List of works - Martin D Eastgate

A Mild, Functional Group Tolerant Addition of Organozinc Nucleophiles to N-Activated Quinolines and Isoquinolines

scientific article published on 15 August 2017

An Enantioselective Total Synthesis of (+)-Duocarmycin SA.

scientific article published on 20 March 2018

C-H Arylation in the Formation of a Complex Pyrrolopyridine, the Commercial Synthesis of the Potent JAK2 Inhibitor, BMS-911543

scientific article published on 12 November 2018

Directed, Palladium(II)-Catalyzed Intermolecular Aminohydroxylation of Alkenes Using a Mild Oxidation System

scientific article published on 11 June 2018

Effects of Multiple Catalyst Deactivation Pathways and Continuous Ligand Recycling on the Kinetics of Pd-Catalyzed C-N Coupling Reactions

scientific article published on 24 October 2018

Enantiodivergent Formation of C-P Bonds: Synthesis of P-Chiral Phosphines and Methylphosphonate Oligonucleotides

scientific article published on 16 March 2020

Inhibitors of HIV-1 Attachment: The Discovery and Development of Temsavir and its Prodrug Fostemsavir

scientific article published on 22 December 2017

Leveraging a "Catch-Release" Logic Gate Process for the Synthesis and Nonchromatographic Purification of Thioether- or Amine-Bridged Macrocyclic Peptides.

scientific article published on 14 March 2018

Ligand-Enabled Pd(II)-Catalyzed C(sp3)-H Lactonization Using Molecular Oxygen as Oxidant

scientific article published on 24 April 2020

Ni(COD)(DQ): An Air-Stable 18-Electron Nickel(0)-Olefin Precatalyst

scientific article published on 17 February 2020

Nickel-Catalyzed 1,2-Diarylation of Simple Alkenyl Amides

scientific article published on 17 December 2018

Overcoming the Limitations of γ- and δ-C-H Arylation of Amines through Ligand Development

scientific article published on 14 December 2018

Strategy To Prepare 3-Bromo- and 3-Chloropyrazoles.

scientific article published on 11 February 2018

Synthesis of 2'-Methyl-6-methoxyguanosine from the Parent Ribonucleoside Guanosine

scientific article published on 11 October 2018

Unlocking P(V): Reagents for chiral phosphorothioate synthesis.

scientific article

Utilizing Native Directing Groups: Mechanistic Understanding of a Direct Arylation Leads to Formation of Tetracyclic Heterocycles via Tandem Intermolecular, Intramolecular C-H Activation

scientific article published on 04 June 2019

Zinc Acetate-Promoted Buchwald-Hartwig Couplings of Heteroaromatic Amines