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List of works by Piotr F J Lipiński

Affinity of fentanyl and its derivatives for the σ1-receptor

scientific article published on 13 June 2019

Antinociceptive and Cytotoxic Activity of Opioid Peptides with Hydrazone and Hydrazide Moieties at the C-Terminus

scientific article published on 28 July 2020

Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity

scientific article published on 08 September 2018

Chirality measures of α-amino acids.

scientific article

Conformational latitude - activity relationship of KPPR tetrapeptide analogues toward their ability to inhibit binding of vascular endothelial growth factor 165 to neuropilin-1.

scientific article published on 3 May 2017

Design, synthesis and in vitro biological evaluation of a small cyclic peptide as inhibitor of vascular endothelial growth factor binding to neuropilin-1

scientific article published on 21 April 2016

Fentanyl Family at the Mu-Opioid Receptor: Uniform Assessment of Binding and Computational Analysis

scientific article published on 19 February 2019

Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds.

scientific article published in November 2016

In Vivo, In Vitro and In Silico Studies of the Hybrid Compound AA3266, an Opioid Agonist/NK1R Antagonist with Selective Cytotoxicity

scientific article published on 19 October 2020

Molecular dynamics of fentanyl bound to μ-opioid receptor

scientific article published on 03 May 2019

On the Substituent Effect in the First Excited Singlet State of Monosubstituted Benzenes.

scientific article published on 26 April 2018

Radiochemical Synthesis and Evaluation of Novel Radioconjugates of Neurokinin 1 Receptor Antagonist Aprepitant Dedicated for NK1R-Positive Tumors

scientific article published on 18 August 2020

SCRAMBLE'N'GAMBLE: a tool for fast and facile generation of random data for statistical evaluation of QSAR models.

scientific article published on 5 June 2017

Structural Insights into σ₁ Receptor Interactions with Opioid Ligands by Molecular Dynamics Simulations.

scientific article published on 18 February 2018

Structural studies on radiopharmaceutical DOTA-minigastrin analogue (CP04) complexes and their interaction with CCK2 receptor.

scientific article published on 16 April 2018

Structure-activity relationship study of a small cyclic peptide H-c[Lys-Pro-Glu]-Arg-OH: a potent inhibitor of Vascular Endothelial Growth Factor interaction with Neuropilin-1.

scientific article published on 14 November 2016

Structure-activity relationship study of tetrapeptide inhibitors of the Vascular Endothelial Growth Factor A binding to Neuropilin-1.

scientific article published on 13 June 2017

The analgesic hybrid of dermorphin/substance P and analog of enkephalin improve wound healing in streptozotocin-induced diabetic rats

scientific article published on 19 November 2019

Triazolopeptides Inhibiting the Interaction between Neuropilin-1 and Vascular Endothelial Growth Factor-165.

scientific article published on 6 May 2019

β2-Homo-Amino Acid Scan of µ-Selective Opioid Tetrapeptide TAPP

scientific article published on 25 May 2020