List of works - Adam Kraszewski

31P NMR Studies on Oxidative Transformations of Aryl Nucleoside H-Phosphonate Diesters

A cautionary note on the use of the 31P NMR spectroscopy in stereochemical correlation analysis

scientific article

A convenient stereochemical notation for p-chiral nucleotide analogs

scientific article published on 01 March 2007

A new method for the synthesis of nucleoside 2′,3′-O,O-cyclic phosphorodithioates via aryl cyclic phosphites as intermediates

article published in 2001

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 2. Dinucleoside monophosphate analogues

scientific article published in January 2006

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 4. A relationship between the Dp/Lp notation and stereochemistry of reactions

scientific article

A proposal for a convenient notation forP-chiral nucleotide analogues. Part 3. Compounds with one nucleoside residue and nonnucleosidic derivatives

scientific article published on 01 January 2006

A proposal for a new stereochemical notation for P-chiral nucleotide analogues and related compounds

scientific article published in January 2005

ARYL NUCLEOSIDE H-PHOSPHONATES AS A TOOL FOR INVESTIGATION OF STEREOSPECIFICITY DURING COUPLING

scientific article published on 01 January 2005

Aryl H-Phosphonates 18. Synthesis, properties, and biological activity of 2',3'-dideoxynucleoside (N-heteroaryl)phosphoramidates of increased lipophilicity

scientific article published on 4 June 2015

Aryl H-phosphonates 17: (N-aryl)phosphoramidates of pyrimidine nucleoside analogues and their synthesis, selected properties, and anti-HIV activity

scientific article published on 9 September 2011

Aryl H-phosphonates. 19. New anti-HIV pronucleotide phosphoramidate diesters containing amino- and hydroxypyridine auxiliaries

scientific article published on 17 December 2018

Aryl H-phosphonates. Part IV. A new method for internucleotide bond formation based on transesterification of aryl nucleoside H-phosphonate diesters

article published in 1996

Aryl nucleoside H-phosphonates. Part 15: Synthesis, properties and, anti-HIV activity of aryl nucleoside 5'-alpha-hydroxyphosphonates

scientific article published on 14 November 2005

Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters

scientific article published on 23 February 2009

ArylH-Phosphonates. 14. Synthesis of New Nucleotide Analogues with Phosphonate−Phosphate Internucleosidic Linkage

scientific article published on 01 October 2003

ArylH-Phosphonates. 6. Synthetic Studies on the Preparation of NucleosideN-Alkyl-H-phosphonamidates

Chemical and Stereochemical Aspects of Oxidative Coupling of HPhosphonate and H-Phosphonothioate Diesters. Reactions with N,N-, N,Oand O,O-Binucleophiles

Chemical synthesis of genes for human insulin ⬇️

scientific article published on December 1, 1978

Chemoselectivity in oxidative coupling of bifunctional nucleophiles with dinucleoside H-phosphonate and dinucleoside H-phosphonothioate diesters

scientific article published on 01 May 2003

DEVELOPING SYNTHETIC METHODS FOR BIOACTIVE PHOSPHORUS COMPOUNDS USING H-PHOSPHONATE CHEMISTRY: A PROGRESS REPORT

scientific article published on 01 January 2005

Developing Synthetic Methods for Bioactive Phosphorus Compounds Using H-Phosphonate Chemistry: A Progress Report

scientific article published on 01 May 2003

Different nucleobase orientations in two cyclic 2',3'-phosphates of purine ribonucleosides: Et(3)NH(2',3'-cAMP) and Et(3)NH(2',3'-cGMP)xH(2)O

scientific article published on 15 June 2006

Exploring Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents

H-Phosphonate Chemistry in the Synthesis of Electrically Neutral and Charged Antiviral and Anticancer Pronucleotides

scientific article

H-Phosphonates: Versatile synthetic precursors to biologically active phosphorus compounds

How to get the most out of two phosphorus chemistries. Studies on H-phosphonates

scientific article

New 3'-O-aromatic acyl-5-fluoro-2'-deoxyuridine derivatives as potential anticancer agents

scientific article published on 04 March 2016

New antiglioma zwitterionic pronucleotides with an FdUMP framework

scientific article published on 21 December 2017

Novel reactivity of Fhit proteins: catalysts for fluorolysis of nucleoside 5'-phosphoramidates and nucleoside 5'-phosphosulfates to generate nucleoside 5'-phosphorofluoridates

scientific article published on 01 June 2015

Nucleoside 3′,5′-Cyclic H-Phosphonates, New Useful Precursors for the Synthesis of Nucleoside 3′,5′-Cyclic Phosphates and Their Analogues

scientific article published on 01 August 2013

Nucleoside Phosphonates. Development of Synthetic Methods and Reagents

NucleosideH-Phosphonates. 18. Synthesis of Unprotected Nucleoside 5‘-H-Phosphonates and Nucleoside 5‘-H-Phosphonothioates and Their Conversion into the 5‘-Phosphorothioate and 5‘-Phosphorodithioate Monoesters

Prevalence of beta allele of the insulin gene in type II diabetes mellitus.

scientific article published in March 1994

Recent Advances in H-Phosphonate Chemistry. Part 2. Synthesis of C-Phosphonate Derivatives

scientific article published on 01 January 2015

Recent advances in H-phosphonate chemistry. Part 1. H-phosphonate esters: synthesis and basic reactions

scientific article

Reinvestigation of the 31P NMR evidence for the formation of diorganyl phosphoropyridinium intermediates

article

Searching for anti-glioma activity. Ribonucleoside analogues with modifications in nucleobase and sugar moieties

scientific article published on 10 November 2016

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 1. Synthesis and 31P NMR analysis of 16 diribonulceoside (3'-5')-H-phosphonates and the corresponding phosphorothioates

scientific article

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 5. The role of Brønsted and H-bonding base catalysis in ribonucleoside H-phosphonate condensation-chemical and stereochemical consequences

scientific article published on August 2010

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 7. Stereoselective formation of ribonucleoside (RP)- and (SP)-3′-H-phosphonothioate monoesters

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 3: Investigations on a mechanism of asymmetric induction

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 6: Optimization of the reaction conditions towards highest stereoselectivity

Studies on Aryl H-Phosphonates. Synthesis of Nucleoside N-Alkylphosphonamidates

Studies on Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents. Part III. Further Studies on Transesterification of Nucleoside H-Phosphonate Diesters with Amino Alcohols

Studies on aryl H-phosphonates. 3. Mechanistic investigations related to the disproportionation of diphenyl H-phosphonate under anhydrous basic conditions

Studies on aryl H-phosphonates. I. An efficient method for the preparation of deoxyribo- and ribonucleoside 3′-H-phosphonate monoesters by transesterification of diphenyl H-phosphonate

Studies on reactions of nucleoside H-phosphonate diesters with bifunctional reagents. Part 4. Chemoselectivity during oxidative coupling of nucleoside H-phosphonate diesters with amino alcohols controlled by protonation of the amino function

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 1. Reaction with amino alcohols

article published in 1993

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 2. Stability of nucleoside H-phosphonate diesters in the presence of amino alcohols

Studies on the decomposition pathways of diastereoisomeric mixtures of aryl nucleoside α-hydroxyphosphonates under hydrolytic conditions. Synthesis of α-hydroxyphosphonate monoesters

The case of sulfonation in the chemical synthesis of oligonucleotides ⬇️

scientific article published on May 24, 1980

The case of triethylammonium cation loss during purification of certain nucleotide analogues: a cautionary note

scientific article

List of works by Adam Kraszewski

31P NMR Studies on Oxidative Transformations of Aryl Nucleoside H-Phosphonate Diesters

A cautionary note on the use of the 31P NMR spectroscopy in stereochemical correlation analysis

A convenient stereochemical notation for p-chiral nucleotide analogs

A new method for the synthesis of nucleoside 2′,3′-O,O-cyclic phosphorodithioates via aryl cyclic phosphites as intermediates

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 2. Dinucleoside monophosphate analogues

A proposal for a convenient notation for P-chiral nucleotide analogues. Part 4. A relationship between the Dp/Lp notation and stereochemistry of reactions

A proposal for a convenient notation forP-chiral nucleotide analogues. Part 3. Compounds with one nucleoside residue and nonnucleosidic derivatives

A proposal for a new stereochemical notation for P-chiral nucleotide analogues and related compounds

ARYL NUCLEOSIDE H-PHOSPHONATES AS A TOOL FOR INVESTIGATION OF STEREOSPECIFICITY DURING COUPLING

Aryl H-Phosphonates 18. Synthesis, properties, and biological activity of 2',3'-dideoxynucleoside (N-heteroaryl)phosphoramidates of increased lipophilicity

Aryl H-phosphonates 17: (N-aryl)phosphoramidates of pyrimidine nucleoside analogues and their synthesis, selected properties, and anti-HIV activity

Aryl H-phosphonates. 19. New anti-HIV pronucleotide phosphoramidate diesters containing amino- and hydroxypyridine auxiliaries

Aryl H-phosphonates. Part IV. A new method for internucleotide bond formation based on transesterification of aryl nucleoside H-phosphonate diesters

Aryl nucleoside H-phosphonates. Part 15: Synthesis, properties and, anti-HIV activity of aryl nucleoside 5'-alpha-hydroxyphosphonates

Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters

ArylH-Phosphonates. 14. Synthesis of New Nucleotide Analogues with Phosphonate−Phosphate Internucleosidic Linkage

ArylH-Phosphonates. 6. Synthetic Studies on the Preparation of NucleosideN-Alkyl-H-phosphonamidates

Chemical and Stereochemical Aspects of Oxidative Coupling of HPhosphonate and H-Phosphonothioate Diesters. Reactions with N,N-, N,Oand O,O-Binucleophiles

Chemical synthesis of genes for human insulin ⬇️

Chemoselectivity in oxidative coupling of bifunctional nucleophiles with dinucleoside H-phosphonate and dinucleoside H-phosphonothioate diesters

DEVELOPING SYNTHETIC METHODS FOR BIOACTIVE PHOSPHORUS COMPOUNDS USING H-PHOSPHONATE CHEMISTRY: A PROGRESS REPORT

Developing Synthetic Methods for Bioactive Phosphorus Compounds Using H-Phosphonate Chemistry: A Progress Report

Different nucleobase orientations in two cyclic 2',3'-phosphates of purine ribonucleosides: Et(3)NH(2',3'-cAMP) and Et(3)NH(2',3'-cGMP)xH(2)O

Exploring Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents

H-Phosphonate Chemistry in the Synthesis of Electrically Neutral and Charged Antiviral and Anticancer Pronucleotides

H-Phosphonates: Versatile synthetic precursors to biologically active phosphorus compounds

How to get the most out of two phosphorus chemistries. Studies on H-phosphonates

New 3'-O-aromatic acyl-5-fluoro-2'-deoxyuridine derivatives as potential anticancer agents

New antiglioma zwitterionic pronucleotides with an FdUMP framework

Novel reactivity of Fhit proteins: catalysts for fluorolysis of nucleoside 5'-phosphoramidates and nucleoside 5'-phosphosulfates to generate nucleoside 5'-phosphorofluoridates

Nucleoside 3′,5′-Cyclic H-Phosphonates, New Useful Precursors for the Synthesis of Nucleoside 3′,5′-Cyclic Phosphates and Their Analogues

Nucleoside Phosphonates. Development of Synthetic Methods and Reagents

NucleosideH-Phosphonates. 18. Synthesis of Unprotected Nucleoside 5‘-H-Phosphonates and Nucleoside 5‘-H-Phosphonothioates and Their Conversion into the 5‘-Phosphorothioate and 5‘-Phosphorodithioate Monoesters

Prevalence of beta allele of the insulin gene in type II diabetes mellitus.

Recent Advances in H-Phosphonate Chemistry. Part 2. Synthesis of C-Phosphonate Derivatives

Recent advances in H-phosphonate chemistry. Part 1. H-phosphonate esters: synthesis and basic reactions

Reinvestigation of the 31P NMR evidence for the formation of diorganyl phosphoropyridinium intermediates

Searching for anti-glioma activity. Ribonucleoside analogues with modifications in nucleobase and sugar moieties

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 1. Synthesis and 31P NMR analysis of 16 diribonulceoside (3'-5')-H-phosphonates and the corresponding phosphorothioates

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 5. The role of Brønsted and H-bonding base catalysis in ribonucleoside H-phosphonate condensation-chemical and stereochemical consequences

Stereochemistry of internucleotide bond formation by the H-phosphonate method. 7. Stereoselective formation of ribonucleoside (RP)- and (SP)-3′-H-phosphonothioate monoesters

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 3: Investigations on a mechanism of asymmetric induction

Stereochemistry of internucleotide bond formation by the H-phosphonate method. Part 6: Optimization of the reaction conditions towards highest stereoselectivity

Studies on Aryl H-Phosphonates. Synthesis of Nucleoside N-Alkylphosphonamidates

Studies on Reactions of Nucleoside H-Phosphonates with Bifunctional Reagents. Part III. Further Studies on Transesterification of Nucleoside H-Phosphonate Diesters with Amino Alcohols

Studies on aryl H-phosphonates. 3. Mechanistic investigations related to the disproportionation of diphenyl H-phosphonate under anhydrous basic conditions

Studies on aryl H-phosphonates. I. An efficient method for the preparation of deoxyribo- and ribonucleoside 3′-H-phosphonate monoesters by transesterification of diphenyl H-phosphonate

Studies on reactions of nucleoside H-phosphonate diesters with bifunctional reagents. Part 4. Chemoselectivity during oxidative coupling of nucleoside H-phosphonate diesters with amino alcohols controlled by protonation of the amino function

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 1. Reaction with amino alcohols

Studies on reactions of nucleoside H-phosphonates with bifunctional reagents. Part 2. Stability of nucleoside H-phosphonate diesters in the presence of amino alcohols

Studies on the decomposition pathways of diastereoisomeric mixtures of aryl nucleoside α-hydroxyphosphonates under hydrolytic conditions. Synthesis of α-hydroxyphosphonate monoesters

The case of sulfonation in the chemical synthesis of oligonucleotides ⬇️

The case of triethylammonium cation loss during purification of certain nucleotide analogues: a cautionary note

The role of nucleophilic catalysis in chemistry and stereochemistry of ribonucleosideH-phosphonate condensation

Unusual Stereochemistry of Esterification of Uridine 3′-H-Phosphonothioate