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List of works by Josef Jampílek

1,3-substituted imidazolidine-2,4,5-triones: synthesis and inhibition of cholinergic enzymes ⬇️

scientific article published on 05 September 2011

5-Lipoxygenase, leukotrienes biosynthesis and potential antileukotrienic agents.

scientific article

A Rapid and Simple TLC-Densitometric Method for Assay of Clobetasol Propionate in Topical Solution.

scientific article published on 3 November 2017

Anti-infective and herbicidal activity of N-substituted 2-aminobenzothiazoles

scientific article published on 17 October 2012

Antibacterial and herbicidal activity of ring-substituted 3-hydroxynaphthalene-2-carboxanilides

scientific article published on 8 July 2013

Anticancer Efficacy of Antibacterial Quinobenzothiazines

scientific article published in 2023

Antifungal properties of new series of quinoline derivatives

scientific article published on 3 February 2006

Antimicrobial evaluation of some arylsulfanylpyrazinecarboxylic acid derivatives

scientific article published in May 2007

Antimycobacterial N-alkoxyphenylhydroxynaphthalenecarboxamides affecting photosystem II.

scientific article published on 21 March 2017

Asymmetric Primaquine and Halogenaniline Fumardiamides as Novel Biologically Active Michael Acceptors

scientific article published on 14 July 2018

Azone analogues: classification, design, and transdermal penetration principles ⬇️

scientific article published on November 9, 2010

Bioactivity of Methoxylated and Methylated 1-Hydroxynaphthalene-2-Carboxanilides: Comparative Molecular Surface Analysis

scientific article published on 18 August 2019

Biological Activities and ADMET-Related Properties of Novel Set of Cinnamanilides

scientific article published on 09 September 2020

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5

scientific article published on 30 June 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

scientific article published on 28 December 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4

scientific article published on 31 December 2018

Chronic Inflammatory Diseases, Anti-Inflammatory Agents and Their Delivery Nanosystems

scientific article published on 06 January 2021

Consensus-Based Pharmacophore Mapping for New Set of N-(disubstituted-phenyl)-3-hydroxyl-naphthalene-2-carboxamides

scientific article published on 09 September 2020

Design and Discovery of New Antibacterial Agents: Advances, Perspectives, Challenges

scientific article published on 18 September 2017

Design and synthesis of anticancer 1-hydroxynaphthalene-2-carboxanilides with a p53 independent mechanism of action

article

Designing a Dynamic Dissolution Method: A Review of Instrumental Options and Corresponding Physiology of Stomach and Small Intestine ⬇️

scientific article published on March 12, 2013

Determination of critical parameters of drug substance influencing dissolution: a case study

scientific article

Dibasic Derivatives of Phenylcarbamic Acid against Mycobacterial Strains: Old Drugs and New Tricks?

scientific article published on 28 September 2018

Graphenic Materials for Biomedical Applications

scientific article published on 11 December 2019

Halogenated 1-Hydroxynaphthalene-2-Carboxanilides Affecting Photosynthetic Electron Transport in Photosystem II.

scientific article published on 12 October 2017

Heterocycles in Medicinal Chemistry

scientific article published on 25 October 2019

How can we bolster the antifungal drug discovery pipeline?

scientific article published on 27 July 2016

In vitro bactericidal activity of 4- and 5-chloro-2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides against MRSA.

scientific article

In vitro permeation of micronized and nanonized alaptide from semisolid formulations

scientific article

Investigating Spectrum of Biological Activity of 4- and 5-Chloro-2-hydroxy-N-[2-(arylamino)-1-alkyl-2-oxoethyl]benzamides

scientific article published on 14 March 2011

Investigating biological activity spectrum for novel quinoline analogues

scientific article published on 14 November 2006

Investigating biological activity spectrum for novel quinoline analogues 2: hydroxyquinolinecarboxamides with photosynthesis-inhibiting activity

scientific article

Investigating the activity of 2-substituted alkyl-6-(2,5-dioxopyrrolidin-1-yl)hexanoates as skin penetration enhancers

scientific article published on 15 October 2010

Investigating the activity spectrum for ring-substituted 8-hydroxyquinolines.

scientific article published on 12 January 2010

Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenediones

scientific article published on 19 February 2010

Investigating the spectrum of biological activity of ring-substituted salicylanilides and carbamoylphenylcarbamates.

scientific article published on 10 November 2010

Investigation of Anti-Inflammatory Potential of N-Arylcinnamamide Derivatives

scientific article published on 11 December 2019

Investigation of Hydro-Lipophilic Properties of N-Alkoxyphenylhydroxynaphthalenecarboxamides †

scientific article published on 04 July 2018

Investigation of Permeation of Theophylline through Skin Using Selected Piperazine-2,5-Diones

scientific article published on 04 February 2019

Investigation of substituted 6-aminohexanoates as skin penetration enhancers

scientific article

Microwave-assisted synthesis of new substituted anilides of quinaldic acid

scientific article published on 31 January 2012

Modern Approaches to Quality Assurance of Drug Formulations.

scientific article published on 20 May 2015

Novel Benzene-Based Carbamates for AChE/BChE Inhibition: Synthesis and Ligand/Structure-Oriented SAR Study ⬇️

scientific article published on 27 March 2019

Photosynthesis-Inhibiting Activity of N-(Disubstituted-phenyl)-3-hydroxynaphthalene-2-carboxamides

scientific article published on 19 July 2021

Potassium Ferrate (VI) as the Multifunctional Agent in the Treatment of Landfill Leachate

scientific article published on 06 November 2020

Potential of Nanomaterial Applications in Dietary Supplements and Foods for Special Medical Purposes

Potential of Nanonutraceuticals in Increasing Immunity

scientific article published on 09 November 2020

Potential of agricultural fungicides for antifungal drug discovery

scientific article published on 7 November 2015

Preparation of candesartan and atorvastatin nanoparticles by solvent evaporation

Preparation of silica nanoparticles loaded with nootropics and their in vivo permeation through blood-brain barrier.

scientific article published on 17 May 2015

Primaquine hybrids as promising antimycobacterial and antimalarial agents

scientific article

Primary investigation of the preparation of nanoparticles by precipitation

Prodrugs: pharmaceutical design and current perspectives

scientific article published on 01 January 2011

Proline-Based Carbamates as Cholinesterase Inhibitors

scientific article published on 14 November 2017

Quinaldine derivatives: preparation and biological activity

scientific article published on 01 November 2005

RP-HPLC determination of the lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker

scientific article published on 28 March 2008

Recent Advances on Isoniazide Derivatives

scientific article published in January 2008

Recent advances in design of potential quinoxaline anti-infectives

scientific article

Rhodanineacetic acid derivatives as potential drugs: preparation, hydrophobic properties and antifungal activity of (5-arylalkylidene-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)acetic acids

scientific article published on 20 October 2009

Ring-Substituted 1-Hydroxynaphthalene-2-Carboxanilides Inhibit Proliferation and Trigger Mitochondria-Mediated Apoptosis ⬇️

scientific article published on 12 May 2020

Ring-substituted 4-hydroxy-1H-quinolin-2-ones: preparation and biological activity

scientific article published on 13 March 2009

Ring-substituted 8-hydroxyquinoline-2-carboxanilides as photosystem II inhibitors

scientific article published on 7 July 2016

Ring-substituted 8-hydroxyquinoline-2-carboxanilides as potential antimycobacterial agents

scientific article published on 29 June 2015

SAR-mediated Similarity Assessment of the Property Profile for New, Silicon-Based AChE/BChE Inhibitors ⬇️

scientific article published on 29 October 2019

Salicylanilide acetates: synthesis and antibacterial evaluation.

scientific article published on January 2007

Salicylanilide carbamates: Promising antibacterial agents with high in vitro activity against methicillin-resistant Staphylococcus aureus (MRSA).

scientific article published on 13 June 2015

Spectroscopic (FT-IR, FT-Raman) investigations and quantum chemical calculations of 4-hydroxy-2-oxo-1,2-dihydroquinoline-7-carboxylic acid

scientific article published on 9 November 2013

Study of Stability of New Mutual Prodrugs with Antimycobacterial Activity

scientific article published in May 2008

Substituted pyrazinecarboxamides: synthesis and biological evaluation.

scientific article published on 29 March 2006

Synthesis and Antimicrobial Evaluation of 1-[(2-Substituted phenyl)carbamoyl]naphthalen-2-yl Carbamates

scientific article published on 07 September 2016

Synthesis and In Vitro Antimycobacterial Activity of Novel N-Arylpiperazines Containing an Ethane-1,2-diyl Connecting Chain.

scientific article published on 30 November 2017

Synthesis and Spectrum of Biological Activities of Novel N-arylcinnamamides

scientific article published on 07 August 2018

Synthesis and antimicrobial evaluation of new 2-substituted 5,7-di-tert-butylbenzoxazoles.

scientific article published on 19 June 2006

Synthesis and antimycobacterial and photosynthesis-inhibiting evaluation of 2-[(E)-2-substituted-ethenyl]-1,3-benzoxazoles.

scientific article published on 13 August 2014

Synthesis and antimycobacterial evaluation of substituted pyrazinecarboxamides

scientific article published in May 2008

Synthesis, antimycobacterial, antifungal and photosynthesis-inhibiting activity of chlorinated N-phenylpyrazine-2-carboxamides.

scientific article published on 26 November 2010

Synthesis, physico-chemical properties and penetration activity of alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopyrrolidin-1-yl)hexanoates as potential transdermal penetration enhancers

scientific article published on 12 November 2009

Taguchi Method and Response Surface Methodology in the Treatment of Highly Contaminated Tannery Wastewater Using Commercial Potassium Ferrate.

scientific article

Targeting defective sphingosine kinase 1 in Niemann-Pick type C disease with an activator mitigates cholesterol accumulation

scientific article published on 08 May 2020

The Antimicrobial Activity of Annona emarginata (Schltdl.) H. Rainer and Most Active Isolated Compounds against Clinically Important Bacteria.

scientific article

The Forty-Sixth Euro Congress on Drug Synthesis and Analysis: Snapshot †.

scientific article published on 28 October 2017

The study of naphthoquinones and their complexes with DNA by using Raman spectroscopy and surface enhanced Raman spectroscopy: new insight into interactions of DNA with plant secondary metabolites.

scientific article

Towards Intelligent Drug Design System: Application of Artificial Dipeptide Receptor Library in QSAR-Oriented Studies

scientific article published on 06 August 2018

Utilization of NIR spectroscopy in candesartan cilexetil stability study

Vibrational spectroscopic and molecular docking study of (2E)-N-(4-chloro-2-oxo-1,2-dihydroquinolin-3-yl)-3-phenylprop-2-enamide

scientific article

Vibrational spectroscopic, 1H NMR and quantum chemical computational study of 4-hydroxy-2-oxo-1,2-dihydroquinoline-8-carboxylic acid

scientific article

X-ray and Thermal Analysis of Selected Drugs Containing Acetaminophen

scientific article published on 13 December 2020

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