amidine type Peptide bond isosteres

scientific article published on 28 March 2011

Reactions of N-Arylsulfonyl-2,3-cis- and N-Arylsulfonyl-2,3-trans-3-alkyl-2-vinylaziridines with Organocopper Reagents: Importance of 2,3-cis-Stereochemistry in Controlling Regio- and Stereoselectivity ⬇️

scientific article published on 01 October 1998

Samarium(II)-Promoted Radical Spirocyclization onto an Aromatic Ring ⬇️

scientific article published on 01 October 2003

Structure-Based Design of Novel Potent Protein Kinase CK2 (CK2) Inhibitors with Phenyl-azole Scaffolds ⬇️

scientific article published on March 7, 2012

Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents

scientific article published on 19 June 2013

Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents

scientific article

Structure–Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3)

scientific article published on 12 April 2018

Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4.

scientific article

Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres

scientific article

Synthesis of Triazolo- and Oxadiazolopiperazines by Gold(I)-Catalyzed Domino Cyclization: Application to the Design of a Mitogen Activated Protein (MAP) Kinase Inhibitor

scientific article published on 31 December 2018

Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide–Polyketide Macrocycle

scientific article published on 27 February 2018

Total Synthesis of Dictyodendrins A-F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole

scientific article published on 09 August 2020

Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles

scientific article published on 31 May 2017

Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle.

scientific article published on 10 April 2018

X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution

scientific article

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