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List of works by Alireza Foroumadi

2,3-Diaminopyridinium 6-carboxypyridine-2-carboxylate ⬇️

scientific article published on November 16, 2011

2-Amino-3-cyano-4-(5-arylisoxazol-3-yl)-4H-chromenes: synthesis and in vitro cytotoxic activity.

scientific article published on 20 January 2012

2-Amino-4-(nitroalkyl)-4H-chromene-3-carbonitriles as New Cytotoxic Agents

scientific article published on January 2013

3-Aryl Coumarin Derivatives Bearing Aminoalkoxy Moiety as Multi-Target-Directed Ligands against Alzheimer's Disease

scientific article published on 08 April 2019

4-Aryl-4H-naphthopyrans derivatives: one-pot synthesis, evaluation of Src kinase inhibitory and anti-proliferative activities ⬇️

scientific article published on December 26, 2012

5,6-Dimethoxybenzofuran-3-one derivatives: a novel series of dual Acetylcholinesterase/Butyrylcholinesterase inhibitors bearing benzyl pyridinium moiety

scientific article

6-Cinnamoyl-4-arylaminothienopyrimidines as highly potent cytotoxic agents: Design, synthesis and structure-activity relationship studies

scientific article published on 18 October 2019

9H-Carbazole Derivatives Containing the N-Benzyl-1,2,3-triazole Moiety as New Acetylcholinesterase Inhibitors.

scientific article

A Convenient Method for the Synthesis of Chromeno[4,3-b]pyridines Via Three-component Reaction

scientific article published on 01 January 2018

A review on flavonoid-based scaffolds as multi-target-directed ligands (MTDLs) for Alzheimer's disease

scientific article published on 07 May 2018

Anti-Helicobacter pylori activity and Structure-Activity Relationship study of 2-Alkylthio-5-(nitroaryl)-1,3,4-thiadiazole Derivatives

scientific article published on January 2013

Anti-Helicobacter pylori activity of the methanolic extract of Geum iranicum and its main compounds

scientific article

Anti-proliferative and apoptotic effects of the derivatives from 4-aryl-4H-chromene family on human leukemia K562 cells

scientific article

Anticancer effects of synthetic hexahydrobenzo [g]chromen-4-one derivatives on human breast cancer cell lines.

scientific article published on June 2016

Antinociceptive properties of new coumarin derivatives bearing substituted 3,4-dihydro-2H-benzothiazines.

scientific article

Antiproliferative activity of flavonoids: influence of the sequential methoxylation state of the flavonoid structure

scientific article

Antituberculosis agents. V. Synthesis, evaluation of in vitro antituberculosis activity and cytotoxicity of some 2-(5-nitro-2-furyl)-1,3,4-thiadiazole derivatives

scientific article published on September 2002

Benzofuran-derived benzylpyridinium bromides as potent acetylcholinesterase inhibitors.

scientific article

Caspase-dependent apoptosis induced by two synthetic halogenated flavanones, 3',7-dichloroflavanone and 3',6-dichloroflavanone, on human breast and prostate cancer cells

scientific article published on 20 December 2017

Combined isocyanide-based multi-component Ullmann-type reaction: an efficient access to novel nitrogen-containing pentacyclic compounds

scientific article published on 01 August 2015

Concomitant activation of caspase-9 and down-regulation of IAP proteins as a mechanism of apoptotic death in HepG2, T47D and HCT-116 cells upon exposure to a derivative from 4-aryl-4H-chromenes family

scientific article

Conformationally constrained analogs of N-substituted piperazinylquinolones: synthesis and antibacterial activity of N-(2,3-dihydro-4-hydroxyimino-4H-1-benzopyran-3-yl)-piperazinylquinolones

scientific article published on July 2009

Coumarin derivatives bearing benzoheterocycle moiety: synthesis, cholinesterase inhibitory, and docking simulation study.

scientific article published on June 2017

Coumarin-based bioactive compounds: facile synthesis and biological evaluation of coumarin-fused 1,4-thiazepines.

scientific article published on 29 August 2011

Curcumin-loaded guanidine functionalized PEGylated I3ad mesoporous silica nanoparticles KIT-6: practical strategy for the breast cancer therapy.

scientific article published on 28 June 2014

Cytotoxic Activity and DNA Binding Property of New Aminopyrimidine Derivatives

scholarly article

Cytotoxic activity evaluation and QSAR study of chromene-based chalcones.

scientific article

Cytotoxicity and Apoptosis Inducing Activities of 2-Amino-4H-chromene-3-carbonitrile Derivatives Loaded on Gold Nanoparticles Against Human Breast Cancer Cell Line T47D.

scientific article published on 31 January 2014

Design and synthesis of benzodiazepine-1,2,3-triazole hybrid derivatives as selective butyrylcholinesterase inhibitors

scientific article published on 17 December 2019

Design and synthesis of novel anti-Alzheimer's agents: Acridine-chromenone and quinoline-chromenone hybrids.

scientific article

Design, Synthesis, Biological Evaluation, and Docking Study of Acetylcholinesterase Inhibitors: New Acridone-1,2,4-oxadiazole-1,2,3-triazole Hybrids.

scientific article

Design, synthesis and anticholinesterase activity of novel benzylidenechroman-4-ones bearing cyclic amine side chain

scientific article published on 29 April 2015

Design, synthesis and biological evaluation of novel anti-cytokine 1,2,4-triazine derivatives.

scientific article published on 13 August 2013

Design, synthesis and evaluation of novel multi-target-directed ligands for treatment of Alzheimer's disease based on coumarin and lipoic acid scaffolds

scientific article published on 02 May 2018

Design, synthesis, biological evaluation, and molecular dynamics of novel cholinesterase inhibitors as anti-Alzheimer's agents

scientific article published on 28 May 2019

Design, synthesis, cytotoxicity evaluation and docking studies of 1,2,4-triazine derivatives bearing different arylidene-hydrazinyl moieties as potential mTOR inhibitors.

scientific article published in February 2018

Design, synthesis, docking study and cytotoxic activity evaluation of some novel letrozole analogs

scientific article

Design, synthesis, in vitro cytotoxic activity evaluation, and apoptosis-induction study of new 9(10H)-acridinone-1,2,3-triazoles.

scientific article published on 14 July 2015

Design, synthesis, molecular docking study, and antibacterial evaluation of some new fluoroquinolone analogues bearing a quinazolinone moiety

scientific article published on 08 October 2020

Design, synthesis, molecular modeling and anticholinesterase activity of benzylidene-benzofuran-3-ones containing cyclic amine side chain.

scientific article published on 09 May 2017

Design, synthesis, pharmacological evaluation, and docking study of new acridone-based 1,2,4-oxadiazoles as potential anticonvulsant agents.

scientific article published in February 2016

Determination of the role of calcium on instability of neurotoxic metabolite of ecstasy by HPTLC-mass

scientific article published on 17 January 2013

Discovery of novel 1,2,4-triazolo-1,2,4-triazines with thiomethylpyridine hinge binders as potent c-Met kinase inhibitors

scientific article published on 01 May 2019

Discovery of novel dual inhibitors against Mdm2 and Mdmx proteins by in silico approaches and binding assay.

scientific article published on 30 December 2015

Effects of silica nanoparticle supported ionic liquid as additive on thermal reversibility of human carbonic anhydrase II ⬇️

scientific article published on July 22, 2012

Facile synthesis and antiproliferative activity of 7H-benzo[7,8]chromeno[2,3-d]pyrimidin-8-amines.

scientific article published on 21 December 2016

Folic acid decorated magnetic nanosponge: An efficient nanosystem for targeted curcumin delivery and magnetic resonance imaging

scientific article published on 13 August 2019

Formulation and evaluation of targeted nanoparticles for breast cancer theranostic system.

scientific article

Functionalized N(2-oxyiminoethyl) piperazinyl quinolones as new cytotoxic agents

scientific article published on January 2007

Glutathione Conjugated Polyethylenimine on the Surface of Fe3O4 Magnetic Nanoparticles as a Theranostic Agent for Targeted and Controlled Curcumin Delivery.

scientific article published on 11 January 2018

Imidazo[2,1-b]thiazole derivatives as new inhibitors of 15-lipoxygenase.

scientific article

Imidazolylchromanones containing alkyl side chain as lanosterol 14α-demethylase inhibitors: synthesis, antifungal activity and docking study.

scientific article published on 14 March 2013

In Silico Screening of IL-1β Production Inhibitors Using Chemometric Tools

scientific article published on January 2017

In Vitro Antiplasmodial Activity and Cytotoxic Effect of (Z)-2-Benzylidene-4, 6-Dimethoxybenzofuran-3(2H)-One Derivatives

scientific article published on July 2016

In Vitro Interaction of Geldanamycin with Triazoles and Echinocandins Against Common and Emerging Candida Species

scientific article published on 10 August 2019

In vitro antitumor evaluation of 4H-chromene-3-carbonitrile derivatives as a new series of apoptotic inducers

scientific article published on 19 March 2014

In vitro cytotoxicity and phototoxicity of N-piperazinyl quinolone derivatives with a 2-thienyl group.

scientific article published on 3 April 2007

In vitro immunobiological studies of novel 5-(5-nitrofuran-2-yl)-1, 3, 4-thiadiazoles with piperazinyl-linked benzamidine substituents against Leishmania major

scientific article published on 28 August 2013

Indolinone-based acetylcholinesterase inhibitors: synthesis, biological activity and molecular modeling.

scientific article

Induction of apoptosis through tubulin inhibition in human cancer cells by new chromene-based chalcones

scientific article

Isochaihulactone analogues: synthesis and anti-proliferative activity of novel dibenzylbutyrolactones.

scientific article published on 7 October 2010

Mannich bases of 7-piperazinylquinolones and kojic acid derivatives: synthesis, in vitro antibacterial activity and in silico study.

scientific article published on 11 August 2013

Medicinal plants in the treatment of Helicobacter pylori infections.

scientific article

Molecular identification and antifungal susceptibility profile of Candida species isolated from patients with vulvovaginitis in Tehran, Iran.

scientific article published on 26 December 2017

Monoterpenes as nitrofurantoin resistance modulating agents: minimal structural requirements, molecular dynamics simulations, and the effect of piperitone on the emergence of nitrofurantoin resistance in Enterobacteriaceae

scientific article published on 15 July 2015

N-(2-(Piperazin-1-yl)phenyl)arylamide Derivatives as β-Secretase (BACE1) Inhibitors: Simple Synthesis by Ugi Four-Component Reaction and Biological Evaluation

scientific article published on 19 March 2015

N-Phenyl-2-p-tolylthiazole-4-carboxamide derivatives: Synthesis and cytotoxicity evaluation as anticancer agents

scientific article

N-Substituted piperazinyl quinolones as potential cytotoxic agents: structure-activity relationships study

scientific article

N-substituted indole carbohydrazide derivatives: synthesis and evaluation of their antiplatelet aggregation activity.

scientific article

N-substituted piperazinyl sarafloxacin derivatives: synthesis and in vitro antibacterial evaluation

scientific article published on 03 November 2018

N1,N1-Dimethylpropane-1,2-diaminium bis(6-carboxypyridine-2-carboxylate) monohydrate ⬇️

scientific article published on March 19, 2011

New 7-piperazinylquinolones containing (benzo[d]imidazol-2-yl)methyl moiety as potent antibacterial agents

scientific article published on 07 June 2018

New classes of carbazoles as potential multi-functional anti-Alzheimer's agents

scientific article published on 29 July 2019

New racemic annulated pyrazolo[1,2-b]phthalazines as tacrine-like AChE inhibitors with potential use in Alzheimer's disease

scientific article

New tacrine-derived AChE/BuChE inhibitors: Synthesis and biological evaluation of 5-amino-2-phenyl-4H-pyrano[2,3-b]quinoline-3-carboxylates.

scientific article

New tetracyclic tacrine analogs containing pyrano[2,3-c]pyrazole: efficient synthesis, biological assessment and docking simulation study

scientific article published on 18 October 2014

Novel 3-phenylcoumarin-lipoic acid conjugates as multi-functional agents for potential treatment of Alzheimer's disease

scientific article published on 02 May 2018

Novel N-2-(Furyl)-2-(chlorobenzyloxyimino) Ethyl Piperazinyl Quinolones: Synthesis, Cytotoxic Evaluation and Structure-Activity Relationship

scientific article

One-pot, four-component synthesis of novel cytotoxic agents 1-(5-aryl-1,3,4-oxadiazol-2-yl)-1-(1H-pyrrol-2-yl)methanamines

scientific article published on 16 March 2014

PEGylation of Octreotide Using an α,β-unsaturated-β'-mono-sulfone Functionalized PEG Reagent

scientific article published on January 2012

Phenylimino-2H-chromen-3-carboxamide derivatives as novel small molecule inhibitors of β-secretase (BACE1).

scientific article published on 8 February 2013

Phthalimide-1,2,3-triazole hybrid compounds as tyrosinase inhibitors; synthesis, biological evaluation and molecular docking analysis

Phthalimide-Derived N-Benzylpyridinium Halides Targeting Cholinesterases: Synthesis and Bioactivity of New Potential Anti-Alzheimer's Disease Agents.

scientific article published on 22 February 2016

Polyoxygenated cinnamoylcoumarins as conformationally constrained analogs of cytotoxic diarylpentanoids: synthesis and biological activity.

scientific article published on 8 August 2013

Potent acetylcholinesterase inhibitors: design, synthesis, biological evaluation, and docking study of acridone linked to 1,2,3-triazole derivatives.

scientific article published on 22 January 2015

Protective effect of pentoxifylline on male Wistar rat testicular germ cell apoptosis induced by 3,4-methylenedioxymeth amphetamine

scientific article published on June 2016

Protective effects of physical exercise on MDMA-induced cognitive and mitochondrial impairment.

scientific article published on 21 July 2016

QSAR study of 4-aryl-4H-chromenes as a new series of apoptosis inducers using different chemometric tools

scientific article

Quinoline-based imidazole-fused heterocycles as new inhibitors of 15-lipoxygenase.

scientific article published on 17 July 2016

Recent applications of 1,3-thiazole core structure in the identification of new lead compounds and drug discovery

scientific article published on 13 April 2015

Replacement of the methylene of dihydrochalcones with oxygen: synthesis and biological evaluation of 2-phenoxyacetophenones

scientific article published on 13 July 2012

Structural features of new quinolones and relationship to antibacterial activity against Gram-positive bacteria

scientific article

Structure-based design, synthesis, molecular docking study and biological evaluation of 1,2,4-triazine derivatives acting as COX/15-LOX inhibitors with anti-oxidant activities

scientific article published on 30 March 2016

Synthesis and Biological Investigation of some Novel Sulfonamide and Amide Derivatives Containing Coumarin Moieties

scientific article

Synthesis and Docking Study of Novel 4-Thiazolidinone Derivatives as Anti-Gram-positive and Anti-H. pylori Agents

scientific article published on 01 January 2019

Synthesis and Evaluation of Chroman-4-One Linked to N-Benzyl Pyridinium Derivatives as New Acetylcholinesterase Inhibitors.

scientific article

Synthesis and In vitro cytotoxic activity evaluation of (E)-16-(substituted benzylidene) derivatives of dehydroepiandrosterone

scientific article published on May 2013

Synthesis and In-vitro Antibacterial Activities of Acetylanthracene and Acetylphenanthrene Derivatives of Some Fluoroquinolones

scientific article published on January 2011

Synthesis and anti-cancer activity evaluation of new dimethoxylated chalcone and flavanone analogs

scientific article published on 08 September 2014

Synthesis and anti-cholinesterase activity of new 7-hydroxycoumarin derivatives

scientific article published on 24 May 2014

Synthesis and antibacterial activity of new 7-piperazinyl-quinolones containing a functionalized 2-(furan-3-yl)ethyl moiety

scientific article published on 01 January 2007

Synthesis and antibacterial activity of new N-[2-(thiophen-3-yl)ethyl] piperazinyl quinolones

scientific article published on 01 June 2007

Synthesis and antibacterial activity of new fluoroquinolones containing a substituted N-(phenethyl)piperazine moiety

scientific article published on 27 April 2006

Synthesis and antibacterial activity of novel levofloxacin derivatives containing a substituted thienylethyl moiety

scientific article published on 30 August 2012

Synthesis and antibacterial activity of quinolone-based compounds containing a coumarin moiety

scientific article published in January 2008

Synthesis and anticancer activity of N-substituted 2-arylquinazolinones bearing trans-stilbene scaffold

scientific article published on 26 March 2015

Synthesis and anticholinergic activity of 4-hydroxycoumarin derivatives containing substituted benzyl-1,2,3-triazole moiety.

scientific article published on 20 July 2015

Synthesis and anticholinesterase activity of coumarin-3-carboxamides bearing tryptamine moiety.

scientific article

Synthesis and anticholinesterase activity of new substituted benzo[d]oxazole-based derivatives

scientific article published on 8 November 2016

Synthesis and antidiabetic evaluation of benzenesulfonamide derivatives

scientific article published on January 2013

Synthesis and antifungal activity of 1-[(2-benzyloxy)phenyl]-2-(azol-1-yl)ethanone derivatives: exploring the scaffold flexibility

scientific article published on 28 October 2011

Synthesis and biological evaluation of 2-phenylthiazole-4-carboxamide derivatives as anticancer agents

scientific article published on 16 September 2010

Synthesis and biological evaluation of 3-(trimethoxyphenyl)-2(3H)-thiazole thiones as combretastatin analogs.

scientific article published on 25 October 2013

Synthesis and biological evaluation of 4-amino-5-cinnamoylthiazoles as chalcone-like anticancer agents.

scientific article published on 6 January 2018

Synthesis and biological evaluation of 5-benzylidenerhodanine-3-acetic acid derivatives as AChE and 15-LOX inhibitors

scientific article published on 22 June 2015

Synthesis and biological evaluation of new N-benzylpyridinium-based benzoheterocycles as potential anti-Alzheimer's agents

scientific article published on 13 November 2018

Synthesis and biological evaluation of new coumarins bearing 2,4-diaminothiazole-5-carbonyl moiety

scientific article published on 07 June 2018

Synthesis and biological evaluation of novel benzyl piperazine derivatives of 5-(5-nitroaryl)-1,3,4-thiadiazoles as Anti-Helicobacter pylori agents

scientific article published on 08 August 2013

Synthesis and biological evaluation of novel imidazopyrimidin-3-amines as anticancer agents

scientific article published on 8 November 2016

Synthesis and cholinesterase inhibitory activity of new 2-benzofuran carboxamide-benzylpyridinum salts

scientific article published on 06 June 2018

Synthesis and cytotoxic activity of novel poly-substituted imidazo[2,1-c][1,2,4]triazin-6-amines

scientific article

Synthesis and cytotoxic evaluation of some new[1,3]dioxolo[4,5-g]chromen-8-one derivatives.

scientific article

Synthesis and cytotoxic properties of novel (E)-3-benzylidene-7-methoxychroman-4-one derivatives.

scientific article published on 12 April 2013

Synthesis and evaluation of antiproliferative activity of substituted N-(9-oxo-9H-xanthen-4-yl)benzenesulfonamides.

scientific article published on January 2014

Synthesis and in vitro cytotoxic activity of novel chalcone-like agents

scientific article

Synthesis and in-vitro antibacterial activity of 5-substituted 1-methyl-4-nitro-1H-imidazoles.

scientific article published in August 2008

Synthesis and in-vitro cytotoxicity of poly-functionalized 4-(2-arylthiazol-4-yl)-4H-chromenes.

scientific article published on July 2010

Synthesis and psychobiological evaluation of modafinil analogs in mice.

scientific article published on 19 December 2013

Synthesis and radioligand-binding assay of 2,5-disubstituted thiadiazoles and evaluation of their anticonvulsant activities

scientific article published on 27 August 2020

Synthesis and structure-activity relationship study of benzofuran-based chalconoids bearing benzylpyridinium moiety as potent acetylcholinesterase inhibitors.

scientific article

Synthesis and structure-activity relationship study of tacrine-based pyrano[2,3-c]pyrazoles targeting AChE/BuChE and 15-LOX.

scientific article published on 21 July 2016

Synthesis, biological evaluation and docking study of 3-aroyl-1-(4-sulfamoylphenyl)thiourea derivatives as 15-lipoxygenase inhibitors

scientific article published on 24 May 2014

Synthesis, evaluation, and molecular docking studies of aryl urea-triazole-based derivatives as anti-urease agents

scientific article published on 24 May 2018

Synthesis, in vitro cytotoxicity and apoptosis inducing study of 2-aryl-3-nitro-2H-chromene derivatives as potent anti-breast cancer agents

scientific article published on 6 September 2014

Synthesis, in vitro-antimycobacterial activity and cytotoxicity of some alkyl alpha-(5-aryl-1, 3, 4-thiadiazole-2-ylthio)acetates.

scientific article

The importance of synthetic drugs for type 2 diabetes drug discovery

scientific article

The importance of triazole scaffold in the development of anticonvulsant agents

scientific article published on 11 January 2016

Thiazole in the targeted anticancer drug discovery

scientific article published on 17 July 2019

Thiazolyl N-benzyl-substituted acetamide derivatives: synthesis, Src kinase inhibitory and anticancer activities

scientific article

Trastuzumab-monomethyl auristatin E conjugate exhibits potent cytotoxic activity in vitro against HER2-positive human breast cancer

scientific article published on 24 September 2018

Treatment of Helicobacter pylori infection: Current and future insights

scientific article

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