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List of works by Isao Sakurada

Development of a novel class of potent and selective FIXa inhibitors

scientific article

Development of a novel tricyclic class of potent and selective FIXa inhibitors

scientific article

Discovery and preclinical characterization of 1-methyl-3-(4-methylpyridin-3-yl)-6-(pyridin-2-ylmethoxy)-1H-pyrazolo-[3,4-b]pyrazine (PF470): a highly potent, selective, and efficacious metabotropic glutamate receptor 5 (mGluR5) negative allosteric m

scientific article published on 22 January 2014

Discovery of (-)-6-[2-[4-(3-fluorophenyl)-4-hydroxy-1-piperidinyl]-1-hydroxyethyl]-3,4-dihydro-2(1H)-quinolinone--a potent NR2B-selective N-methyl D-aspartate (NMDA) antagonist for the treatment of pain

scientific article published on 15 August 2007

Discovery of novel aminobenzisoxazole derivatives as orally available factor IXa inhibitors

scientific article published on 6 March 2017

Discovery of novel and orally active NR2B-selective N-methyl-D-aspartate (NMDA) antagonists, pyridinol derivatives with reduced HERG binding affinity

scientific article published on 22 August 2007

Structure-activity relationship study of novel NR2B-selective antagonists with arylamides to avoid reactive metabolites formation.

scientific article published on 19 August 2007

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