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List of works by Marcin Drąg

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Emerging principles in protease-based drug discovery

scientific article published on September 1, 2010
FLIP(L) induces caspase 8 activity in the absence of interdomain caspase 8 cleavage and alters substrate specificity

scientific article published on February 2011
Small ubiquitin-related modifier (SUMO)-specific proteases: profiling the specificities and activities of human SENPs

scientific article
DeSUMOylating enzymes--SENPs

scientific article
A constitutively active and uninhibitable caspase-3 zymogen efficiently induces apoptosis

scientific article
Caspase Substrates and Inhibitors

scientific article published on August 1, 2013
Distribution and paralogue specificity of mammalian deSUMOylating enzymes

scientific article published on September 2010
Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials

scientific article published on 30 September 2009
Aminopeptidase fingerprints, an integrated approach for identification of good substrates and optimal inhibitors

scientific article
Design of ultrasensitive probes for human neutrophil elastase through hybrid combinatorial substrate library profiling

scientific article published on February 3, 2014
Mechanism and specificity of the human paracaspase MALT1.

scientific article
Activation and specificity of human caspase-10.

scientific article published on September 2010
Activity profiling of human deSUMOylating enzymes (SENPs) with synthetic substrates suggests an unexpected specificity of two newly characterized members of the family

scientific article
Metallo-aminopeptidase inhibitors

scientific article published on 10 May 2010
Functional characterization of a SUMO deconjugating protease of Plasmodium falciparum using newly identified small molecule inhibitors

scientific article (publication date: 24 June 2011)
Probing the S1 specificity pocket of the aminopeptidases that generate antigenic peptides.

scientific article published on April 2011
Positional-scanning fluorigenic substrate libraries reveal unexpected specificity determinants of DUBs (deubiquitinating enzymes).

scientific article
SARS hCoV papain-like protease is a unique Lys48 linkage-specific di-distributive deubiquitinating enzyme

scientific article published on June 2015
Synthetic substrates for measuring activity of autophagy proteases-autophagins (Atg4)

scientific article published on October 19, 2010
Comparision of the cytotoxic effects of birch bark extract, betulin and betulinic acid towards human gastric carcinoma and pancreatic carcinoma drug-sensitive and drug-resistant cell lines.

scientific article published on 24 April 2009
Synthesis and structure-activity relationships of phosphonic arginine mimetics as inhibitors of the M1 and M17 aminopeptidases from Plasmodium falciparum

scientific article
Fingerprinting the substrate specificity of M1 and M17 aminopeptidases of human malaria, Plasmodium falciparum

scientific article
Extended substrate specificity and first potent irreversible inhibitor/activity-based probe design for Zika virus NS2B-NS3 protease

scientific article (publication date: December 2016)
Toolbox of Fluorescent Probes for Parallel Imaging Reveals Uneven Location of Serine Proteases in Neutrophils.

scientific article published on 3 July 2017
Structural and functional insights into caseinolytic proteases reveal an unprecedented regulation principle of their catalytic triad

scientific article published on June 24, 2013
Small Molecule Active Site Directed Tools for Studying Human Caspases

scientific article published on 9 November 2015
Expression of aminopeptidase N/CD13 in human ovarian cancers

scientific article published on 01 September 2006
Design of a Selective Substrate and Activity Based Probe for Human Neutrophil Serine Protease 4

scientific article published on July 14, 2015
Small molecules not direct activators of caspases

scientific article published on 01 September 2007
Esters of betulin and betulinic acid with amino acids have improved water solubility and are selectively cytotoxic toward cancer cells.

scientific article published on 14 June 2009
Emerging challenges in the design of selective substrates, inhibitors and activity-based probes for indistinguishable proteases

scientific article published on 4 January 2017
SUMO-mediated regulation of NLRP3 modulates inflammasome activity

scientific article published in Nature Communications
Counter Selection Substrate Library Strategy for Developing Specific Protease Substrates and Probes

scientific article
Two-pronged attack: dual inhibition of Plasmodium falciparum M1 and M17 metalloaminopeptidases by a novel series of hydroxamic acid-based inhibitors

scientific article
The new esters derivatives of betulin and betulinic acid in epidermoid squamous carcinoma treatment - In vitro studies.

scientific article published on 13 April 2015
X-ray crystal structure and specificity of the Plasmodium falciparum malaria aminopeptidase PfM18AAP

scientific article
Synthesis of a HyCoSuL peptide substrate library to dissect protease substrate specificity

scientific article published on 21 September 2017
Activity profiling and structures of inhibitor-bound SARS-CoV-2-PLpro protease provides a framework for anti-COVID-19 drug design

scientific article published on 30 April 2020
Design of Selective Substrates and Activity-Based Probes for Hydrolase Important for Pathogenesis 1 (HIP1) from Mycobacterium tuberculosis.

scientific article published on 15 July 2016
Positional Scanning Substrate Combinatorial Library (PS-SCL) Approach to Define Caspase Substrate Specificity

scientific article published on January 1, 2014
Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors

scientific article published on 5 May 2008
Trojan Horse Strategies Used by Pathogens to Influence the Small Ubiquitin-Like Modifier (SUMO) System of Host Eukaryotic Cells

scientific article published on 03 January 2012
Unnatural amino acids increase activity and specificity of synthetic substrates for human and malarial cathepsin C.

scientific article
Selective imaging of cathepsin L in breast cancer by fluorescent activity-based probes.

scientific article
Barrel-shaped ClpP Proteases Display Attenuated Cleavage Specificities

scientific article published on 25 November 2015
alpha-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases

scientific article published on 20 April 2005
Gingipain aminopeptidase activities in Porphyromonas gingivalis

scientific article published on December 1, 2012
Substrate Specificity and Possible Heterologous Targets of Phytaspase, a Plant Cell Death Protease

scientific article published on 17 August 2015
The elastase-PK101 structure: mechanism of an ultrasensitive activity-based probe revealed

scientific article
Extensive peptide and natural protein substrate screens reveal that mouse caspase-11 has much narrower substrate specificity than caspase-1.

scientific article published on 6 February 2018

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