List of works - Carmen Di Giovanni

Amorfrutins are efficient modulators of peroxisome proliferator-activated receptor gamma (PPARγ) with potent antidiabetic and anticancer properties: a patent evaluation of WO2014177593 A1.

scientific article published in January 2015

Antidepressive effects of a chemically characterized maqui berry extract (Aristotelia chilensis (molina) stuntz) in a mouse model of Post-stroke depression

scientific article published on 22 April 2019

Benzothiopyranoindole-Based Antiproliferative Agents: Synthesis, Cytotoxicity, Nucleic Acids Interaction, and Topoisomerases Inhibition Properties

scientific article published on 01 September 2009

CDC25A and B dual-specificity phosphatase inhibitors: potential agents for cancer therapy.

scientific article published on January 2009

Conformational switch of a flexible loop in human laminin receptor determines laminin-1 interaction

scientific article published on 01 March 2012

Determination of cymoxanil in drinking water and soil using high-performance liquid chromatography.

scientific article

Development of novel selective peptidomimetics containing a boronic acid moiety, targeting the 20S proteasome as anticancer agents

scientific article

Development of peptidomimetic boronates as proteasome inhibitors

article

Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition

scientific article published on 25 January 2012

Discovery of New Inhibitors of Cdc25B Dual Specificity Phosphatases by Structure-Based Virtual Screening

scientific article published on 01 May 2012

Discovery of a novel small molecule inhibitor targeting the frataxin/ubiquitin interaction via structure-based virtual screening and bioassays

scientific article

Discovery of new small molecules inhibiting 67 kDa laminin receptor interaction with laminin and cancer cell invasion

scientific article

Hydromethanolic Extracts from Adansonia digitata L. Edible Parts Positively Modulate Pathophysiological Mechanisms Related to the Metabolic Syndrome

scientific article published on 21 June 2020

Identification of a new series of amides as non-covalent proteasome inhibitors.

scientific article published on 25 January 2014

Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure-based virtual screening.

scientific article

Inhibitors of Cdc25 phosphatases as anticancer agents: a patent review

scientific article published on March 2010

Investigational drugs targeting cyclin-dependent kinases for the treatment of cancer: an update on recent findings (2013-2016).

scientific article published on 8 September 2016

Ligand-based chemoinformatic discovery of a novel small molecule inhibitor targeting CDC25 dual specificity phosphatases and displaying in vitro efficacy against melanoma cells

scientific article published on 13 October 2015

New 2-(aryloxy)-3-phenylpropanoic acids as peroxisome proliferator-activated receptor α/γ dual agonists able to upregulate mitochondrial carnitine shuttle system gene expression

scientific article

Novel inhibitors of signal transducer and activator of transcription 3 signaling pathway: an update on the recent patent literature.

scientific article published on 16 January 2014

Novel non-peptide small molecules preventing IKKβ/NEMO association inhibit NF-κB activation in LPS-stimulated J774 macrophages.

scientific article published on 14 January 2016

Novel quinolinonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, and biological activities

scientific article published on 23 July 2008

STAT-3 inhibitors: state of the art and new horizons for cancer treatment.

scientific article published on January 2011

Structural development studies of PPARs ligands based on tyrosine scaffold

scientific article published on 31 October 2014

Synthesis, biological evaluation and molecular investigation of fluorinated peroxisome proliferator-activated receptors α/γ dual agonists

scientific article

Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity

scientific article

Virtual screening strategies in drug discovery: a critical review.

scientific article published on January 2013

List of works by Carmen Di Giovanni

Amorfrutins are efficient modulators of peroxisome proliferator-activated receptor gamma (PPARγ) with potent antidiabetic and anticancer properties: a patent evaluation of WO2014177593 A1.

Antidepressive effects of a chemically characterized maqui berry extract (Aristotelia chilensis (molina) stuntz) in a mouse model of Post-stroke depression

Benzothiopyranoindole-Based Antiproliferative Agents: Synthesis, Cytotoxicity, Nucleic Acids Interaction, and Topoisomerases Inhibition Properties

CDC25A and B dual-specificity phosphatase inhibitors: potential agents for cancer therapy.

Conformational switch of a flexible loop in human laminin receptor determines laminin-1 interaction

Determination of cymoxanil in drinking water and soil using high-performance liquid chromatography.

Development of novel selective peptidomimetics containing a boronic acid moiety, targeting the 20S proteasome as anticancer agents

Development of peptidomimetic boronates as proteasome inhibitors

Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition

Discovery of New Inhibitors of Cdc25B Dual Specificity Phosphatases by Structure-Based Virtual Screening

Discovery of a novel small molecule inhibitor targeting the frataxin/ubiquitin interaction via structure-based virtual screening and bioassays

Discovery of new small molecules inhibiting 67 kDa laminin receptor interaction with laminin and cancer cell invasion

Hydromethanolic Extracts from Adansonia digitata L. Edible Parts Positively Modulate Pathophysiological Mechanisms Related to the Metabolic Syndrome

Identification of a new series of amides as non-covalent proteasome inhibitors.

Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure-based virtual screening.

Inhibitors of Cdc25 phosphatases as anticancer agents: a patent review

Investigational drugs targeting cyclin-dependent kinases for the treatment of cancer: an update on recent findings (2013-2016).

Ligand-based chemoinformatic discovery of a novel small molecule inhibitor targeting CDC25 dual specificity phosphatases and displaying in vitro efficacy against melanoma cells

New 2-(aryloxy)-3-phenylpropanoic acids as peroxisome proliferator-activated receptor α/γ dual agonists able to upregulate mitochondrial carnitine shuttle system gene expression

Novel inhibitors of signal transducer and activator of transcription 3 signaling pathway: an update on the recent patent literature.

Novel non-peptide small molecules preventing IKKβ/NEMO association inhibit NF-κB activation in LPS-stimulated J774 macrophages.

Novel quinolinonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, and biological activities

STAT-3 inhibitors: state of the art and new horizons for cancer treatment.

Structural development studies of PPARs ligands based on tyrosine scaffold

Synthesis, biological evaluation and molecular investigation of fluorinated peroxisome proliferator-activated receptors α/γ dual agonists

Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity

Virtual screening strategies in drug discovery: a critical review.