List of works - O D Mitkin

2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: new series of highly potent and specific serotonin 5-HT6 receptor antagonists

scientific article published on 01 February 2011

8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists.

scientific article

AVN-492, A Novel Highly Selective 5-HT6R Antagonist: Preclinical Evaluation

scientific article published on 25 May 2017

Antagonists of 5-HT₆ receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines-Synthesis and 'structure-activity' relationship

scientific article published on 17 May 2012

Conical intersection control of heterocyclic photochemical bond scission.

scientific article published in October 2006

Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists.

scientific article published on 2 June 2015

Discovery of novel highly potent hepatitis C virus NS5A inhibitor (AV4025).

scientific article

Dithiane- and trithiane-based photolabile scaffolds for molecular recognition

scientific article published on 01 June 2001

From anti-allergic to anti-Alzheimer's: Molecular pharmacology of Dimebon.

scientific article

Novel oral anti-influenza drug candidate AV5080.

scientific article published on 11 April 2014

Novel oral anti-influenza prodrug candidate AV5075S.

scientific article published on 15 January 2014

Preclinical Development of ONC1-13B, Novel Antiandrogen for Prostate Cancer Treatment

scientific article

Solution phase parallel synthesis of substituted 3-phenylsulfonyl-[1,2,3]triazolo[1,5-a]quinazolines: selective serotonin 5-HT(6) receptor antagonists.

scientific article

Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists.

scientific article published on 5 January 2011

Synthesis and biological evaluation of novel gamma-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists

scientific article (publication date: 15 June 2009)

Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists.

scientific article published on 24 May 2010

Synthesis and structure-activity relationship (SAR) of (5,7-disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as potent serotonin 5-HT(6) receptor (5-HT(6)R) antagonists.

scientific article published on 10 November 2011

Synthesis of substituted diphenyl sulfones and their structure-activity relationship with the antagonism of 5-НТ6 receptors.

scientific article published in June 2013

The aza-type-B photochemical rearrangement: the role of a second carbonyl in heterocyclic photochemistry. Mechanistic and exploratory organic photochemistry

scientific article published on 29 June 2007

List of works by O D Mitkin

2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: new series of highly potent and specific serotonin 5-HT6 receptor antagonists

8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists.

AVN-492, A Novel Highly Selective 5-HT6R Antagonist: Preclinical Evaluation

Antagonists of 5-HT₆ receptors. Substituted 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines-Synthesis and 'structure-activity' relationship

Conical intersection control of heterocyclic photochemical bond scission.

Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists.

Discovery of novel highly potent hepatitis C virus NS5A inhibitor (AV4025).

Dithiane- and trithiane-based photolabile scaffolds for molecular recognition

From anti-allergic to anti-Alzheimer's: Molecular pharmacology of Dimebon.

Novel oral anti-influenza drug candidate AV5080.

Novel oral anti-influenza prodrug candidate AV5075S.

Preclinical Development of ONC1-13B, Novel Antiandrogen for Prostate Cancer Treatment

Solution phase parallel synthesis of substituted 3-phenylsulfonyl-[1,2,3]triazolo[1,5-a]quinazolines: selective serotonin 5-HT(6) receptor antagonists.

Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists.

Synthesis and biological evaluation of novel gamma-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists

Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists.

Synthesis and structure-activity relationship (SAR) of (5,7-disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as potent serotonin 5-HT(6) receptor (5-HT(6)R) antagonists.

Synthesis of substituted diphenyl sulfones and their structure-activity relationship with the antagonism of 5-НТ6 receptors.

The aza-type-B photochemical rearrangement: the role of a second carbonyl in heterocyclic photochemistry. Mechanistic and exploratory organic photochemistry