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List of works by Bruno Cerra

Beyond bile acids: targeting Farnesoid X Receptor (FXR) with natural and synthetic ligands

scientific article

Bile acid derivatives as ligands of the farnesoid x receptor: molecular determinants for bile acid binding and receptor modulation.

scientific article published in January 2014

Binding Mode and Structure-Activity Relationships of ITE as an Aryl Hydrocarbon Receptor (AhR) Agonist.

scientific article published on 20 December 2017

Enantioselective HPLC Analysis to Assist the Chemical Exploration of Chiral Imidazolines

scientific article published on 02 February 2020

Exploiting Chemical Toolboxes for the Expedited Generation of Tetracyclic Quinolines as a Novel Class of PXR Agonists

scientific article published on 27 December 2018

Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor

scientific article published on 20 March 2020

Identification and quantification of oxo-bile acids in human faeces with liquid chromatography-mass spectrometry: A potent tool for human gut acidic sterolbiome studies

scientific article published on 19 November 2018

Optimisation by Design of Experiment of Benzimidazol-2-One Synthesis under Flow Conditions

scientific article published on 03 July 2019

Selected cholesterol biosynthesis inhibitors produce accumulation of the intermediate FF-MAS that targets nucleus and activates LXRα in HepG2 cells.

scientific article published on 9 May 2017

Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms

scientific article published on 01 December 2018

Synthesis of atypical bile acids for use as investigative tools for the genetic defect of 3β-hydroxy-Δ(5)-C27-steroid oxidoreductase deficiency

scientific article published on 19 June 2014

Synthesis, physicochemical properties, and biological activity of bile acids 3-glucuronides: Novel insights into bile acid signalling and detoxification.

scientific article published on 11 December 2017

The Medicinal Chemistry in the Era of Machines and Automation: Recent Advances in Continuous Flow Technology

scientific article published on 21 February 2020