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List of works by T Scior

11-Keto-β-Boswellic Acids Prevent Development of Autoimmune Reactions, Insulitis and Reduce Hyperglycemia During Induction of Multiple Low-Dose Streptozotocin (MLD-STZ) Diabetes in Mice

scientific article published on 07 May 2015

A residue W756 in the P-loop segment of the sodium channel is critical for primaquine binding.

scientific article published on 27 April 2011

Antiprotozoal Nitazoxanide Derivatives: Synthesis, Bioassays and QSAR Study Combined with Docking for Mechanistic Insight.

scientific article

Application of drug repositioning strategy to TOFISOPAM.

scientific article

Are vanadium compounds drugable? Structures and effects of antidiabetic vanadium compounds: a critical review.

scientific article

Characterization of specific allosteric effects of the Na+ channel β1 subunit on the Nav1.4 isoform

scientific article published on 23 December 2016

Chemometric Models of Differential Amino Acids at the Navα and Navβ Interface of Mammalian Sodium Channel Isoforms

scientific article published on 03 August 2020

Chimeric design, synthesis, and biological assays of a new nonpeptide insulin-mimetic vanadium compound to inhibit protein tyrosine phosphatase 1B

scientific article published on September 24, 2010

Computational Binding Study Hints at Ecdysone 20-Mono-Oxygenase as the Hitherto Unknown Target for Ring C-Seco Limonoid-Type Insecticides

scientific article published in 2024

Elucidation of the fragmentation pathways of different phosphatidylinositol phosphate species (PIPx) using IRMPD implemented on a FT-ICR MS.

scientific article published on 3 October 2010

Ethnopharmacology and bioinformatic combination for leads discovery: application to phospholipase A2 inhibitors

scientific article published on November 1, 2001

Exploring electrostatic patterns of human, murine, equine and canine TLR4/MD-2 receptors

scientific article published on 25 December 2019

Five Novel Non-Sialic Acid-Like Scaffolds Inhibit In Vitro H1N1 and H5N2 Neuraminidase Activity of Influenza a Virus

scientific article published on 16 September 2020

How to Valorize Biodiversity? Let's Go Hashing, Extracting, Filtering, Mining, Fishing.

scientific article published on 25 February 2015

How to recognize and workaround pitfalls in QSAR studies: a critical review

scientific article published on January 2009

Identification of Navβ1 residues involved in the modulation of the sodium channel Nav1.4.

scientific article

Integrating computational and mixture-based screening of combinatorial libraries.

scientific article

Interference of boswellic acids with the ligand binding domain of the glucocorticoid receptor

scientific article published on 20 February 2014

Isoniazid is not a lead compound for its pyridyl ring derivatives, isonicotinoyl amides, hydrazides, and hydrazones: a critical review.

scientific article published on January 2006

Large compound databases for structure-activity relationships studies in drug discovery.

scientific article

Mefloquine inhibits voltage dependent Nav1.4 channel by overlapping the local anaesthetic binding site.

scientific article published on 2 January 2017

Modulating testosterone pathway: a new strategy to tackle male skin aging?

scientific article published on 13 September 2012

Pharmacophore design of p38α MAP kinase inhibitors with either 2,4,5-trisubstituted or 1,2,4,5-tetrasubstituted imidazole scaffold.

scientific article published on January 2011

Predicting a double mutant in the twilight zone of low homology modeling for the skeletal muscle voltage-gated sodium channel subunit beta-1 (Nav1.4 β1).

scientific article

Prolyl isomerases in a minimal cell. Catalysis of protein folding by trigger factor from Mycoplasma genitalium.

scientific article

Reverse pharmacognosy: another way to harness the generosity of nature

scientific article published on May 2010

Reviewing and identifying amino acids of human, murine, canine and equine TLR4 / MD-2 receptor complexes conferring endotoxic innate immunity activation by LPS/lipid A, or antagonistic effects by Eritoran, in contrast to species-dependent modulation

scientific article published on 05 April 2013

Synthesis and biological testing of purine derivatives as potential ATP-competitive kinase inhibitors.

scientific article published in February 2005

Synthesis, biological testing, and binding mode prediction of 6,9-diarylpurin-8-ones as p38 MAP kinase inhibitors

scientific article published on 06 April 2007

Three-dimensional mapping of differential amino acids of human, murine, canine and equine TLR4/MD-2 receptor complexes conferring endotoxic activation by lipid A, antagonism by Eritoran and species-dependent activities of Lipid IVA in the mammalian L

scientific article published on 08 August 2013

Why Antidiabetic Vanadium Complexes are Not in the Pipeline of "Big Pharma" Drug Research? A Critical Review

scientific article