List of works - Michel Baltas

Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a biomimetic approach

scientific article

Design, synthesis and biological evaluation of novel hydroxamic acids bearing artemisinin skeleton.

scientific article published on 17 March 2016

Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth.

scientific article published on 20 June 2015

Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A.

scientific article published on 15 March 2016

In Silico Repositioning of Cannabigerol as a Novel Inhibitor of the Enoyl Acyl Carrier Protein (ACP) Reductase (InhA)

scientific article published on 15 July 2019

Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis

scientific article published on 16 July 2016

Small molecules inhibitors of plasminogen activator inhibitor-1 - an overview

scientific article published on 8 January 2015

Structure-Based Virtual Ligand Screening on the XRCC4/DNA Ligase IV Interface.

scientific article published on 11 March 2016

Synthesis and biological evaluation against Leishmania donovani of novel hybrid molecules containing indazole-based 2-pyrone scaffolds

scientific article published on 19 November 2018

Synthesis and biological evaluation of diarylheptanoids as potential antioxidant and anti-inflammatory agents.

scientific article

Synthesis and evaluation of antioxidant phenolic diaryl hydrazones as potent antiangiogenic agents in atherosclerosis.

scientific article published on 30 May 2016

Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis

scientific article published on 04 November 2013

Synthesis, In Silico, and In Vitro Evaluation of Anti-Leishmanial Activity of Oxadiazoles and Indolizine Containing Compounds Flagged against Anti-Targets

scientific article published on 02 April 2019

Synthesis, antioxidant and cytoprotective evaluation of potential antiatherogenic phenolic hydrazones. A structure-activity relationship insight

scientific article published on 23 May 2014

Total Synthesis of Tedarene A.

scientific article

Triazolophthalazines: Easily Accessible Compounds with Potent Antitubercular Activity.

scientific article

List of works by Michel Baltas

Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a biomimetic approach

Design, synthesis and biological evaluation of novel hydroxamic acids bearing artemisinin skeleton.

Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growth.

Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A.

In Silico Repositioning of Cannabigerol as a Novel Inhibitor of the Enoyl Acyl Carrier Protein (ACP) Reductase (InhA)

Pyrrolidinone and pyrrolidine derivatives: Evaluation as inhibitors of InhA and Mycobacterium tuberculosis

Small molecules inhibitors of plasminogen activator inhibitor-1 - an overview

Structure-Based Virtual Ligand Screening on the XRCC4/DNA Ligase IV Interface.

Synthesis and biological evaluation against Leishmania donovani of novel hybrid molecules containing indazole-based 2-pyrone scaffolds

Synthesis and biological evaluation of diarylheptanoids as potential antioxidant and anti-inflammatory agents.

Synthesis and evaluation of antioxidant phenolic diaryl hydrazones as potent antiangiogenic agents in atherosclerosis.

Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis

Synthesis, In Silico, and In Vitro Evaluation of Anti-Leishmanial Activity of Oxadiazoles and Indolizine Containing Compounds Flagged against Anti-Targets

Synthesis, antioxidant and cytoprotective evaluation of potential antiatherogenic phenolic hydrazones. A structure-activity relationship insight

Total Synthesis of Tedarene A.

Triazolophthalazines: Easily Accessible Compounds with Potent Antitubercular Activity.