List of works by Philippe Grellier

A Photoalkylative Fluorogenic Probe of Guttiferone A for Live Cell Imaging and Proteome Labeling in Plasmodium falciparum

scientific article published on 04 November 2020

A Plasmodium falciparum FcB1-schizont-EST collection providing clues to schizont specific gene structure and polymorphism

scientific article

A Protein Phosphatase 1 involved in correct nucleus positioning in trypanosomes

scientific article

A new xanthone from the bark extract of Rheedia acuminata and antiplasmodial activity of its major compounds. ⬇️

scientific article published on 14 October 2010

Activity of Ocimum basilicum, Ocimum canum, and Cymbopogon citratus essential oils against Plasmodium falciparum and mature-stage larvae of Anopheles funestus s.s.

scientific article

Aminocyclopropanes as precursors of endoperoxides with antimalarial activity ⬇️

scientific article published on October 11, 2010

Anti-Plasmodium activity of ceramide analogs

scientific article

Antileishmanial and trypanocidal activity of Brazilian Cerrado plants

article

Antimalarial activity of axidjiferosides, new β-galactosylceramides from the African sponge Axinyssa djiferi

scientific article published on 17 April 2013

Antimalarial and cytotoxic activities of ethnopharmacologically selected medicinal plants from South Vietnam

scientific article

Antimalarial xanthones from Calophyllum caledonicum and Garcinia vieillardii

scientific article published in November 2004

Antiplasmodial Activity of Nitroaromatic Compounds: Correlation with Their Reduction Potential and Inhibitory Action on Plasmodium falciparum Glutathione Reductase

scientific article published on 10 December 2019

Antiplasmodial Biodereplication Based on Highly Efficient Methods

Antiplasmodial alkaloids from Desmos rostrata

scientific article published on 01 December 2008

Antiplasmodial benzophenone derivatives from the root barks of Symphonia globulifera (Clusiaceae).

scientific article published on 29 March 2010

Antiplasmodial benzophenones from the trunk latex of Moronobea coccinea (Clusiaceae). ⬇️

scientific article published on 4 December 2008

Antiplasmodial phenolic compounds from Piptadenia pervillei

scientific article

Antiplasmodial, antitrypanosomal, and cytotoxic activities of prenylated flavonoids isolated from the stem bark of Artocarpus styracifolius

scientific article published on 8 April 2010

Antivascular and anti-parasite activities of natural and hemisynthetic flavonoids from New Caledonian Gardenia species (Rubiaceae).

scientific article published on 8 January 2015

Bile Salt Hydrolase Activities: A Novel Target to Screen Anti-Giardia Lactobacilli?

scientific article published on 8 February 2018

Bile-Salt-Hydrolases from the Probiotic Strain Lactobacillus johnsonii La1 Mediate Anti-giardial Activity in Vitro and in Vivo.

scientific article published in January 2017

Bioactive properties of plant species ingested by chimpanzees (Pan troglodytes schweinfurthii) in the Kibale National Park, Uganda

scientific article published on January 2006

Biochemical properties and cellular localization of Plasmodium falciparum protein disulfide isomerase

scientific article (publication date: March 2007)

Brazilian Cerrado Qualea grandiflora Mart. Leaves Exhibit Antiplasmodial and Trypanocidal Activities In vitro

scientific article

Characterization of PfDYN2, a dynamin-like protein of Plasmodium falciparum expressed in schizonts

scientific article (publication date: June 2007)

Clerodane and labdane diterpenoids from Nuxia sphaerocephala

scientific article

Constituents of Burasaïa madagascarensis: a new clerodane-type diterpene

scientific article published in April 2002

Corynanthean-Epicatechin Flavoalkaloids from Corynanthe pachyceras ⬇️

scientific article published on 07 June 2020

Deconjugated Bile Salts Produced by Extracellular Bile-Salt Hydrolase-Like Activities from the Probiotic Lactobacillus johnsonii La1 Inhibit Giardia duodenalis In vitro Growth

scientific article

Dendropsophin 1, a novel antimicrobial peptide from the skin secretion of the endemic Colombian frog Dendropsophus columbianus

scientific article

Design, synthesis and antimalarial activity of novel, quinoline-based, zinc metallo-aminopeptidase inhibitors.

scientific article

Design, synthesis and antimalarial activity of trifluoromethylartemisinin-mefloquine dual molecules

scientific article

Design, synthesis and in vitro antimalarial activity of an acylhydrazone library

scientific article

Detection, characterization, and screening of heme-binding molecules by mass spectrometry for malaria drug discovery

scientific article

Diarylheptanoid Glucosides from Pyrostria major and Their Antiprotozoal Activities

Diversity of apostome ciliates, Chromidina spp. (Oligohymenophorea, Opalinopsidae), parasites of cephalopods of the Mediterranean Sea

scientific article

Dynamic molecular events associated to Plasmodium berghei gametogenesis through proteomic approach

scientific article published on 15 November 2017

Eumitrins C-E: Structurally diverse xanthone dimers from the vietnamese lichen Usnea baileyi

scientific article published on 06 December 2019

Evaluation of nucleoside hydrolase inhibitors for treatment of African trypanosomiasis

scientific article

Flavonoids from Dalbergia louvelii and their antiplasmodial activity.

scientific article published on 30 October 2003

Fluoroartemisinin: trifluoromethyl analogues of artemether and artesunate.

scientific article published in May 2004

Goniomedines A and B: unprecedented bisindole alkaloids formed through fusion of two indole moieties via a dihydropyran unit

scientific article published on 06 August 2012

Heme-binding activity of methoxyflavones from Pentzia monodiana Maire (Asteraceae).

scientific article

Identification of novel Trypanosoma cruzi prolyl oligopeptidase inhibitors by structure-based virtual screening.

scientific article

In vitro antiplasmodial activity and cytotoxicity of 33 West African plants used for treatment of malaria.

scientific article published on April 2005

In vitro investigation of Brazilian Cerrado plant extract activity against Plasmodium falciparum, Trypanosoma cruzi and T. brucei gambiense.

scientific article published on 29 July 2015

Inactivation of Plasmodium falciparum in whole blood using the amustaline and glutathione pathogen reduction technology

scientific article published on 04 March 2020

Isolation, characterization and antiplasmodial activity of steroidal alkaloids from Funtumia elastica (Preuss) Stapf

scientific article

Malaria and obesity: obese mice are resistant to cerebral malaria

scientific article published on 19 May 2008

Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation, and Preliminary SAR Studies.

scientific article published in February 2016

Molecular Networking Reveals Serpentinine-Related Bisindole Alkaloids from Picralima nitida, a Previously Well-Investigated Species

scientific article published on 24 February 2020

Molecular, functional and structural properties of the prolyl oligopeptidase of Trypanosoma cruzi (POP Tc80), which is required for parasite entry into mammalian cells

scientific article

New ether diglycosides from Matayba guianensis with antiplasmodial activity

scientific article published on 01 July 2005

New ferrocenic pyrrolo[1,2-a]quinoxaline derivatives: synthesis, and in vitro antimalarial activity

scientific article published on 17 September 2008

Novel N-(4-Piperidinyl)benzamide antimalarials with mammalian protein farnesyltransferase inhibitory activity

scientific article published on October 2005

Novel antimalarial compounds isolated in a survey of self-medicative behavior of wild chimpanzees in Uganda

scientific article published on August 2004

Oligopeptidase B, a missing enzyme in mammals and a potential drug target for trypanosomatid diseases.

scientific article published on 16 October 2019

Orally active antimalarials: hydrolytically stable derivatives of 10-trifluoromethyl anhydrodihydroartemisinin

scientific article published in March 2004

Photochemical inactivation with amotosalen and long-wavelength ultraviolet light of Plasmodium and Babesia in platelet and plasma components.

scientific article

Plasmodium falciparum genes differentially expressed during merozoite morphogenesis.

scientific article

PlasmodiumTelomeric Sequences: Structure, Stability and Quadruplex Targeting by Small Compounds

scholarly article by Anne De Cian published in November 2008

Pleiokomenines A and B: Dimeric Aspidofractinine Alkaloids Tethered with a Methylene Group.

scientific article published on 7 November 2017

Preparative isolation, fast centrifugal partition chromatography purification and biological activity of cajaflavanone from Derris ferruginea stems

scientific article

Probiotics for the control of parasites: an overview.

scientific article

Prolyl Oligopeptidase From Leishmania infantum: Biochemical Characterization and Involvement in Macrophage Infection

scientific article published on 28 May 2020

Prolyl oligopeptidase of Trypanosoma brucei hydrolyzes native collagen, peptide hormones and is active in the plasma of infected mice.

scientific article published on 24 February 2010

Prolylisoxazoles: potent inhibitors of prolyloligopeptidase with antitrypanosomal activity

scientific article published in September 2003

Pseudoguanolide sesquiterpene lactones from Vernoniopsis caudata and their in vitro antiplasmodial activities.

scientific article published on May 2005

Redescription of Dicyemennea eledones (Wagener, 1857) (Phylum Dicyemida) from Eledone cirrhosa (Lamarck, 1798) (Mollusca: Cephalopoda: Octopoda).

scientific article

Revealing a Novel Otubain-Like Enzyme from Leishmania infantum with Deubiquitinating Activity toward K48-Linked Substrate

scientific article

Revisiting Previously Investigated Plants: A Molecular Networking-Based Study of Geissospermum laeve.

scientific article

Screening extracts of Madagascan plants in search of antiplasmodial compounds

scientific article published on September 2004

Sesquiterpenoids from Teucrium ramosissimum

scientific article published in July 2009

Specific human antibodies do not inhibit Trypanosoma cruzi oligopeptidase B and cathepsin B, and immunoglobulin G enhances the activity of trypomastigote-secreted oligopeptidase B.

scientific article published on 16 February 2005

Spiranthenones A and B, tetraprenylated phloroglucinol derivatives from the leaves of Spiranthera odoratissima.

scientific article

Streamlined targeting of Amaryllidaceae alkaloids from the bulbs of Crinum scillifolium using spectrometric and taxonomically-informed scoring metabolite annotations

scientific article published on 26 August 2020

Structure and total synthesis of (-)-myrionidine and (-)-schoberine, antimalarial alkaloids from Myrioneuron nutans

scientific article

Synthesis and Antiplasmodial Activity of Novel Fosmidomycin Derivatives and Conjugates with Artemisinin and Aminochloroquinoline

scientific article published on 21 October 2020

Synthesis and antimalarial activity of some new 1,2-dioxolane derivatives

scientific article published in December 2002

Synthesis and antimalarial evaluation of a series of piperazinyl flavones

scientific article published on 18 November 2006

Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives.

scientific article

Synthesis and antimalarial evaluation of new N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives.

scientific article

Synthesis and in vitro and in vivo antimalarial activity of N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives.

scientific article published on February 2003

Synthesis and in vitro antiplasmodial activity of ferrocenyl aminoquinoline derivatives

scientific article published on 3 December 2014

Synthesis of novel guttiferone A derivatives: in-vitro evaluation toward Plasmodium falciparum, Trypanosoma brucei and Leishmania donovani

scientific article published on 10 May 2013

Synthesis, antimalarial activity, and molecular modeling of new pyrrolo[1,2-a]quinoxalines, bispyrrolo[1,2-a]quinoxalines, bispyrido[3,2-e]pyrrolo[1,2-a]pyrazines, and bispyrrolo[1,2-a]thieno[3,2-e]pyrazines

scientific article published on April 2004

The antiplasmodium effects of a traditional South American remedy: Zanthoxylum chiloperone var. angustifolium against chloroquine resistant and chloroquine sensitive strains of Plasmodium falciparum

The traditional medicine Spilanthes acmella, and the alkylamides spilanthol and undeca-2E-ene-8,10-diynoic acid isobutylamide, demonstrate in vitro and in vivo antimalarial activity ⬇️

scientific article

Theionbrunonines A and B: Dimeric Vobasine Alkaloids Tethered by a Thioether Bridge from Mostuea brunonis

scientific article published on 10 October 2018

Towards the synthesis of bisubstrate inhibitors of protein farnesyltransferase: Synthesis and biological evaluation of new farnesylpyrophosphate analogues

scientific article

Triterpenes from the exudate of Gardenia urvillei

scientific article published on 19 November 2015

Vital role for Plasmodium berghei Kinesin8B in axoneme assembly during male gamete formation and mosquito transmission.

scientific article published in March 2020

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