Search filters

List of works by Andrew M Beekman

A small molecule drug conjugate (SMDC) of DUPA and a duocarmycin built on the solid phase

scientific article published on 27 November 2019

Discovery and Synthesis of Boletopsins 13 and 14, Brominated Fungal Metabolites of Terrestrial Origin.

scientific article published on 24 July 2015

First syntheses of the biologically active fungal metabolites pestalotiopsones A, B, C and F.

scientific article published in February 2013

Identification of Small-Molecule Inhibitors of the Antiapoptotic Protein Myeloid Cell Leukaemia-1 (Mcl-1).

scientific article published on 30 November 2015

Identification of selective protein-protein interaction inhibitors using efficient peptide-directed ligand design

scientific article published on 22 March 2019

Peptide-Directed Binding for the Discovery of Modulators of α-Helix-Mediated Protein-Protein Interactions: Proof-of-Concept Studies with the Apoptosis Regulator Mcl-1.

scientific article published on 2 July 2017

Rac1 plays a role in CXCL12 but not CCL3-induced chemotaxis and Rac1 GEF inhibitor NSC23766 has off target effects on CXCR4.

scientific article

Ravynic acid, an antibiotic polyeneyne tetramic acid from Penicillium sp. elucidated through synthesis

scientific article published on 21 July 2016

Small-Molecule and Peptide Inhibitors of the Pro-Survival Protein Mcl-1

scientific article published on 23 December 2015

Stereochemical assignment of the fungal metabolites pestalotiopsones D and E through enantiopure synthesis.

scientific article published on 29 October 2013

Syntheses of the fungal metabolites boletopsins 7, 11, and 12 from the Papua New Guinea medicinal mushroom Boletopsis sp.

scientific article