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List of works by Kamil Kuder

(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands

scientific article published on 10 August 2015

4-tert-Pentylphenoxyalkyl derivatives - Histamine H receptor ligands and monoamine oxidase B inhibitors

scientific article published on 31 October 2018

8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation

scientific article published on 19 June 2020

A Taxicab geometry quantification system to evaluate the performance of in silico methods: a case study on adenosine receptors ligands

scientific article published on 28 February 2020

Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands

scientific article published on 12 February 2019

Anticonvulsive effect of nonimidazole histamine H3 receptor antagonists.

scientific article published in June 2014

Aryl-1,3,5-triazine derivatives as histamine H4 receptor ligands.

scientific article

Chlorophenoxy aminoalkyl derivatives as histamine H(3)R ligands and antiseizure agents.

scientific article published on 2 December 2015

Cholinesterase inhibitory activity of chlorophenoxy derivatives-Histamine H3 receptor ligands.

scientific article published on 20 April 2016

Corrigendum to "Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands" [Eur. J. Med. Chem. 185 (2020) 111785]

scientific article published on 10 August 2020

Diether (substituted) piperidine derivatives as novel, histamine H3 receptor ligands.

scientific article published in April 2009

Diether derivatives of homo- or substituted piperidines as non-imidazole histamine H3 receptor ligands

scientific article

Discovery of Potential, Dual-Active Histamine H Receptor Ligands with Combined Antioxidant Properties

scientific article published on 15 April 2021

Discovery of novel lead in the group of N-substituted piperazine ether derivatives with potential histamine H3 receptor activity.

scientific article published in January 2014

Dual-acting diether derivatives of piperidine and homopiperidine with histamine H(3) receptor antagonistic and anticholinesterase activity

scientific article published on 02 May 2012

Dual-targeting approach on histamine H3 and sigma-1 receptor ligands as promising pharmacological tools in the treatment of CNS-linked disorders

scientific article published on 05 August 2020

Fluorescent GPCR ligands as new tools in pharmacology-update, years 2008-early 2014.

scientific article published on January 2014

Fluorescent GPCR ligands as new tools in pharmacology.

scientific article published on January 2008

H3 histamine receptor antagonist pitolisant reverses some subchronic disturbances induced by olanzapine in mice.

scientific article published on 24 May 2016

Histamine H Receptor Ligands-KSK-59 and KSK-73-Reduce Body Weight Gain in a Rat Model of Excessive Eating

scientific article published on 25 October 2021

Histamine H3 receptor ligands in the group of (homo)piperazine derivatives

scientific article published on 23 November 2017

KSK19 - Novel histamine H3 receptor ligand reduces body weight in diet induced obese mice

scientific article published on 08 July 2019

Monocyclic and Fused Azines and Azoles as Histamine H₄ Receptor Ligands

scientific article published on 11 April 2016

N-substituted piperazine derivatives as potential multitarget agents acting on histamine H3 receptor and cancer resistance proteins

scientific article published on 29 August 2020

Non-imidazole-based histamine H3 receptor antagonists with anticonvulsant activity in different seizure models in male adult rats.

scientific article

Novel multi-target directed ligands based on annelated xanthine scaffold with aromatic substituents acting on adenosine receptor and monoamine oxidase B. Synthesis, in vitro and in silico studies

scientific article published on 02 February 2019

Novel, Dual Target-Directed Annelated Xanthine Derivatives Acting on Adenosine Receptors and Monoamine Oxidase B

scientific article published on 12 March 2020

Optimization and preclinical evaluation of novel histamine H3receptor ligands: Acetyl and propionyl phenoxyalkyl piperazine derivatives

scientific article published on 10 November 2018

Piperidine variations in search for non-imidazole histamine H(3) receptor ligands.

scientific article

Probing an artificial polypeptide receptor library using a series of novel histamine H3 receptor ligands

scientific article

Rational design of new multitarget histamine H3 receptor ligands as potential candidates for treatment of Alzheimer's disease

scientific article published on 21 August 2020

Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands

scientific article published on 17 October 2019

Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties

scientific article

Structural modifications and in vitro pharmacological evaluation of 4-pyridyl-piperazine derivatives as an active and selective histamine H3 receptor ligands

scientific article published on 20 June 2019

Structural modifications in the distal, regulatory region of histamine H<sub>3</sub> receptor antagonists leading to the identification of a potent anti-obesity agent

scientific article published on 24 November 2020

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

scientific article

Synthesis and biological activity of novel tert-butyl and tert-pentylphenoxyalkyl piperazine derivatives as histamine H3R ligands

Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.

scientific article

The histamine H3 receptor inverse agonist pitolisant reduces body weight in obese mice

scientific article published on 25 May 2018