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List of works by Ewelina Węglarz-Tomczak

A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases

scientific article published on 9 April 2016

An integrated approach to the ligand binding specificity of Neisseria meningitidis M1 alanine aminopeptidase by fluorogenic substrate profiling, inhibitory studies and molecular modeling.

scientific article

Controlling the Helix Handedness of ααβ-Peptide Foldamers through Sequence Shifting

scientific article published on 12 January 2017

Controlling the Helix Handedness of ααβ-Peptide Foldamers through Sequence Shifting.

scientific article published on 12 January 2017

Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues

scientific article

Discovery of potent inhibitors of PLproCoV2 by screening a library of selenium-containing compounds

scientific article published on 21 May 2020

Ebselen as a highly active inhibitor of PLProCoV2

scientific article published on 18 May 2020

Estimating kinetic constants in the Michaelis-Menten model from one enzymatic assay using Approximate Bayesian Computation

scientific article published on 21 July 2019

Helix-loop-helix peptide foldamers and their use in the construction of hydrolase mimetics

scientific article published on 17 July 2018

Identification of ebselen and its analogues as potent covalent inhibitors of papain-like protease from SARS-CoV-2

scientific article

Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study.

scientific article published on 20 September 2016

M2R: a Python add-on to cobrapy for modifying human genome-scale metabolic reconstruction using the gut microbiota models

scientific article published in 2021

Neutral metalloaminopeptidases APN and MetAP2 as newly discovered anticancer molecular targets of actinomycin D and its simple analogs.

scientific article

Simultaneous Integration of Gene Expression and Nutrient Availability for Studying the Metabolism of Hepatocellular Carcinoma Cell Lines

scientific article published on 24 March 2021

Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases.

scientific article

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