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List of works by Allan J B Watson

A Multicomponent Route to Functionalized Amides and Oxazolidinones

scientific article published on 01 December 2017

A flow platform for degradation-free CuAAC bioconjugation

scientific article published in Nature Communications

A modular synthesis of functionalised phenols enabled by controlled boron speciation

scientific article published on 01 March 2015

A one-pot tandem chemoselective allylation/cross-coupling via temperature control of a multi-nucleophile/electrophile system

scientific article published on 01 August 2017

Amidation of esters with amino alcohols using organobase catalysis

scientific article published on 16 September 2014

Amidation of unactivated ester derivatives mediated by trifluoroethanol

scientific article published on 01 April 2017

Biocatalytic Synthesis of Chiral N-Functionalized Amino Acids

scientific article published on 21 September 2018

Bismesitylmagnesium: a thermally stable and non-nucleophilic carbon-centred base reagent for the efficient preparation of silyl enol ethers

scientific article published on 27 September 2007

Catalytic Enantioselective Synthesis of α-Chiral Azaheteroaryl Ethylamines by Asymmetric Protonation

scientific article published on 01 August 2018

Chan-Evans-Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine Problem

scientific article published on 18 April 2016

Chemoselective One-Pot Synthesis of Functionalized Amino-azaheterocycles Enabled by COware

scientific article published on 14 November 2017

Chemoselective Suzuki-Miyaura Cross-Coupling via Kinetic Transmetallation.

scientific article

Chemoselective boronic ester synthesis by controlled speciation.

scientific article published on 29 September 2014

Chemoselective oxidation of aryl organoboron systems enabled by boronic acid-selective phase transfer

scientific article

Contra-Thermodynamic, Photocatalytic E→Z Isomerization of Styrenyl Boron Species: Vectors to Facilitate Exploration of 2D Chemical Space.

scientific article published on 2 February 2018

Correction to "Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides".

scientific article published on 2 August 2017

Cyrene as a bio-based solvent for HATU mediated amide coupling

scientific article published on 01 April 2018

Deoxyfluorination with CuF2 : Enabled by Using a Lewis Base Activating Group

scientific article published on 28 February 2020

Determining the Origin of Rate-Independent Chemoselectivity in CuAAC Reactions: An Alkyne-Specific Shift in Rate-Determining Step.

scientific article published on 16 February 2017

Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second Bromodomain.

scientific article published on 15 April 2018

Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.

scientific article published on 30 January 2017

First experimental evidence for a bis-ethene chromium(I) complex forming from an activated ethene oligomerization catalyst

scientific article published on 18 December 2020

In situ generation of Mes2Mg as a non-nucleophilic carbon-centred base reagent for the efficient one-pot conversion of ketones to silyl enol ethers.

scientific article

Interrogating Pd(II) Anion Metathesis Using a Bifunctional Chemical Probe: A Transmetalation Switch.

scientific article published on 19 December 2017

Mechanism of Cu-Catalyzed Aryl Boronic Acid Halodeboronation Using Electrophilic Halogen: Development of a Base-Catalyzed Iododeboronation for Radiolabeling Applications

scientific article published on 25 March 2019

Mechanistic Development and Recent Applications of the Chan-Lam Amination

scientific article published on 22 November 2019

Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides.

scientific article published on 6 July 2017

N-Alkyl-α-amino acids in Nature and their biocatalytic preparation

scientific article published on 26 January 2019

Ni vs. Pd in Suzuki-Miyaura sp2-sp2 cross-coupling: a head-to-head study in a comparable precatalyst/ligand system

scientific article published on 03 May 2019

One-Pot Homologation of Boronic Acids: A Platform for Diversity-Oriented Synthesis

scientific article published on 03 December 2015

Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.

scientific article published on 30 November 2017

Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators

scientific article

Scalable total synthesis and comprehensive structure-activity relationship studies of the phytotoxin coronatine.

scientific article published on 16 March 2018

Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation

scientific article (publication date: 2016)

Soft scorpionate anions as platforms for novel heterocycles.

scientific article

Speciation control during Suzuki-Miyaura cross-coupling of haloaryl and haloalkenyl MIDA boronic esters

scientific article published on 08 May 2015

Spectroscopic Studies of the Chan-Lam Amination: A Mechanism-Inspired Solution to Boronic Ester Reactivity.

scientific article

Strategy for Conditional Orthogonal Sequential CuAAC Reactions Using a Protected Aromatic Ynamine.

scientific article published on 28 April 2017

Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode

scientific article

Synthesis of 2-BMIDA 6,5-bicyclic heterocycles by Cu(i)/Pd(0)/Cu(ii) cascade catalysis of 2-iodoaniline/phenols

scientific article published on 01 July 2016

Synthesis of functionalised 4H-quinolizin-4-ones via tandem Horner-Wadsworth-Emmons olefination/cyclisation.

scientific article published in May 2013

Tandem Chemoselective Suzuki-Miyaura Cross-Coupling Enabled by Nucleophile Speciation Control

scientific article published in July 2015

Towards energetically viable asymmetric deprotonations: selectivity at more elevated temperatures with C2-symmetric magnesium bisamides

scientific article published on 18 January 2011

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