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List of works by Stefan Geschwindner

Agonists and Antagonists of Protease-Activated Receptor 2 Discovered within a DNA-Encoded Chemical Library Using Mutational Stabilization of the Target

scientific article published on 09 January 2018

Avidity-Based Affinity Enhancement Using Nanoliposome-Amplified SPR Sensing Enables Low Picomolar Detection of Biologically Active Neuregulin 1

scientific article published on 27 November 2019

Discovery of a Novel Oral Glucocorticoid Receptor Modulator (AZD9567) with Improved Side Effect Profile.

scientific article published on 9 February 2018

Fragments as Novel Starting Points for tRNA-Guanine Transglycosylase Inhibitors Found by Alternative Screening Strategies

scientific article published on 29 January 2020

Harnessing the Versatility of Optical Biosensors for Target-Based Small-Molecule Drug Discovery

scientific article

Hot-Spotting with Thermal Scanning: A Ligand- and Structure-Independent Assessment of Target Ligandability.

scientific article

Mining Natural Products for Macrocycles to Drug Difficult Targets

scientific article published on 18 December 2020

Perspectives on optical biosensor utility in small-molecule screening

scientific article

Regenerable Biosensors for Small-Molecule Kinetic Characterization Using SPR

scientific article published on 08 December 2020

The current impact of water thermodynamics for small-molecule drug discovery

scientific article published on 10 September 2019

X-ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors

scientific article published on 8 November 2017