List of works - Arun K Ghosh

A Photochemical Route to Optically Active Hexahydro-4H-furopyranol, a High-Affinity P2 Ligand for HIV-1 Protease Inhibitors

scientific article published on 16 July 2019

Copper-Catalyzed Stille Cross-Coupling Reaction and Application in the Synthesis of the Spliceostatin Core Structure

scientific article published on 09 June 2020

Design and Development of Highly Potent HIV-1 Protease Inhibitors with a Crown-Like Oxotricyclic Core as the P2-Ligand To Combat Multidrug-Resistant HIV Variants.

scientific article published on 18 April 2017

Design and Synthesis of Highly Potent HIV-1 Protease Inhibitors Containing Tricyclic Fused Ring Systems as Novel P2 Ligands: Structure-Activity Studies, Biological and X-ray Structural Analysis.

scientific article published on 15 May 2018

Design and Synthesis of Potent HIV-1 Protease Inhibitors Containing Bicyclic Oxazolidinone Scaffold as the P2 Ligands: Structure-Activity Studies and Biological and X-ray Structural Studies

article

Design and synthesis of herboxidiene derivatives that potently inhibit in vitro splicing

scientific article published on 01 February 2021

Design of Highly Potent, Dual Acting and Central Nervous System Penetrating HIV-1 Protease Inhibitors with Excellent Potency against Multidrug-Resistant HIV-1 Variants.

scientific article published on 13 February 2018

Design, Synthesis, Biological Evaluation, and X-ray Studies of HIV-1 Protease Inhibitors with Modified P2' Ligands of Darunavir

scientific article published on 6 November 2017

Development of an Efficient Enzyme Production and Structure-Based Discovery Platform for BACE1 Inhibitors

scientific article published on 22 October 2019

Differentiating Isomeric Deprotonated Glucuronide Drug Metabolites via Ion/Molecule Reactions in Tandem Mass Spectrometry

scientific article published on 23 July 2018

Enantioselective Synthesis of Spliceostatin G and Evaluation of Bioactivity of Spliceostatin G and Its Methyl Ester.

scientific article published on 8 December 2017

Enantioselective Synthesis of Thailanstatin A Methyl Ester and Evaluation of in Vitro Splicing Inhibition

scientific article published on 26 April 2018

Enantioselective Synthesis of a Cyclopropane Derivative of Spliceostatin A and Evaluation of Bioactivity

scientific article published on 05 November 2018

Enantioselective Total Syntheses of (+)-Fendleridine and (+)-Acetylaspidoalbidine

scientific article published on 02 April 2019

Enantioselective Total Synthesis of (+)-Monocerin, a Dihydroisocoumarin Derivative with Potent Antimalarial Properties

scientific article published on 29 April 2019

Fluorescent Probes for Monitoring Serine Ubiquitination

scientific article published on 27 March 2020

Herboxidiene Features That Mediate Conformation-Dependent SF3B1 Interactions to Inhibit Splicing

scientific article published on 22 February 2021

Highly Selective and Potent Human β-Secretase 2 (BACE2) Inhibitors against Type 2 Diabetes: Design, Synthesis, X-ray Structure and Structure-Activity Relationship Studies

scientific article published on 05 February 2019

Lewis Acid-Catalyzed Vinyl Acetal Rearrangement of 4,5-Dihydro-1,3-dioxepines: Stereoselective Synthesis of cis- and trans-2,3-Disubstituted Tetrahydrofurans

scientific article published on 05 August 2020

Potent HIV-1 Protease Inhibitors Containing Carboxylic and Boronic Acids: Effect on Enzyme Inhibition and Antiviral Activity and Protein-Ligand X-ray Structural Studies

scientific article published on 04 October 2019

Structure-Based Design of Highly Potent HIV-1 Protease Inhibitors Containing New Tricyclic Ring P2-Ligands: Design, Synthesis, Biological, and X-ray Structural Studies

scientific article published on 29 April 2020

The Chiron Approach to (3R,3aS,6aR)-Hexahydrofuro[2,3-b]furan-3-ol, a Key Subunit of HIV-1 Protease Inhibitor Drug, Darunavir

scientific article published on 03 December 2020

The Curtius Rearrangement: Applications in Modern Drug Discovery and Medicinal Chemistry

scientific article published on 11 October 2018

The Curtius rearrangement: mechanistic insight and recent applications in natural product syntheses

scientific article published on 26 February 2018

Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry

scientific article published on 02 December 2019

List of works by Arun K Ghosh