List of works - Artur Świerczek

A Novel, Pan-PDE Inhibitor Exerts Anti-Fibrotic Effects in Human Lung Fibroblasts via Inhibition of TGF-β Signaling and Activation of cAMP/PKA Signaling

scientific article published on 03 June 2020

A new class of 5-HT 1A receptor antagonists with procognitive and antidepressant properties

scientific article published in September 2021

Advances in Discovery of PDE10A Inhibitors for CNS-Related Disorders. Part 1: Overview of the Chemical and Biological Research

scientific article published on 01 January 2019

Advances in the Discovery of PDE10A Inhibitors for CNS-Related Disorders. Part 2: Focus on Schizophrenia

scientific article published on 01 January 2019

Comparative Assessment of the New PDE7 Inhibitor - GRMS-55 and Lisofylline in Animal Models of Immune-Related Disorders: A PK/PD Modeling Approach

scientific article published on 02 January 2020

Correction to: Comparative Assessment of the New PDE7 Inhibitor - GRMS-55 and Lisofylline in Animal Models of Immune-Related Disorders: A PK/PD Modeling Approach

scientific article published on 21 January 2020

Design and Synthesis of Novel Aminoalkanamides Targeting Neurodegeneration and Symptoms of Alzheimer’s Disease

scientific article published on 17 September 2021

Influence of inflammatory disorders on pharmacokinetics of lisofylline in rats: implications for studies in humans

scientific article published on 11 December 2018

New imidazopyridines with phosphodiesterase 4 and 7 inhibitory activity and their efficacy in animal models of inflammatory and autoimmune diseases

scientific article published on 19 September 2020

Novel amide derivatives of 1,3-dimethyl-2,6-dioxopurin-7-yl-alkylcarboxylic acids as multifunctional TRPA1 antagonists and PDE4/7 inhibitors: A new approach for the treatment of pain

scientific article published on 10 September 2018

Novel anilide and benzylamide derivatives of arylpiperazinylalkanoic acids as 5-HT1A/5-HT7 receptor antagonists and phosphodiesterase 4/7 inhibitors with procognitive and antidepressant activity

scientific article published on 17 June 2020

Novel butanehydrazide derivatives of purine-2,6-dione as dual PDE4/7 inhibitors with potential anti-inflammatory activity: Design, synthesis and biological evaluation.

scientific article published on 27 January 2018

Novel phosphodiesterases inhibitors from the group of purine-2,6-dione derivatives as potent modulators of airway smooth muscle cell remodelling

scientific article published on 06 November 2019

PDE7-Selective and Dual Inhibitors: Advances in Chemical and Biological Research.

scientific article published on 16 January 2017

PK/PD Modeling of the PDE7 Inhibitor-GRMS-55 in a Mouse Model of Autoimmune Hepatitis

scientific article published on 21 April 2021

PK/PD studies on non-selective PDE inhibitors in rats using cAMP as a marker of pharmacological response.

scientific article

Physiologically based modeling of lisofylline pharmacokinetics following intravenous administration in mice

scientific article published on 08 February 2015

List of works by Artur Świerczek