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List of works by Allen Duplantier

1-[(1-Methyl-1H-imidazol-2-yl)methyl]-4-phenylpiperidines as mGluR2 Positive Allosteric Modulators for the Treatment of Psychosis ⬇️

scientific article published on March 2, 2011

3-(Imidazolyl methyl)-3-aza-bicyclo[3.1.0]hexan-6-yl)methyl ethers: a novel series of mGluR2 positive allosteric modulators.

scientific article

7-Oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridines as novel inhibitors of human eosinophil phosphodiesterase.

scientific article published on June 1998

Discovering Drugs for the Treatment of Ebola Virus.

scientific article published on 4 August 2017

Discovery of 4-(5-methyloxazolo[4,5-b]pyridin-2-yl)-1,4-diazabicyclo[3.2.2]nonane (CP-810,123), a novel alpha 7 nicotinic acetylcholine receptor agonist for the treatment of cognitive disorders in schizophrenia: synthesis, SAR development, and in vi

scientific article published in February 2010

Discovery of a novel Kv7 channel opener as a treatment for epilepsy.

scientific article published on May 2015

Discovery, SAR, and pharmacokinetics of a novel 3-hydroxyquinolin-2(1H)-one series of potent D-amino acid oxidase (DAAO) inhibitors

scientific article

Discovery, synthesis and SAR of azinyl- and azolylbenzamides antagonists of the P2X₇ receptor.

scientific article published on 2 July 2011

Galanin function in the central nervous system

scientific article published on September 2006

Isoxazolyl, oxazolyl, and thiazolylpropionic acid derivatives as potent alpha(4)beta(1) integrin antagonists

scientific article

Mitigating the Impact of Antibacterial Drug Resistance through Host-Directed Therapies: Current Progress, Outlook, and Challenges.

scientific article

Modulation of NMDA receptor function by inhibition of D-amino acid oxidase in rodent brain.

scientific article

New Steroidal 4-Aminoquinolines Antagonize Botulinum Neurotoxin Serotype A in Mouse Embryonic Stem Cell Derived Motor Neurons in Post-intoxication Model.

scientific article published on 31 January 2018

Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X7 receptor antagonists leading to the discovery of the clinical candidate CE-224,535.

scientific article published on 24 April 2011

Robust biofilm assay for quantification and high throughput screening applications

scientific article published on 28 February 2019

SAR of a series of 5,6-dihydro-(9H)-pyrazolo[3,4-c]-1,2,4-triazolo[4,3-alpha]pyridines as potent inhibitors of human eosinophil phosphodiesterase

scientific article published on 01 January 2007

Searching for Therapeutics Against Botulinum Neurotoxins: A True Challenge for Drug Discovery.

scientific article published on 13 April 2016

Second generation of diazachrysenes: Protection of Ebola virus infected mice and mechanism of action

scientific article published on 31 October 2018

Synthesis of [F]Favipiravir and Biodistribution in C3H/HeN Mice as Assessed by Positron Emission Tomography

scientific article published in Scientific Reports

Systematic N-methylation of oxytocin: Impact on pharmacology and intramolecular hydrogen bonding network.

scientific article published on 31 May 2016

The Human Cathelicidin Antimicrobial Peptide LL-37 as a Potential Treatment for Polymicrobial Infected Wounds

scientific article published on 03 July 2013

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