Search filters

List of works by Erik A A Wallén

2(S)-(Cycloalk-1-enecarbonyl)-1-(4-phenyl-butanoyl)pyrrolidines and 2(S)-(aroyl)-1-(4-phenylbutanoyl)pyrrolidines as prolyl oligopeptidase inhibitors

scientific article

4-Phenylbutanoyl-2(S)-acylpyrrolidines and 4-phenylbutanoyl-L-prolyl-2(S)-acylpyrrolidines as prolyl oligopeptidase inhibitors.

scientific article published in July 2002

An introduction of a pyridine group into the structure of prolyl oligopeptidase inhibitors

scientific article published on 17 August 2006

Azulene-based compounds for targeting orexin receptors

scientific article published on 20 July 2018

Beneficial effect of prolyl oligopeptidase inhibition on spatial memory in young but not in old scopolamine-treated rats

scientific article

Binding kinetics and duration of in vivo action of novel prolyl oligopeptidase inhibitors.

scientific article

Characterization of the binding properties of SIRT2 inhibitors with a N-(3-phenylpropenoyl)-glycine tryptamide backbone.

scientific article published on 24 July 2008

Chroman-4-one and chromone based somatostatin β-turn mimetics.

scientific article

Chroman-4-one- and chromone-based sirtuin 2 inhibitors with antiproliferative properties in cancer cells.

scientific article

Conformationally rigid N-acyl-5-alkyl-L-prolyl-pyrrolidines as prolyl oligopeptidase inhibitors.

scientific article published in August 2003

Development of molecules stimulating the activity of KLK3 - an update.

scientific article

Dicarboxylic acid azacycle l-prolyl-pyrrolidine amides as prolyl oligopeptidase inhibitors and three-dimensional quantitative structure-activity relationship of the enzyme-inhibitor interactions.

scientific article published in July 2005

Dicarboxylic acid bis(L-prolyl-pyrrolidine) amides as prolyl oligopeptidase inhibitors.

scientific article published in September 2002

Mimetics of the disulfide bridge between the N- and C-terminal cysteines of the KLK3-stimulating peptide B-2.

scientific article published on 5 December 2009

N(epsilon)-thioacetyl-lysine-containing tri-, tetra-, and pentapeptides as SIRT1 and SIRT2 inhibitors.

scientific article

N,N'-Bisbenzylidenebenzene-1,4-diamines and N,N'-Bisbenzylidenenaphthalene-1,4-diamines as Sirtuin Type 2 (SIRT2) Inhibitors

scientific article published on 01 December 2006

N-(3-(4-Hydroxyphenyl)-propenoyl)-amino acid tryptamides as SIRT2 inhibitors

scientific article published on 13 February 2007

New Prolyl Oligopeptidase Inhibitors Developed from Dicarboxylic Acid Bis(l-prolyl-pyrrolidine) Amides ⬇️

scientific article published on October 9, 2003

Oxadiazole-carbonylaminothioureas as SIRT1 and SIRT2 inhibitors.

scientific article published on 22 July 2008

Pharmacological characterization of the orexin/hypocretin receptor agonist Nag 26

scientific article published on 05 September 2018

Replacement of the Disulfide Bridge in a KLK3-Stimulating Peptide Using Orthogonally Protected Building Blocks.

scientific article published on 16 December 2013

Structure-Activity Relationships of 1-Benzoylazulenes at the OX1 and OX2 Orexin Receptors

scientific article published on 02 April 2019

Substrate-dependent, non-hyperbolic kinetics of pig brain prolyl oligopeptidase and its tight binding inhibition by JTP-4819.

scientific article published in August 2002

Synthesis and biological evaluation of novel 123I-labeled 4-(4-iodophenyl)butanoyl-l-prolyl-(2S)-pyrrolidines for imaging prolyl oligopeptidase in vivo

scientific article published on 12 April 2014

Synthesis of 1,3,6-Trisubstituted Azulenes

scientific article published on 11 November 2015

Synthesis of 2,3,6,8-tetrasubstituted chromone scaffolds

scientific article published on 01 September 2006

Synthesis of 3-aminomethyl-2-aryl- 8-bromo-6-chlorochromones

scientific article published on 01 February 2007

Synthesis of orthogonally protected disulfide bridge mimetics

scientific article published on 22 December 2010

Paulina is supported by:

About Paulina

Help