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List of works by Olaf Prante

(18)F- and (68)Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1.

scientific article published on 23 June 2016

(18)F-glyco-RGD peptides for PET imaging of integrin expression: efficient radiosynthesis by click chemistry and modulation of biodistribution by glycosylation

scientific article published on 16 December 2013

18F-Labeled FAUC 346 and BP 897 derivatives as subtype-selective potential PET radioligands for the dopamine D3 receptor.

scientific article

18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET imaging of mammary carcinoma

scientific article published on 10 September 2019

3,4,6-Tri-O-acetyl-2-deoxy-2-[18F]fluoroglucopyranosyl Phenylthiosulfonate: A Thiol-Reactive Agent for the Chemoselective18F-Glycosylation of Peptides

scientific article published on 01 January 2007

99mTc-MIP-1404 SPECT/CT for Assessment of Whole-Body Tumor Burden and Treatment Response in Patients With Biochemical Recurrence of Prostate Cancer

scientific article published on 17 June 2020

99mTc-MIP-1404 SPECT/CT for Patients With Metastatic Prostate Cancer: Interobserver and Intraobserver Variability in Treatment-Related Longitudinal Tracer Uptake Assessments of Prostate-Specific Membrane Antigen-Positive Lesions

scientific article published on 01 February 2020

A dopaminergic mechanism of antipsychotic drug efficacy, failure, and failure reversal: the role of the dopamine transporter

scientific article published on 23 July 2018

A series of 18F-labelled pyridinylphenyl amides as subtype-selective radioligands for the dopamine D3 receptor

scientific article

A series of 2-O-trifluoromethylsulfonyl-D-mannopyranosides as precursors for concomitant 18F-labeling and glycosylation by click chemistry

scientific article published on 8 February 2009

Assessment of Treatment Response by 99mTc-MIP-1404 SPECT/CT: A Pilot Study in Patients With Metastatic Prostate Cancer

scientific article published on 01 August 2018

Biodistribution studies of two 18F-labeled pyridinylphenyl amides as subtype selective radioligands for the dopamine D3 receptor

scientific article published on 26 December 2013

Characterization of 18F-FDG uptake in human endothelial cells in vitro

scientific article published on March 2004

Characterization of uptake of 3-[(131)I]iodo-alpha-methyl-L-tyrosine in human monocyte-macrophages

scientific article published on April 2004

Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers

scientific article

Detection of monoamine oxidase a in brain of living rats with [18F]fluoroethyl-harmol PET.

scientific article published on 24 September 2014

Development of 18F-Fluoroglycosylated PSMA-Ligands with Improved Renal Clearance Behavior

scientific article published on 17 February 2020

Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior

scientific article published on 29 April 2017

Discovery of a dopamine D4 selective PET ligand candidate taking advantage of a click chemistry based REM linker

scientific article

Disentangling inflammatory from fibrotic disease activity by fibroblast activation protein imaging

scientific article published on 21 July 2020

Effects of Recombinant Human Thyroid-Stimulating Hormone Superagonists on Thyroidal Uptake of18F-Fluorodeoxyglucose and Radioiodide ⬇️

scientific article (publication date: July 2011)

Estimation of [177Lu]PSMA-617 tumor uptake based on voxel-wise 3D Monte Carlo tumor dosimetry in patients with metastasized castration resistant prostate cancer

scientific article published on 14 July 2020

Evaluation of18F-Labeled Benzodioxine Piperazine-Based Dopamine D4Receptor Ligands: Lipophilicity as a Determinate of Nonspecific Binding

scientific article published on 23 November 2011

Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters

scientific article published on 11 December 2013

First Experience With SPECT/CT Using a 99mTc-Labeled Inhibitor for Prostate-Specific Membrane Antigen in Patients With Biochemical Recurrence of Prostate Cancer

scientific article published on 01 January 2017

H-CRRETAWAC-OH, a lead structure for the development of radiotracer targeting integrin α5β1?

scientific article

Identification of Boronic Acid Derivatives as an Active Form of N-Alkylaminoferrocene-Based Anticancer Prodrugs and Their Radiolabeling with 18F

scientific article published on 13 March 2019

Improved radiosynthesis and preliminary in vivo evaluation of a (18)F-labeled glycopeptide-peptoid hybrid for PET imaging of neurotensin receptor 2.

scientific article published on 7 February 2015

In Vitro and In Vivo Characterization of Selected Fluorine-18 Labeled Radioligands for PET Imaging of the Dopamine D3 Receptor.

scientific article published on 29 August 2016

In vitro and initial in vivo evaluation of (68)Ga-labeled transferrin receptor (TfR) binding peptides as potential carriers for enhanced drug transport into TfR expressing cells

scientific article

In vitro characterization of the thyroidal uptake of O-(2-[(18)F]fluoroethyl)-L-tyrosine

scientific article published on 22 February 2007

In vitro studies on the signal transduction of thyroidal uptake of 18F-FDG and 131I-Iodide.

scientific article published on August 2006

In vivo monitoring of the antiangiogenic effect of neurotensin receptor-mediated radiotherapy by small-animal positron emission tomography: a pilot study

scientific article

Induction and repair of DNA double-strand breaks in blood lymphocytes of patients undergoing 18F-FDG PET/CT examinations ⬇️

scientific article published on August 2, 2012

Labeling and glycosylation of peptides using click chemistry: a general approach to (18)F-glycopeptides as effective imaging probes for positron emission tomography

scientific article

Microwave-Assisted Rapid One-Pot Synthesis of Fused and Non-Fused Indoles and 5-[18 F]Fluoroindoles from Phenylazocarboxylates

scientific article

Multimerization of cRGD Peptides by Click Chemistry: Synthetic Strategies, Chemical Limitations, and Influence on Biological Properties ⬇️

scientific article published on October 18, 2010

Multimodal Bone Metastasis-associated Epidermal Growth Factor Receptor Imaging in an Orthotopic Rat Model

scientific article

Non-Invasive Characterization of Experimental Bone Metastasis in Obesity Using Multiparametric MRI and PET/CT

scientific article published on 18 May 2022

Optimization and synthesis of an18F-labeled dopamine D3receptor ligand using [18F]fluorophenylazocarboxylictert-butylester

scientific article published on 28 December 2015

PET radiopharmaceuticals for imaging integrin expression: tracers in clinical studies and recent developments.

scientific article published on 11 June 2014

Perturbed Development of Striatal Dopamine Transporters in Fatty Versus Lean Zucker Rats: a Follow-up Small Animal PET Study

scientific article published on 24 December 2014

Pharmacological characterization of low-to-moderate affinity opioid receptor agonists and brain imaging with 18F-labeled derivatives in rats

scientific article published on 31 July 2020

Prediction of early metastatic disease in experimental breast cancer bone metastasis by combining PET/CT and MRI parameters to a Model-Averaged Neural Network

scientific article published on 13 November 2018

Prototypic 18F-Labeled Argininamide-Type Neuropeptide Y Y1R Antagonists as Tracers for PET Imaging of Mammary Carcinoma.

scientific article published on 21 February 2017

Radioligands for the dopamine receptor subtypes

scientific article published on March 2013

Radiopharmaceuticals for imaging and endoradiotherapy of neurotensin receptor-positive tumors.

scientific article published on 7 November 2017

Radiosynthesis and Preclinical Evaluation of 18F-Fluoroglycosylated Octreotate for Somatostatin Receptor Imaging.

scientific article published on 07 October 2016

Radiosynthesis and evaluation of 18F-labeled dopamine D4-receptor ligands

scientific article published on 16 July 2020

Radiosynthesis and validation of ¹⁸F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain.

scientific article

Radiosynthesis of an F-fluoroglycosylated aminoferrocene for in-vivo imaging of reactive oxygen species activity by PET

article

Recent trends in pharmaceutical radiochemistry for molecular PET imaging

scientific article published on 24 July 2014

Regulation of uptake of 18F-FDG by a follicular human thyroid cancer cell line with mutation-activated K-ras

scientific article

Specific binding of [(18)F]fluoroethyl-harmol to monoamine oxidase A in rat brain cryostat sections, and compartmental analysis of binding in living brain

scientific article published on 19 September 2015

Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands

scientific article

Sweetening pharmaceutical radiochemistry by (18)f-fluoroglycosylation: a short review.

scientific article published on June 2014

Syntheses and radiofluorination of two derivatives of 5-cyano-indole as selective ligands for the dopamine subtype-4 receptor

Syntheses, receptor bindings, in vitro and in vivo stabilities and biodistributions of DOTA-neurotensin(8-13) derivatives containing β-amino acid residues - a lesson about the importance of animal experiments

scientific article published in December 2013

Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents

scientific article

Synthesis and evaluation of a (18)F-labeled diarylpyrazole glycoconjugate for the imaging of NTS1-positive tumors

scientific article published on 6 November 2013

Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging.

scientific article published in December 2014

Synthesis and in vitro and in vivo evaluation of an (18)F-labeled neuropeptide Y analogue for imaging of breast cancer by PET.

scientific article published on 13 March 2015

Synthesis and in vivo evaluation of an (18)F-labeled glycoconjugate of PD156707 for imaging ETA receptor expression in thyroid carcinoma by positron emission tomography

scientific article published on 19 September 2013

Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype

scientific article

Synthesis of a (68)ga-labeled peptoid-Peptide hybrid for imaging of neurotensin receptor expression in vivo

scientific article published on 21 May 2010

Synthesis, biological evaluation and radiosynthesis of buprenorphine-derived phenylazocarboxamides as novel μ-opioid receptor ligands

scientific article published on 06 May 2020

Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET.

scientific article

Targeting Fibroblast Activation Protein: Radiosynthesis and Preclinical Evaluation of an 18F-labeled FAP Inhibitor

scientific article published on 24 April 2020

Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors

scientific article published on 10 March 2017

[(68)Ga]Ga-DO(2)A-(OBu-l-tyr)(2): synthesis, (68)Ga-radiolabeling and in vitro studies of a novel (68)Ga-DO(2)A-tyrosine conjugate as potential tumor tracer for PET.

scientific article

[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor

scientific article published on 6 December 2017

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