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List of works by Christopher J Helal

A platform for automated nanomole-scale reaction screening and micromole-scale synthesis in flow.

scientific article

Correction to Application of Structure-Based Design and Parallel Chemistry to Identify a Potent, Selective, and Brain Penetrant Phosphodiesterase 2A Inhibitor

scientific article published on 06 April 2018

Discovery and Lead Optimization of Atropisomer D1 Agonists with Reduced Desensitization

scientific article published on 11 December 2018

Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation.

scientific article published on 2 March 2018

High-Throughput Ligand Screening Enables the Enantioselective Conjugate Borylation of Cyclobutenones to Access Synthetically Versatile Tertiary Cyclobutylboronates

scientific article published on 31 October 2019

Identification of a Potent, Highly Selective, and Brain Penetrant Phosphodiesterase 2A Inhibitor Clinical Candidate.

scientific article published on 2 January 2018

Introduction of a Crystalline, Shelf-Stable Reagent for the Synthesis of Sulfur(VI) Fluorides

scientific article published on 12 January 2018

Parallel Synthesis of 1H-Pyrazolo[3,4-d]pyrimidines via Condensation of N-Pyrazolylamides and Nitriles.

scientific article published on 6 October 2017

Ru/Ni Dual Catalytic Desulfinative Photoredox Csp2-Csp3 Cross-Coupling of Alkyl Sulfinate Salts and Aryl Halides

scientific article published on 28 November 2017

Synthetic Approaches to the New Drugs Approved During 2017

scientific article published on 15 April 2019

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