Search filters

List of works by Gweneal Chevé

A combined ligand-based and target-based drug design approach for G-protein coupled receptors: application to salvinorin A, a selective kappa opioid receptor agonist.

scientific article

Axl kinase as a key target for oncology: focus on small molecule inhibitors

scientific article

Comparative protein modeling of 1-deoxy-D-xylulose-5-phosphate reductoisomerase enzyme from Plasmodium falciparum: a potential target for antimalarial drug discovery.

scientific article

Design, synthesis, and biological evaluation of bifunctional thyrointegrin inhibitors: new anti-angiogenesis analogs

scientific article published on 14 March 2011

Determination and validation of mTOR kinase-domain 3D structure by homology modeling

scientific article published on 30 July 2015

Increased susceptibility of low-density lipoprotein to ex vivo oxidation in mice transgenic for human apolipoprotein B treated with 1 melatonin-related compound is not associated with atherosclerosis progression

scientific article published in September 2005

Recent advances in drug design of epidermal growth factor receptor inhibitors

scientific article published on January 2013

Recent progress in the design, study, and development of c-Jun N-terminal kinase inhibitors as anticancer agents.

scientific article

Structural elucidation of the DFG-Asp in and DFG-Asp out states of TAM kinases and insight into the selectivity of their inhibitors.

scientific article published on 10 October 2014

Structure-activity relationships of neuropeptide FF and related peptidic and non-peptidic derivatives.

scientific article

Targeting the methyl erythritol phosphate (MEP) pathway for novel antimalarial, antibacterial and herbicidal drug discovery: inhibition of 1-deoxy-D-xylulose-5-phosphate reductoisomerase (DXR) enzyme.

scientific article published on January 2007